Synthesis and Antiviral Activity of Novel 1,3,4-Thiadiazole Inhibitors of DDX3X
Brai, Annalaura, Ronzini, Stefania, Riva, Valentina, Botta, Lorenzo, Zamperini, Claudio, Borgini, Matteo, Trivisani, Claudia Immacolata, Garbelli, Anna, Pennisi, Carla, Boccuto, Adele, Saladini, Francesco, Zazzi, Maurizio, Maga, Giovanni, Botta, Maurizio
Published in Molecules (Basel, Switzerland) (04.11.2019)
Published in Molecules (Basel, Switzerland) (04.11.2019)
Get full text
Journal Article
Rhodanine derivatives as potent anti-HIV and anti-HSV microbicides
Tintori, Cristina, Iovenitti, Giulia, Ceresola, Elisa Rita, Ferrarese, Roberto, Zamperini, Claudio, Brai, Annalaura, Poli, Giulio, Dreassi, Elena, Cagno, Valeria, Lembo, David, Canducci, Filippo, Botta, Maurizio
Published in PloS one (05.06.2018)
Published in PloS one (05.06.2018)
Get full text
Journal Article
Design, Synthesis, Biological Activity, and ADME Properties of Pyrazolo[3,4-d]pyrimidines Active in Hypoxic Human Leukemia Cells: A Lead Optimization Study
Radi, Marco, Dreassi, Elena, Brullo, Chiara, Crespan, Emmanuele, Tintori, Cristina, Bernardo, Vincenzo, Valoti, Massimo, Zamperini, Claudio, Daigl, Henry, Musumeci, Francesca, Carraro, Fabio, Naldini, Antonella, Filippi, Irene, Maga, Giovanni, Schenone, Silvia, Botta, Maurizio
Published in Journal of medicinal chemistry (28.04.2011)
Published in Journal of medicinal chemistry (28.04.2011)
Get full text
Journal Article
Indolylarylsulfones Carrying a Heterocyclic Tail as Very Potent and Broad Spectrum HIV‑1 Non-nucleoside Reverse Transcriptase Inhibitors
Famiglini, Valeria, La Regina, Giuseppe, Coluccia, Antonio, Pelliccia, Sveva, Brancale, Andrea, Maga, Giovanni, Crespan, Emmanuele, Badia, Roger, Riveira-Muñoz, Eva, Esté, José A, Ferretti, Rosella, Cirilli, Roberto, Zamperini, Claudio, Botta, Maurizio, Schols, Dominique, Limongelli, Vittorio, Agostino, Bruno, Novellino, Ettore, Silvestri, Romano
Published in Journal of medicinal chemistry (11.12.2014)
Published in Journal of medicinal chemistry (11.12.2014)
Get full text
Journal Article
A New Strategy for Glioblastoma Treatment: In Vitro and In Vivo Preclinical Characterization of Si306, a Pyrazolo[3,4- d ]Pyrimidine Dual Src/P-Glycoprotein Inhibitor
Fallacara, Anna Lucia, Zamperini, Claudio, Podolski-Renić, Ana, Dinić, Jelena, Stanković, Tijana, Stepanović, Marija, Mancini, Arianna, Rango, Enrico, Iovenitti, Giulia, Molinari, Alessio, Bugli, Francesca, Sanguinetti, Maurizio, Torelli, Riccardo, Martini, Maurizio, Maccari, Laura, Valoti, Massimo, Dreassi, Elena, Botta, Maurizio, Pešić, Milica, Schenone, Silvia
Published in Cancers (01.06.2019)
Published in Cancers (01.06.2019)
Get full text
Journal Article
Noncanonical-NF-κB activation and DDX3 inhibition reduces the HIV-1 reservoir by elimination of latently infected cells ex-vivo
Jansen, Jade, Kroeze, Stefanie, Man, Shirley, Andreini, Matteo, Bakker, Jan-Willem, Zamperini, Claudio, Tarditi, Alessia, Kootstra, Neeltje A, Geijtenbeek, Teunis B H
Published in Microbiology spectrum (11.01.2024)
Published in Microbiology spectrum (11.01.2024)
Get full text
Journal Article
Development and in Vitro Evaluation of a Microbicide Gel Formulation for a Novel Non-Nucleoside Reverse Transcriptase Inhibitor Belonging to the N-Dihydroalkyloxybenzyloxopyrimidines (N-DABOs) Family
Tintori, Cristina, Brai, Annalaura, Lang, Maria Chiara Dasso, Deodato, Davide, Greco, Antonia Michela, Bizzarri, Bruno Mattia, Cascone, Lorena, Casian, Alexandru, Zarriperini, Claudio, Dreassi, Elena, Crespan, Emmanuele, Maga, Giovanni, Vanham, Guido, Ceresola, Elisa, Canducci, Filippo, Arien, Kevin K., Botta, Maurizio
Published in Journal of medicinal chemistry (24.03.2016)
Published in Journal of medicinal chemistry (24.03.2016)
Get full text
Journal Article
Targeting DDX3X Helicase Activity with BA103 Shows Promising Therapeutic Effects in Preclinical Glioblastoma Models
Brai, Annalaura, Riva, Valentina, Clementi, Letizia, Falsitta, Lucia, Zamperini, Claudio, Sinigiani, Virginia, Festuccia, Claudio, Sabetta, Samantha, Aiello, Davide, Roselli, Camilla, Garbelli, Anna, Trivisani, Claudia Immacolata, Maccari, Laura, Bugli, Francesca, Sanguinetti, Maurizio, Calandro, Pierpaolo, Chiariello, Mario, Quaranta, Paola, Botta, Lorenzo, Angelucci, Adriano, Maga, Giovanni, Botta, Maurizio
Published in Cancers (07.11.2021)
Published in Cancers (07.11.2021)
Get full text
Journal Article
Identification of potent c-Src inhibitors strongly affecting the proliferation of human neuroblastoma cells
Radi, Marco, Brullo, Chiara, Crespan, Emmanuele, Tintori, Cristina, Musumeci, Francesca, Biava, Mariangela, Schenone, Silvia, Dreassi, Elena, Zamperini, Claudio, Maga, Giovanni, Pagano, Dafne, Angelucci, Adriano, Bologna, Mauro, Botta, Maurizio
Published in Bioorganic & medicinal chemistry letters (01.10.2011)
Published in Bioorganic & medicinal chemistry letters (01.10.2011)
Get full text
Journal Article
The Pyrazolo[3,4- d ]Pyrimidine Derivative Si306 Encapsulated into Anti-GD2-Immunoliposomes as Therapeutic Treatment of Neuroblastoma
Rango, Enrico, Pastorino, Fabio, Brignole, Chiara, Mancini, Arianna, Poggialini, Federica, Di Maria, Salvatore, Zamperini, Claudio, Iovenitti, Giulia, Fallacara, Anna Lucia, Sabetta, Samantha, Clementi, Letizia, Valoti, Massimo, Schenone, Silvia, Angelucci, Adriano, Ponzoni, Mirco, Dreassi, Elena, Botta, Maurizio
Published in Biomedicines (12.03.2022)
Published in Biomedicines (12.03.2022)
Get full text
Journal Article
CYP-dependent Metabolism of Antitumor Pyrazolo[3,4-d]pyrimidine Derivatives Is Characterized by an Oxidative Dechlorination Reaction
Zamperini, Claudio, Dreassi, Elena, Vignaroli, Giulia, Radi, Marco, Dragoni, Stefania, Schenone, Silvia, Musumeci, Francesca, Valoti, Massimo, Antiochia, Riccarda, Botta, Maurizio
Published in DRUG METABOLISM AND PHARMACOKINETICS (2014)
Published in DRUG METABOLISM AND PHARMACOKINETICS (2014)
Get full text
Journal Article
A combined targeted/phenotypic approach for the identification of new antiangiogenics agents active on a zebrafish model: From in silico screening to cyclodextrin formulation
Radi, Marco, Evensen, Lasse, Dreassi, Elena, Zamperini, Claudio, Caporicci, Marialessandra, Falchi, Federico, Musumeci, Francesca, Schenone, Silvia, Lorens, James B., Botta, Maurizio
Published in Bioorganic & medicinal chemistry letters (01.09.2012)
Published in Bioorganic & medicinal chemistry letters (01.09.2012)
Get full text
Journal Article
DDX3X Helicase Inhibitors as a New Strategy To Fight the West Nile Virus Infection
Brai, Annalaura, Martelli, Francesco, Riva, Valentina, Garbelli, Anna, Fazi, Roberta, Zamperini, Claudio, Pollutri, Alessandro, Falsitta, Lucia, Ronzini, Stefania, Maccari, Laura, Maga, Giovanni, Giannecchini, Simone, Botta, Maurizio
Published in Journal of medicinal chemistry (14.03.2019)
Published in Journal of medicinal chemistry (14.03.2019)
Get full text
Journal Article
DDX3X inhibitors, an effective way to overcome HIV-1 resistance targeting host proteins
Brai, Annalaura, Riva, Valentina, Saladini, Francesco, Zamperini, Claudio, Trivisani, Claudia Immacolata, Garbelli, Anna, Pennisi, Carla, Giannini, Alessia, Boccuto, Adele, Bugli, Francesca, Martini, Maurizio, Sanguinetti, Maurizio, Zazzi, Maurizio, Dreassi, Elena, Botta, Maurizio, Maga, Giovanni
Published in European journal of medicinal chemistry (15.08.2020)
Published in European journal of medicinal chemistry (15.08.2020)
Get full text
Journal Article
Human DDX3 protein is a valuable target to develop broad spectrum antiviral agents
Brai, Annalaura, Fazi, Roberta, Tintori, Cristina, Zamperini, Claudio, Bugli, Francesca, Sanguinetti, Maurizio, Stigliano, Egidio, Esté, José, Badia, Roger, Franco, Sandra, Martinez, Miguel A., Martinez, Javier P., Meyerhans, Andreas, Saladini, Francesco, Zazzi, Maurizio, Garbelli, Anna, Maga, Giovanni, Botta, Maurizio
Published in Proceedings of the National Academy of Sciences - PNAS (10.05.2016)
Published in Proceedings of the National Academy of Sciences - PNAS (10.05.2016)
Get full text
Journal Article
Efficient optimization of pyrazolo[3,4-d]pyrimidines derivatives as c-Src kinase inhibitors in neuroblastoma treatment
Molinari, Alessio, Fallacara, Anna Lucia, Di Maria, Salvatore, Zamperini, Claudio, Poggialini, Federica, Musumeci, Francesca, Schenone, Silvia, Angelucci, Adriano, Colapietro, Alessandro, Crespan, Emmanuele, Kissova, Miroslava, Maga, Giovanni, Botta, Maurizio
Published in Bioorganic & medicinal chemistry letters (15.11.2018)
Published in Bioorganic & medicinal chemistry letters (15.11.2018)
Get full text
Journal Article
Si113-prodrugs selectively activated by plasmin against hepatocellular and ovarian carcinoma
Rango, Enrico, D'Antona, Lucia, Iovenitti, Giulia, Brai, Annalaura, Mancini, Arianna, Zamperini, Claudio, Trivisani, Claudia Immacolata, Marianelli, Stefano, Fallacara, Anna Lucia, Molinari, Alessio, Cianciusi, Annarita, Schenone, Silvia, Perrotti, Nicola, Dreassi, Elena, Botta, Maurizio
Published in European journal of medicinal chemistry (05.11.2021)
Published in European journal of medicinal chemistry (05.11.2021)
Get full text
Journal Article
Abstract 2201: Preclinical development of novel pyrazolo[3,4- d ]pyrimidines structure-based TKIs for the treatment of glioblastoma
Mancini, Arianna, Fallacara, Anna Lucia, Zamperini, Claudio, Iovenitti, Giulia, Molinari, Alessio, Rango, Enrico, Angelucci, Adriano, Schenone, Silvia, Botta, Maurizio
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Published in Cancer research (Chicago, Ill.) (01.07.2019)
Get full text
Journal Article
Prodrugs of Pyrazolo[3,4‑d]pyrimidines: From Library Synthesis to Evaluation as Potential Anticancer Agents in an Orthotopic Glioblastoma Model
Vignaroli, Giulia, Iovenitti, Giulia, Zamperini, Claudio, Coniglio, Federica, Calandro, Pierpaolo, Molinari, Alessio, Fallacara, Anna Lucia, Sartucci, Andrea, Calgani, Alessia, Colecchia, David, Mancini, Andrea, Festuccia, Claudio, Dreassi, Elena, Valoti, Massimo, Musumeci, Francesca, Chiariello, Mario, Angelucci, Adriano, Botta, Maurizio, Schenone, Silvia
Published in Journal of medicinal chemistry (27.07.2017)
Published in Journal of medicinal chemistry (27.07.2017)
Get full text
Journal Article
Pyrazolo[3,4-d]pyrimidines-loaded human serum albumin (HSA) nanoparticles: Preparation, characterization and cytotoxicity evaluation against neuroblastoma cell line
Fallacara, Anna Lucia, Mancini, Arianna, Zamperini, Claudio, Dreassi, Elena, Marianelli, Stefano, Chiariello, Mario, Pozzi, Gianni, Santoro, Francesco, Botta, Maurizio, Schenone, Silvia
Published in Bioorganic & medicinal chemistry letters (15.07.2017)
Published in Bioorganic & medicinal chemistry letters (15.07.2017)
Get full text
Journal Article