Synthesis and SAR studies of novel 2-(6-aminomethylaryl-2-aryl-4-oxo-quinazolin-3(4H)-yl)acetamide Vasopressin V₁b receptor antagonists
Napier, Susan E, Letourneau, Jeffrey J, Ansari, Nasrin, Auld, Douglas S, Baker, James, Best, Stuart, Campbell-Wan, Leigh, Chan, Ray, Craighead, Mark, Desai, Hema, Ho, Koc-Kan, MacSweeney, Cliona, Milne, Rachel, Richard Morphy, J, Neagu, Irina, Ohlmeyer, Michael H.J, Pick, Jack, Presland, Jeremy, Riviello, Chris, Zanetakos, Heather A, Zhao, Jiuqiao, Webb, Maria L
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
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Journal Article
Synthesis and SAR studies of novel 2-(4-oxo-2-aryl-quinazolin-3(4H)-yl)acetamide vasopressin V₁b receptor antagonists
Napier, Susan E, Letourneau, Jeffrey J, Ansari, Nasrin, Auld, Douglas S, Baker, James, Best, Stuart, Campbell-Wan, Leigh, Chan, Jui-Hsiang, Craighead, Mark, Desai, Hema, Goan, Katharine A, Ho, Koc-Kan, Hulskotte, Ellen G.J, MacSweeney, Cliona P, Milne, Rachel, Morphy, J. Richard, Neagu, Irina, Ohlmeyer, Michael H.J, Peeters, Ard W.M.M, Presland, Jeremy, Riviello, Chris, Ruigt, Ge S.F, Thomson, Fiona J, Zanetakos, Heather A, Zhao, Jiuqiao, Webb, Maria L
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
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Journal Article
Identification and optimization of novel 2-(4-oxo-2-aryl-quinazolin-3(4 H)-yl)acetamide vasopressin V3 (V1b) receptor antagonists
Letourneau, Jeffrey J., Riviello, Christopher M., Li, Hong, Cole, Andrew G., Ho, Koc-Kan, Zanetakos, Heather A., Desai, Hema, Zhao, Jiuqiao, Auld, Douglas S., Napier, Susan E., Thomson, Fiona J., Goan, Katharine A., Morphy, J. Richard, Ohlmeyer, Michael H.J., Webb, Maria L.
Published in Bioorganic & medicinal chemistry letters (15.09.2010)
Published in Bioorganic & medicinal chemistry letters (15.09.2010)
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Journal Article
Synthesis and SAR studies of novel 2-(6-aminomethylaryl-2-aryl-4-oxo-quinazolin-3(4 H)-yl)acetamide Vasopressin V 1b receptor antagonists
Napier, Susan E., Letourneau, Jeffrey J., Ansari, Nasrin, Auld, Douglas S., Baker, James, Best, Stuart, Campbell-Wan, Leigh, Chan, Ray, Craighead, Mark, Desai, Hema, Ho, Koc-Kan, MacSweeney, Cliona, Milne, Rachel, Richard Morphy, J., Neagu, Irina, Ohlmeyer, Michael H.J., Pick, Jack, Presland, Jeremy, Riviello, Chris, Zanetakos, Heather A., Zhao, Jiuqiao, Webb, Maria L.
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Get full text
Journal Article
Synthesis and SAR studies of novel 2-(4-oxo-2-aryl-quinazolin-3(4 H)-yl)acetamide vasopressin V 1b receptor antagonists
Napier, Susan E., Letourneau, Jeffrey J., Ansari, Nasrin, Auld, Douglas S., Baker, James, Best, Stuart, Campbell-Wan, Leigh, Chan, Jui-Hsiang, Craighead, Mark, Desai, Hema, Goan, Katharine A., Ho, Koc-Kan, Hulskotte, Ellen G.J., MacSweeney, Cliona P., Milne, Rachel, Morphy, J. Richard, Neagu, Irina, Ohlmeyer, Michael H.J., Peeters, Ard W.M.M., Presland, Jeremy, Riviello, Chris, Ruigt, Ge S.F., Thomson, Fiona J., Zanetakos, Heather A., Zhao, Jiuqiao, Webb, Maria L.
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
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Journal Article
Synthesis and SAR studies of novel 2-(6-aminomethylaryl-2-aryl-4-oxo-quinazolin-3(4H)-yl)acetamide Vasopressin V sub(1b receptor antagonists)
Napier, Susan E, Letourneau, Jeffrey J, Ansari, Nasrin, Auld, Douglas S, Baker, James, Best, Stuart, Campbell-Wan, Leigh, Chan, Ray, Craighead, Mark, Desai, Hema, Ho, Koc-Kan, MacSweeney, Cliona, Milne, Rachel, Morphy, JRichard, Neagu, Irina, Ohlmeyer, Michael HJ, Pick, Jack, Presland, Jeremy, Riviello, Chris, Zanetakos, Heather A, Zhao, Jiuqiao, Webb, Maria L
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Published in Bioorganic & medicinal chemistry letters (15.06.2011)
Get full text
Journal Article
Synthesis and SAR studies of novel 2-(4-oxo-2-aryl-quinazolin-3(4H)-yl)acetamide vasopressin V sub(1b receptor antagonists)
Napier, Susan E, Letourneau, Jeffrey J, Ansari, Nasrin, Auld, Douglas S, Baker, James, Best, Stuart, Campbell-Wan, Leigh, Chan, Jui-Hsiang, Craighead, Mark, Desai, Hema, Goan, Katharine A, Ho, Koc-Kan, Hulskotte, Ellen GJ, MacSweeney, Cliona P, Milne, Rachel, Morphy, JRichard, Neagu, Irina, Ohlmeyer, Michael HJ, Peeters, Ard WMM, Presland, Jeremy, Riviello, Chris, Ruigt, Ge SF, Thomson, Fiona J, Zanetakos, Heather A, Zhao, Jiuqiao, Webb, Maria L
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
Published in Bioorganic & medicinal chemistry letters (15.03.2011)
Get full text
Journal Article