Immunoproteasome-selective and non-selective inhibitors: A promising approach for the treatment of multiple myeloma
Ettari, Roberta, Zappalà, Maria, Grasso, Silvana, Musolino, Caterina, Innao, Vanessa, Allegra, Alessandro
Published in Pharmacology & therapeutics (Oxford) (01.02.2018)
Published in Pharmacology & therapeutics (Oxford) (01.02.2018)
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Journal Article
Lead Discovery of SARS-CoV‑2 Main Protease Inhibitors through Covalent Docking-Based Virtual Screening
Amendola, Giorgio, Ettari, Roberta, Previti, Santo, Di Chio, Carla, Messere, Anna, Di Maro, Salvatore, Hammerschmidt, Stefan J, Zimmer, Collin, Zimmermann, Robert A, Schirmeister, Tanja, Zappalà, Maria, Cosconati, Sandro
Published in Journal of chemical information and modeling (26.04.2021)
Published in Journal of chemical information and modeling (26.04.2021)
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Journal Article
Optimization Strategy of Novel Peptide-Based Michael Acceptors for the Treatment of Human African Trypanosomiasis
Ettari, Roberta, Previti, Santo, Maiorana, Santina, Amendola, Giorgio, Wagner, Annika, Cosconati, Sandro, Schirmeister, Tanja, Hellmich, Ute A, Zappalà, Maria
Published in Journal of medicinal chemistry (12.12.2019)
Published in Journal of medicinal chemistry (12.12.2019)
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Journal Article
Dihydrochalcones as antitumor agents
De Luca, Fabiola, Di Chio, Carla, Zappalà, Maria, Ettari, Roberta
Published in Current medicinal chemistry (01.09.2022)
Published in Current medicinal chemistry (01.09.2022)
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Journal Article
Drug Combination Studies of Isoquinolinone AM12 with Curcumin or Quercetin: A New Combination Strategy to Synergistically Inhibit 20S Proteasome
Di Chio, Carla, Previti, Santo, Starvaggi, Josè, De Luca, Fabiola, Calabrò, Maria Luisa, Zappalà, Maria, Ettari, Roberta
Published in International journal of molecular sciences (01.10.2024)
Published in International journal of molecular sciences (01.10.2024)
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Journal Article
Immunoproteasome-Selective Inhibitors: A Promising Strategy to Treat Hematologic Malignancies, Autoimmune and Inflammatory Diseases
Ettari, Roberta, Previti, Santo, Bitto, Alessandra, Grasso, Silvana, Zappalà, Maria
Published in Current medicinal chemistry (01.01.2016)
Published in Current medicinal chemistry (01.01.2016)
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Journal Article
Development of Novel Peptide-Based Michael Acceptors Targeting Rhodesain and Falcipain‑2 for the Treatment of Neglected Tropical Diseases (NTDs)
Previti, Santo, Ettari, Roberta, Cosconati, Sandro, Amendola, Giorgio, Chouchene, Khawla, Wagner, Annika, Hellmich, Ute A, Ulrich, Kathrin, Krauth-Siegel, R. Luise, Wich, Peter R, Schmid, Ira, Schirmeister, Tanja, Gut, Jiri, Rosenthal, Philip J, Grasso, Silvana, Zappalà, Maria
Published in Journal of medicinal chemistry (24.08.2017)
Published in Journal of medicinal chemistry (24.08.2017)
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Journal Article
Blunting Neuroinflammation by Targeting the Immunoproteasome with Novel Amide Derivatives
Imbesi, Chiara, Ettari, Roberta, Irrera, Natasha, Zappalà, Maria, Pallio, Giovanni, Bitto, Alessandra, Mannino, Federica
Published in International journal of molecular sciences (27.06.2023)
Published in International journal of molecular sciences (27.06.2023)
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Journal Article
Development of novel dipeptide nitriles as inhibitors of rhodesain of Trypanosoma brucei rhodesiense
Di Chio, Carla, Previti, Santo, Amendola, Giorgio, Ravichandran, Rahul, Wagner, Annika, Cosconati, Sandro, Hellmich, Ute A., Schirmeister, Tanja, Zappalà, Maria, Ettari, Roberta
Published in European journal of medicinal chemistry (05.06.2022)
Published in European journal of medicinal chemistry (05.06.2022)
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Journal Article
Dipeptide Nitrile CD34 with Curcumin: A New Improved Combination Strategy to Synergistically Inhibit Rhodesain of Trypanosoma brucei rhodesiense
Di Chio, Carla, Previti, Santo, Totaro, Noemi, De Luca, Fabiola, Allegra, Alessandro, Schirmeister, Tanja, Zappalà, Maria, Ettari, Roberta
Published in International journal of molecular sciences (09.05.2023)
Published in International journal of molecular sciences (09.05.2023)
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Journal Article
The Inhibition of Cysteine Proteases Rhodesain and TbCatB: A Valuable Approach to Treat Human African Trypanosomiasis
Ettari, Roberta, Previti, Santo, Tamborini, Lucia, Cullia, Gregorio, Grasso, Silvana, Zappalà, Maria
Published in Mini reviews in medicinal chemistry (01.01.2016)
Published in Mini reviews in medicinal chemistry (01.01.2016)
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Journal Article
Virtual Screening Strategy and In Vitro Tests to Identify New Inhibitors of the Immunoproteasome
Culletta, Giulia, Tutone, Marco, Ettari, Roberta, Perricone, Ugo, Di Chio, Carla, Almerico, Anna Maria, Zappalà, Maria
Published in International journal of molecular sciences (22.06.2023)
Published in International journal of molecular sciences (22.06.2023)
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Journal Article
Development of isoquinolinone derivatives as immunoproteasome inhibitors
Ettari, Roberta, Iraci, Nunzio, Di Chio, Carla, Previti, Santo, Danzè, Mariafernanda, Zappalà, Maria
Published in Bioorganic & medicinal chemistry letters (01.01.2022)
Published in Bioorganic & medicinal chemistry letters (01.01.2022)
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Journal Article