Functionally selective signaling and broad metabolic benefits by novel insulin receptor partial agonists
Wu, Margaret, Carballo-Jane, Ester, Zhou, Haihong, Zafian, Peter, Dai, Ge, Liu, Mindy, Lao, Julie, Kelly, Terri, Shao, Dan, Gorski, Judith, Pissarnitski, Dmitri, Kekec, Ahmet, Chen, Ying, Previs, Stephen F, Scapin, Giovanna, Gomez-Llorente, Yacob, Hollingsworth, Scott A, Yan, Lin, Feng, Danqing, Huo, Pei, Walford, Geoffrey, Erion, Mark D, Kelley, David E, Lin, Songnian, Mu, James
Published in Nature communications (17.02.2022)
Published in Nature communications (17.02.2022)
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Author Correction: Functionally selective signaling and broad metabolic benefits by novel insulin receptor partial agonists
Wu, Margaret, Carballo-Jane, Ester, Zhou, Haihong, Zafian, Peter, Dai, Ge, Liu, Mindy, Lao, Julie, Kelly, Terri, Shao, Dan, Gorski, Judith, Pissarnitski, Dmitri, Kekec, Ahmet, Chen, Ying, Previs, Stephen F, Scapin, Giovanna, Gomez-Llorente, Yacob, Hollingsworth, Scott A, Yan, Lin, Feng, Danqing, Huo, Pei, Walford, Geoffrey, Erion, Mark D, Kelley, David E, Lin, Songnian, Mu, James
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Published in Nature communications (23.01.2024)
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Estrogen receptor (ER) subtype agonists alter monoamine levels in the female rat brain
Lubbers, Laura S., Zafian, Peter T., Gautreaux, Claris, Gordon, Marisa, Alves, Stephen E., Correa, Lucia, Lorrain, Daniel S., Hickey, Gerard J., Luine, Victoria
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Published in The Journal of steroid biochemistry and molecular biology (01.11.2010)
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Discovery and investigation of a novel class of thiophene-derived antagonists of the human glucagon receptor
Duffy, Joseph L., Kirk, Brian A., Konteatis, Zenon, Campbell, Elizabeth L., Liang, Rui, Brady, Edward J., Candelore, Mari Rios, Ding, Victor D.H., Jiang, Guoqiang, Liu, Frank, Qureshi, Sajjad A., Saperstein, Richard, Szalkowski, Deborah, Tong, Sharon, Tota, Lauri M., Xie, Dan, Yang, Xiaodong, Zafian, Peter, Zheng, Song, Chapman, Kevin T., Zhang, Bei B., Tata, James R.
Published in Bioorganic & medicinal chemistry letters (01.03.2005)
Published in Bioorganic & medicinal chemistry letters (01.03.2005)
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Engineering Glucose Responsiveness Into Insulin
Kaarsholm, Niels C, Lin, Songnian, Yan, Lin, Kelly, Theresa, van Heek, Margaret, Mu, James, Wu, Margaret, Dai, Ge, Cui, Yan, Zhu, Yonghua, Carballo-Jane, Ester, Reddy, Vijay, Zafian, Peter, Huo, Pei, Shi, Shuai, Antochshuk, Valentyn, Ogawa, Aimie, Liu, Franklin, Souza, Sandra C, Seghezzi, Wolfgang, Duffy, Joseph L, Erion, Mark, Nargund, Ravi P, Kelley, David E
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Published in Diabetes (New York, N.Y.) (01.02.2018)
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Discovery of Insulin Receptor Partial Agonists MK-5160 and MK-1092 as Novel Basal Insulins with Potential to Improve Therapeutic Index
Pissarnitski, Dmitri A, Kekec, Ahmet, Yan, Lin, Zhu, Yuping, Feng, Danqing D, Huo, Pei, Madsen-Duggan, Christina, Moyes, Christopher R, Nargund, Ravi P, Kelly, Terri, Zhang, Xiaoping, Carballo-Jane, Ester, Gorski, Judith, Zafian, Peter, Qatanani, Mo, Kaarsholm, Niels, Meng, Fanyu, Jia, Xiujuan, Lee, Keun-Joong, Wang, Weixun, Xu, Sherrie, Hohn, Michael J, Iammarino, Michael J, McCoy, Mark A, Okoh, Grace A, Liang, Yingkai, Hollingsworth, Scott A, Erion, Mark D, Kelley, David E, Garbaccio, Robert M, Zhang, Amy, Mu, James, Lin, Songnian
Published in Journal of medicinal chemistry (14.04.2022)
Published in Journal of medicinal chemistry (14.04.2022)
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Spatial and temporal studies of metabolic activity: contrasting biochemical kinetics in tissues and pathways during fasted and fed states
Daurio, Natalie A, Wang, Yichen, Chen, Ying, Zhou, Haihong, Carballo-Jane, Ester, Mane, Joel, Rodriguez, Carlos G, Zafian, Peter, Houghton, Andrea, Addona, George, McLaren, David G, Zhang, Rena, Shyong, Bao Jen, Bateman, Kevin, Downes, Daniel P, Webb, Maria, Kelley, David E, Previs, Stephen F
Published in American journal of physiology: endocrinology and metabolism (01.06.2019)
Published in American journal of physiology: endocrinology and metabolism (01.06.2019)
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Superior Glycemic Control With a Glucose-Responsive Insulin Analog: Hepatic and Nonhepatic Impacts
Moore, Mary Courtney, Kelley, David E, Camacho, Raul C, Zafian, Peter, Ye, Tian, Lin, Songnian, Kaarsholm, Niels C, Nargund, Ravi, Kelly, Terri M, Van Heek, Margaret, Previs, Stephen F, Moyes, Christopher, Smith, Marta S, Farmer, Ben, Williams, Phil, Cherrington, Alan D
Published in Diabetes (New York, N.Y.) (01.06.2018)
Published in Diabetes (New York, N.Y.) (01.06.2018)
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Erratum. Engineering Glucose Responsiveness Into Insulin. Diabetes 2018;67:299-308
Kaarsholm, Niels C, Lin, Songnian, Yan, Lin, Kelly, Theresa, van Heek, Margaret, Mu, James, Wu, Margaret, Dai, Ge, Cui, Yan, Zhu, Yonghua, Carballo-Jane, Ester, Reddy, Vijay, Zafian, Peter, Huo, Pei, Shi, Shuai, Antochshuk, Valentyn, Ogawa, Aimie, Liu, Franklin, Souza, Sandra C, Seghezzi, Wolfgang, Duffy, Joseph L, Erion, Mark, Nargund, Ravi P, Kelley, David E
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Published in Diabetes (New York, N.Y.) (01.05.2018)
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A novel insulin secretagogue is a phosphodiesterase inhibitor
LEIBOWITZ, M. D, CHHABI BISWAS, BERGER, J, BRADY, E. J, CONTI, M, CULLINAN, C. A, HAYES, N. S, MANGANIELLO, V. C, SAPERSTEIN, R, LU-HU WANG, ZAFIAN, P. T
Published in Diabetes (New York, N.Y.) (1995)
Published in Diabetes (New York, N.Y.) (1995)
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Gary J. Hom, Michael J. Forrest, Thomas J. Bach, Edward Brady, Mari Rios Candelore, Margaret A. Cascieri, Donna J. Fletcher, Michael H. Fisher, Susan A. Iliff, Robert Mathvink, Joseph Metzger, Victor Pecore, Richard Saperstein, Thomas Shih, Ann E. Weber, Matthew Wyvratt, Peter Zafian, D. Euan MacIntyre
Published in The Journal of pharmacology and experimental therapeutics (01.04.2001)
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Published in The Journal of pharmacology and experimental therapeutics (01.04.2001)
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