Chemical synthesis of peptides within the insulin superfamily
Liu, Fa, Zaykov, Alexander N., Levy, Jay J., DiMarchi, Richard D., Mayer, John P.
Published in Journal of peptide science (01.05.2016)
Published in Journal of peptide science (01.05.2016)
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Journal Article
Chemical Synthesis of Human Insulin-Like Peptide-6
Wu, Fangzhou, Mayer, John P., Zaykov, Alexander N., Zhang, Fa, Liu, Fa, DiMarchi, Richard D.
Published in Chemistry : a European journal (04.07.2016)
Published in Chemistry : a European journal (04.07.2016)
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Journal Article
Chemical Synthesis of Insulin Analogs through a Novel Precursor
Zaykov, Alexander N, Mayer, John P, Gelfanov, Vasily M, DiMarchi, Richard D
Published in ACS chemical biology (21.03.2014)
Published in ACS chemical biology (21.03.2014)
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Journal Article
A long-acting LEAP2 analog reduces hepatic steatosis and inflammation and causes marked weight loss in mice
Shankar, Kripa, Metzger, Nathan P., Lawrence, Connor, Gupta, Deepali, Osborne-Lawrence, Sherri, Varshney, Salil, Singh, Omprakash, Richard, Corine P., Zaykov, Alexander N., Rolfts, Rebecca, DuBois, Barent N., Perez-Tilve, Diego, Mani, Bharath K., Hammer, Suntrea T.G., Zigman, Jeffrey M.
Published in Molecular metabolism (Germany) (01.06.2024)
Published in Molecular metabolism (Germany) (01.06.2024)
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Journal Article
Peptide Model of the Mutant Proinsulin Syndrome. II. Nascent Structure and Biological Implications
Yang, Yanwu, Glidden, Michael D, Dhayalan, Balamurugan, Zaykov, Alexander N, Chen, Yen-Shan, Wickramasinghe, Nalinda P, DiMarchi, Richard D, Weiss, Michael A
Published in Frontiers in endocrinology (Lausanne) (01.03.2022)
Published in Frontiers in endocrinology (Lausanne) (01.03.2022)
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Journal Article
Peptide Model of the Mutant Proinsulin Syndrome. I. Design and Clinical Correlation
Dhayalan, Balamurugan, Glidden, Michael D, Zaykov, Alexander N, Chen, Yen-Shan, Yang, Yanwu, Phillips, Nelson B, Ismail-Beigi, Faramarz, Jarosinski, Mark A, DiMarchi, Richard D, Weiss, Michael A
Published in Frontiers in endocrinology (Lausanne) (01.03.2022)
Published in Frontiers in endocrinology (Lausanne) (01.03.2022)
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Journal Article
Pursuit of a perfect insulin
Zaykov, Alexander N, Mayer, John P, DiMarchi, Richard D
Published in Nature reviews. Drug discovery (01.06.2016)
Published in Nature reviews. Drug discovery (01.06.2016)
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Journal Article
Synthesis of relaxin‐2 and insulin‐like peptide 5 enabled by novel tethering and traceless chemical excision
Thalluri, Kishore, Kou, Binbin, Yang, Xu, Zaykov, Alexander N., Mayer, John P., Gelfanov, Vasily M., Liu, Fa, DiMarchi, Richard D.
Published in Journal of peptide science (01.06.2017)
Published in Journal of peptide science (01.06.2017)
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Journal Article
High-Yield Synthesis of Human Insulin-Like Peptide 5 Employing a Nonconventional Strategy
Zaykov, Alexander N, Gelfanov, Vasily M, Liu, Fa, DiMarchi, Richard D
Published in Organic letters (15.06.2018)
Published in Organic letters (15.06.2018)
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Journal Article
A Disulfide Scan of Insulin by [3 + 1] Methodology Exhibits Site-Specific Influence on Bioactivity
Brunel, Florence M, Mayer, John P, Gelfanov, Vasily M, Zaykov, Alexander N, Finan, Brian, Perez-Tilve, Diego, DiMarchi, Richard D
Published in ACS chemical biology (16.08.2019)
Published in ACS chemical biology (16.08.2019)
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Journal Article
Synthesis and Characterization of the R27S Genetic Variant of Insulin‐like Peptide 5
Zaykov, Alexander N., Gelfanov, Vasily M., Liu, Fa, DiMarchi, Richard D.
Published in ChemMedChem (23.04.2018)
Published in ChemMedChem (23.04.2018)
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Journal Article
A general synthesis of dirhodium metallopeptides as MDM2 ligands
Zaykov, Alexander N, Ball, Zachary T
Published in Chemical communications (Cambridge, England) (21.10.2011)
Published in Chemical communications (Cambridge, England) (21.10.2011)
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Journal Article
Toward once-monthly insulin therapy via synergy in two pharmacokinetic protractors: Fc-conjugation and fatty acid acylation
Zaykov, Alexander N., Gelfanov, Vasily M., Tagmose, Tina M., Demozay, Damien, Manfè, Valentina, Rohlfs, Rebecca, Rivir, Marita, Perez-Tilve, Diego, Finan, Brian, DiMarchi, Richard D.
Published in RSC chemical biology (31.07.2024)
Published in RSC chemical biology (31.07.2024)
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Journal Article
ChemInform Abstract: Chemical Synthesis of Peptides within the Insulin Superfamily
Liu, Fa, Zaykov, Alexander N., Levy, Jay J., Di Marchi, Richard D., Mayer, John P.
Published in ChemInform (01.06.2016)
Published in ChemInform (01.06.2016)
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Journal Article