A review of methods for solubility determination in biopharmaceutical drug characterization
Veseli, Ardita, Žakelj, Simon, Kristl, Albin
Published in Drug development and industrial pharmacy (02.11.2019)
Published in Drug development and industrial pharmacy (02.11.2019)
Get more information
Journal Article
Suitability of RPMI 2650 cell models for nasal drug permeability prediction
Sibinovska, Nadica, Žakelj, Simon, Kristan, Katja
Published in European journal of pharmaceutics and biopharmaceutics (01.12.2019)
Published in European journal of pharmaceutics and biopharmaceutics (01.12.2019)
Get full text
Journal Article
The Magic of Crystal Structure-Based Inhibitor Optimization: Development of a Butyrylcholinesterase Inhibitor with Picomolar Affinity and in Vivo Activity
Košak, Urban, Brus, Boris, Knez, Damijan, Žakelj, Simon, Trontelj, Jurij, Pišlar, Anja, Šink, Roman, Jukič, Marko, Živin, Marko, Podkowa, Adrian, Nachon, Florian, Brazzolotto, Xavier, Stojan, Jure, Kos, Janko, Coquelle, Nicolas, Sałat, Kinga, Colletier, Jacques-Philippe, Gobec, Stanislav
Published in Journal of medicinal chemistry (11.01.2018)
Published in Journal of medicinal chemistry (11.01.2018)
Get full text
Journal Article
Suitability and functional characterization of two Calu-3 cell models for prediction of drug permeability across the airway epithelial barrier
Sibinovska, Nadica, Žakelj, Simon, Roškar, Robert, Kristan, Katja
Published in International journal of pharmaceutics (30.07.2020)
Published in International journal of pharmaceutics (30.07.2020)
Get full text
Journal Article
Stereoselective Activity of 1‑Propargyl-4-styrylpiperidine-like Analogues That Can Discriminate between Monoamine Oxidase Isoforms A and B
Knez, Damijan, Colettis, Natalia, Iacovino, Luca G, Sova, Matej, Pišlar, Anja, Konc, Janez, Lešnik, Samo, Higgs, Josefina, Kamecki, Fabiola, Mangialavori, Irene, Dolšak, Ana, Žakelj, Simon, Trontelj, Jurij, Kos, Janko, Binda, Claudia, Marder, Mariel, Gobec, Stanislav
Published in Journal of medicinal chemistry (13.02.2020)
Published in Journal of medicinal chemistry (13.02.2020)
Get full text
Journal Article
Applicability of RPMI 2650 and Calu-3 Cell Models for Evaluation of Nasal Formulations
Sibinovska, Nadica, Žakelj, Simon, Trontelj, Jurij, Kristan, Katja
Published in Pharmaceutics (06.02.2022)
Published in Pharmaceutics (06.02.2022)
Get full text
Journal Article
Treatment of canine cognitive dysfunction with novel butyrylcholinesterase inhibitor
Zakošek Pipan, Maja, Prpar Mihevc, Sonja, Štrbenc, Malan, Košak, Urban, German Ilić, Ilija, Trontelj, Jurij, Žakelj, Simon, Gobec, Stanislav, Pavlin, Darja, Majdič, Gregor
Published in Scientific reports (13.09.2021)
Published in Scientific reports (13.09.2021)
Get full text
Journal Article
Development of an in-vivo active reversible butyrylcholinesterase inhibitor
Košak, Urban, Brus, Boris, Knez, Damijan, Šink, Roman, Žakelj, Simon, Trontelj, Jurij, Pišlar, Anja, Šlenc, Jasna, Gobec, Martina, Živin, Marko, Tratnjek, Larisa, Perše, Martina, Sałat, Kinga, Podkowa, Adrian, Filipek, Barbara, Nachon, Florian, Brazzolotto, Xavier, Więckowska, Anna, Malawska, Barbara, Stojan, Jure, Raščan, Irena Mlinarič, Kos, Janko, Coquelle, Nicolas, Colletier, Jacques-Philippe, Gobec, Stanislav
Published in Scientific reports (21.12.2016)
Published in Scientific reports (21.12.2016)
Get full text
Journal Article
Biopharmaceutical classification of desloratadine - not all drugs are classified the easy way
Berginc, Katja, Sibinovska, Nadica, Žakelj, Simon, Trontelj, Jurij, Legen, Igor
Published in Acta Pharmaceutica (01.06.2020)
Published in Acta Pharmaceutica (01.06.2020)
Get full text
Journal Article
Paper
The effect of lipid composition and liposome size on the release properties of liposomes-in-hydrogel
Hurler, Julia, Žakelj, Simon, Mravljak, Janez, Pajk, Stane, Kristl, Albin, Schubert, Rolf, Škalko-Basnet, Nataša
Published in International journal of pharmaceutics (01.11.2013)
Published in International journal of pharmaceutics (01.11.2013)
Get full text
Journal Article
Mechanical properties and drug permeability of the PA6 membranes prepared by immersion precipitation from PA6 – formic acid – water system
Aulova, Alexandra, Cvenkel, Anže, Žakelj, Simon, Planinšek, Odon, Kristl, Albin, Emri, Igor
Published in Journal of membrane science (15.09.2018)
Published in Journal of membrane science (15.09.2018)
Get full text
Journal Article
Indoles and 1-(3-(benzyloxy)benzyl)piperazines: Reversible and selective monoamine oxidase B inhibitors identified by screening an in-house compound library
Knez, Damijan, Hrast, Martina, Frlan, Rok, Pišlar, Anja, Žakelj, Simon, Kos, Janko, Gobec, Stanislav
Published in Bioorganic chemistry (01.02.2022)
Published in Bioorganic chemistry (01.02.2022)
Get full text
Journal Article
Determination of permeability coefficients of ophthalmic drugs through different layers of porcine, rabbit and bovine eyes
Loch, Christian, Zakelj, Simon, Kristl, Albin, Nagel, Stefan, Guthoff, Rudolf, Weitschies, Werner, Seidlitz, Anne
Published in European journal of pharmaceutical sciences (30.08.2012)
Published in European journal of pharmaceutical sciences (30.08.2012)
Get full text
Journal Article
8-Hydroxyquinolylnitrones as multifunctional ligands for the therapy of neurodegenerative diseases
Knez, Damijan, Diez-Iriepa, Daniel, Chioua, Mourad, Gottinger, Andrea, Denic, Milica, Chantegreil, Fabien, Nachon, Florian, Brazzolotto, Xavier, Skrzypczak-Wiercioch, Anna, Meden, Anže, Pišlar, Anja, Kos, Janko, Žakelj, Simon, Stojan, Jure, Sałat, Kinga, Serrano, Julia, Fernández, Ana Patricia, Sánchez-García, Aitana, Martínez-Murillo, Ricardo, Binda, Claudia, López-Muñoz, Francisco, Gobec, Stanislav, Marco-Contelles, José
Published in Acta pharmaceutica Sinica. B (01.05.2023)
Published in Acta pharmaceutica Sinica. B (01.05.2023)
Get full text
Journal Article
Decreasing acidity in a series of aldose reductase inhibitors: 2-Fluoro-4-(1H-pyrrol-1-yl)phenol as a scaffold for improved membrane permeation
Chatzopoulou, Maria, Patsilinakos, Alexandros, Vallianatou, Theodosia, Prnova, Marta Soltesova, Žakelj, Simon, Ragno, Rino, Stefek, Milan, Kristl, Albin, Tsantili-Kakoulidou, Anna, Demopoulos, Vassilis J.
Published in Bioorganic & medicinal chemistry (01.04.2014)
Published in Bioorganic & medicinal chemistry (01.04.2014)
Get full text
Journal Article