Substituted 2-Iminopiperidines as Inhibitors of Human Nitric Oxide Synthase Isoforms
Webber, R. Keith, Metz, Suzanne, Moore, William M, Connor, Jane R, Currie, Mark G, Fok, Kam F, Hagen, Timothy J, Hansen, Donald W, Jerome, Gina M, Manning, Pamela T, Pitzele, Barnett S, Toth, Mihaly V, Trivedi, Mahima, Zupec, Mark E, Tjoeng, F. Siong
Published in Journal of medicinal chemistry (01.01.1998)
Published in Journal of medicinal chemistry (01.01.1998)
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Design and Synthesis of Novel Imidazole-Substituted Dipeptide Amides as Potent and Selective Inhibitors of Candida albicans MyristoylCoA:Protein N-Myristoyltransferase and Identification of Related Tripeptide Inhibitors with Mechanism-Based Antifungal Activity
Devadas, Balekudru, Freeman, Sandra K, Zupec, Mark E, Lu, Hwang-Fun, Nagarajan, Srinivasan R, Kishore, Nandini S, Lodge, Jennifer K, Kuneman, David W, McWherter, Charles A, Vinjamoori, Dutt V, Getman, Daniel P, Gordon, Jeffrey I, Sikorski, James A
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Published in Journal of medicinal chemistry (01.08.1997)
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Conformationally Constrained [p-(ω-Aminoalkyl)phenacetyl]-l-seryl-l-lysyl Dipeptide Amides as Potent Peptidomimetic Inhibitors of Candida albicans and Human Myristoyl-CoA:Protein N-Myristoyl Transferase
Nagarajan, Srinivasan R, Devadas, Balekudru, Zupec, Mark E, Freeman, Sandra K, Brown, David L, Lu, Hwang-Fun, Mehta, Pramod P, Kishore, Nandini S, McWherter, Charles A, Getman, Daniel P, Gordon, Jeffrey I, Sikorski, James A
Published in Journal of medicinal chemistry (09.05.1997)
Published in Journal of medicinal chemistry (09.05.1997)
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Design and Syntheses of Potent and Selective Dipeptide Inhibitors of Candida albicans Myristoyl-CoA:Protein N-Myristoyltransferase
Devadas, Balekudru, Zupec, Mark E, Freeman, Sandra K, Brown, David L, Nagarajan, Srinivasan, Sikorski, James A, McWherter, Charles A, Getman, Daniel P, Gordon, Jeffrey I
Published in Journal of medicinal chemistry (01.05.1995)
Published in Journal of medicinal chemistry (01.05.1995)
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Antiplatelet and antithrombotic effects of platelet glycoprotein IIb/IIIa (GPIIb/IIIa) inhibition by arginine-glycine-aspartic acid-serine (RGDS) and arginine-glycine-aspartic acid (RGD) (O-me)Y (SC-46749)
NICHOLSON, N. S, PANZER-KNODLE, S. G, ADAMS, S. P, FEIGEN, L. P, SALYERS, A. K, TAITE, B. B, KING, L. W, MIYANO, M, GORCZINSKI, R. J, WILLIAMS, M. H, ZUPEC, M. E, TJOENG, F. S
Published in The Journal of pharmacology and experimental therapeutics (01.03.1991)
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Published in The Journal of pharmacology and experimental therapeutics (01.03.1991)
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In vitro and in vivo effects of a peptide mimetic (SC-47643) of RGD as an antiplatelet and antithrombotic agent
Nicholson, N.S., Panzer-Knodle, S.G., Salyers, A.K., Taite, B.B., King, L.W., Miyano, M., Gorczynski, R.J., Williams, M.H., Zupec, M.E., Tjoeng, F.S., Adams, S.P., Feigen, L.P.
Published in Thrombosis research (01.06.1991)
Published in Thrombosis research (01.06.1991)
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Substrate specificity of recombinant human renal renin: effect of histidine in the P2 subsite of pH dependence
Green, David W, Aykent, Serdar, Gierse, James K, Zupec, Mark E
Published in Biochemistry (Easton) (01.03.1990)
Published in Biochemistry (Easton) (01.03.1990)
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Differential structure-activity relationships of atrial peptides as natriuretics and renal vasodilators in the dog
Katsube, N., Wakitani, K., Fok, K.F., Tjoeng, F.S., Zupec, M.E., Eubanks, S.R., Adams, S.P., Needleman, P.
Published in Biochemical and biophysical research communications (16.04.1985)
Published in Biochemical and biophysical research communications (16.04.1985)
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Chemical synthesis of bovine transforming growth factor-α: Synthesis, characterization and biological activity
Tou, Jacob S., McGrath, Mike F., Zupec, Mark E., Byatt, John C., Violand, Bernie N., Kaempfe, Larry A., Vineyard, Billy D.
Published in Biochemical and biophysical research communications (16.03.1990)
Published in Biochemical and biophysical research communications (16.03.1990)
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Phosphorylation of high- and low-molecular-mass atrial natriuretic peptide analogs by cyclic AMP-dependent protein kinase
Olins, Gillian M., Mehta, Pramod P., Blehm, Delores J., Patton, Dennis R., Zupec, Mark E., Whipple, Deborah E., Tjoeng, Foe S., Adams, Steven P., Olins, Peter O., Gierse, James K.
Published in FEBS letters (30.11.1987)
Published in FEBS letters (30.11.1987)
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Multiple peptide synthesis using a single support (MPS3)
Tjoeng, F S, Towery, D S, Bulock, J W, Whipple, D E, Fok, K F, Williams, M H, Zupec, M E, Adams, S P
Published in International journal of peptide and protein research (01.02.1990)
Published in International journal of peptide and protein research (01.02.1990)
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Selective peptidic and peptidomimetic inhibitors of Candida albicans myristoylCoA: Protein N-myristoyltransferase: A new approach to antifungal therapy
Sikorski, James A., Devadas, Balekudru, Zupec, Mark E., Freeman, Sandra K., Brown, David L., Lu, Hwang-Fun, Nagarajan, Srinivasan, Mehta, Pramod P., Wade, Arlene C., Kishore, Nandini S., Bryant, Martin L., Getman, Daniel P., McWherter, Charles A., Gordon, Jeffrey I.
Published in Biopolymers (1997)
Published in Biopolymers (1997)
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Scanning alanine mutagenesis and de-peptidization of a Candida albicans myristoyl-CoA:protein N-myristoyltransferase octapeptide substrate reveals three elements critical for molecular recognition
McWherter, C A, Rocque, W J, Zupec, M E, Freeman, S K, Brown, D L, Devadas, B, Getman, D P, Sikorski, J A, Gordon, J I
Published in The Journal of biological chemistry (02.05.1997)
Published in The Journal of biological chemistry (02.05.1997)
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A novel series of orally active antiplatelet agents
Zablocki, Jeffery A., Tjoeng, Foe S., Bovy, Philippe R., Miyano, Masateru, Garland, Robert B., Williams, Kenneth, Schretzman, Lori, Zupec, Mark E., Rico, Joseph G., Lindmark, Richard J., Toth, Mihaly V., McMackins, Dudley E., Adams, Steven P., Panzer-Knodle, Susan G., Nicholson, Nancy S., Taite, Beatrice B., Salyers, Anita K., King, Lucy W., Campion, James G., Feigen, Larry P.
Published in Bioorganic & medicinal chemistry (01.05.1995)
Published in Bioorganic & medicinal chemistry (01.05.1995)
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Replacements for lysine in l-seryl- l-lysyl dipeptide amide inhibitors of candida albicans myristoyl-CoA:protein N-myristoyltransferase
Brown, David L., Devadas, Balekudru, Lu, Hwang-Fun, Nagarajan, Srinivasan, Zupec, Mark E., Freeman, Sandra K., McWherter, Charles A., Getman, Daniel P., Sikorski, James A.
Published in Bioorganic & medicinal chemistry letters (04.02.1997)
Published in Bioorganic & medicinal chemistry letters (04.02.1997)
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N-myristoylation of Arf proteins in Candida albicans : an in vivo assay for evaluating antifungal inhibitors of myristoyl-CoA : protein N-myristoyltransferase : Candida albicans
LODGE, J. K, JACKSON-MACHELSKI, E, DEVADAS, B, ZUPEC, M. E, GETMAN, D. P, KISHORE, N, FREEMAN, S. K, MCWHERTER, C. A, SIKORSKI, J. A, GORDON, J. I
Published in Microbiology (Society for General Microbiology) (1997)
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Published in Microbiology (Society for General Microbiology) (1997)
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Potent in Vitro and in Vivo Inhibitors of Platelet Aggregation Based Upon the Arg-Gly-Asp Sequence of Fibrinogen. (Aminobenzamidino)succinyl (ABAS) Series of Orally Active Fibrinogen Receptor Antagonists
Zablocki, Jeffery A, Rico, Joseph G, Garland, Robert B, Rogers, Thomas E, Williams, Kenneth, Schretzman, Lori A, Rao, Shashidhar A, Bovy, Philippe R, Tjoeng, Foe S
Published in Journal of medicinal chemistry (01.06.1995)
Published in Journal of medicinal chemistry (01.06.1995)
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Design of orally active, non-peptide fibrinogen receptor antagonists. An evolutionary process from the RGD sequence to novel anti-platelet aggregation agents
Bovy, P.R., Tjoeng, F.S., Rico, J.G., Rogers, T.E., Lindmark, R.J., Zablocki, J.A., Garland, R.B., McMackins, D.E., Dayringer, H., Tóth, M.V., Zupec, M.E., Rao, S., Panzer-Knodle, S.G., Nicholson, N.S., Salyers, A., Taite, B.B., Herin, M., Miyano, M., Feigen, L.P., Adams, S.P.
Published in Bioorganic & medicinal chemistry (01.09.1994)
Published in Bioorganic & medicinal chemistry (01.09.1994)
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Journal Article
Potent in vitro and in vivo inhibitors of platelet aggregation based upon the Arg-Gly-Asp sequence of fibrinogen. (Aminobenzamidino)succinyl (ABAS) series of orally activ fibrinogen receptor antagonists
ZABLOCKI, J. A, RICO, J. G, TOTH, M. V, ZUPEC, M. E, MCMACKINS, D. E, ADAMS, S. P, MIYANO, M, MARKOS, C. S, MILTON, M. N, PAULSON, S, HERIN, M, JACQMIN, P, GARLAND, R. B, NICHOLSON, N. S, PANZER-KNODLE, S. G, HAAS, N. F, PAGE, J. D, SZALONY, J. A, TAITE, B. B, SALYERS, A. K, KING, L. W, CAMPION, J. G, FEIGEN, L. P, ROGERS, T. E, WILLIAMS, K, SCHRETZMAN, L. A, RAO, S. A, BOVY, P. R, TJOENG, F. S, LINDMARK, R. J
Published in Journal of medicinal chemistry (1995)
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Published in Journal of medicinal chemistry (1995)
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N-Myristoylation of Arf proteins in Candida albicans: an in vivo assay for evaluating antifungal inhibitors of myristoyl-CoA:protein N-myristoyltransferase
Lodge, Jennifer K, Jackson-Machelski, Emily, Devadas, Balekudru, Zupec, Mark E, Getman, Daniel P, Kishore, Nandini, Freeman, Sandra K, McWherter, Charles A, Sikorski, James A, Gordon, Jeffrey I
Published in Microbiology (Society for General Microbiology) (01.02.1997)
Published in Microbiology (Society for General Microbiology) (01.02.1997)
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