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Published in Molecular pharmacology (01.03.2004)
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Evaluation of the receptor selectivity of the H3 receptor antagonists, iodophenpropit and thioperamide: an interaction with the 5‐HT3 receptor revealed
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Published in British journal of pharmacology (01.10.1995)
Published in British journal of pharmacology (01.10.1995)
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Screening of cattle urine samples for the presence of beta-agonists with a functional test : some preliminary results
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Published in Analyst (London) (01.12.1994)
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Pharmacological characterisation of the histamine H3 receptor in the rat hippocampus
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Published in Brain research (30.03.1998)
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Published in Farmaco (Società chimica italiana : 1989) (30.10.1999)
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Characterization of the Binding Site of the Histamine H3 Receptor. 1. Various Approaches to the Synthesis of 2-(1H-Imidazol-4-yl)cyclopropylamine and Histaminergic Activity of (1R,2R)- and (1S,2S)-2-(1H-Imidazol-4-yl)- cyclopropylamine
De Esch, Iwan J. P, Vollinga, Roeland C, Goubitz, Kees, Schenk, Henk, Appelberg, Ulf, Hacksell, Uli, Lemstra, Sylvia, Zuiderveld, Obbe P, Hoffmann, Marcel, Leurs, Rob, Menge, Wiro M. P. B, Timmerman, Henk
Published in Journal of medicinal chemistry (08.04.1999)
Published in Journal of medicinal chemistry (08.04.1999)
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Synthesis and pharmacological evaluation of some amino-acid-containing cyproheptadine derivatives as dual antagonists of histamine H1- and leukotriene D4-receptors
Zhang, MQ, van de Stolpe, A, Zuiderveld, OP, Timmerman, H
Published in European journal of medicinal chemistry (01.01.1997)
Published in European journal of medicinal chemistry (01.01.1997)
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Opioids activate brain analgesic circuits through cytochrome P450/epoxygenase signaling
Ding, Xinxin, Hough, Lindsay B, Conroy, Jennie L, Fang, Cheng, Gu, Jun, Zeitlin, Scott O, Yang, Weizhu, Yang, Jun, VanAlstine, Melissa A, Nalwalk, Julia W, Albrecht, Phillip J, Mazurkiewicz, Joseph E, Snyder-Keller, Abigail, Shan, Zhixing, Zhang, Shao-Zhong, Wentland, Mark P, Behr, Melissa, Knapp, Brian I, Bidlack, Jean M, Zuiderveld, Obbe P, Leurs, Rob
Published in Nature neuroscience (01.03.2010)
Published in Nature neuroscience (01.03.2010)
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8R-Lisuride Is a Potent Stereospecific Histamine H 1 -Receptor Partial Agonist
Bakker, R. A., Weiner, D. M., ter Laak, T., Beuming, T., Zuiderveld, O. P., Edelbroek, M., Hacksell, U., Timmerman, H., Brann, M. R., Leurs, R.
Published in Molecular pharmacology (01.03.2004)
Published in Molecular pharmacology (01.03.2004)
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N-substituted piperidinyl alkyl imidazoles: Discovery of methimepip as a potent and selective histamine H-3 receptor agonist
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Published in Journal of medicinal chemistry (24.03.2005)
Published in Journal of medicinal chemistry (24.03.2005)
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Identification of 4-(1H-imidazol-4(5)-ylmethyl)pyridine (immethridine) as a novel, potent, and highly selective histamine H-3 receptor agonist
Kitbunnadaj, R, Zuiderveld, OP, Christophe, B, Hulscher, S, Menge, WMPB, Gelens, E, Snip, E, Bakker, RA, Celanire, S, Gillard, M, Talaga, P, Timmerman, H, Leurs, R
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Published in Journal of medicinal chemistry (06.05.2004)
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A selective human H-4-receptor agonist: (-)-2-cyano-1-methyl-3-{(2R,5R)-5-[1H-imidazol-4(5)-yl]tetrahydrofuran-2-yl}methylguanidine
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Published in Journal of medicinal chemistry (03.07.2003)
Published in Journal of medicinal chemistry (03.07.2003)
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Synthesis and structure-activity relationships of conformationally constrained histamine H-3 receptor agonists
Kitbunnadaj, R, Zuiderveld, OP, De Esch, IJP, Vollinga, RC, Bakker, R, Lutz, M, Spek, AL, Cavoy, E, Deltent, MF, Menge, WMPB, Timmerman, H, Leurs, R
Published in Journal of medicinal chemistry (04.12.2003)
Published in Journal of medicinal chemistry (04.12.2003)
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Journal Article
Pharmacological characterisation of the histamine H sub(3) receptor in the rat hippocampus
Alves-Rodrigues, A, Timmerman, H, Willems, E, Lemstra, S, Zuiderveld, O P, Leurs, R
Published in Brain research (30.03.1998)
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Published in Brain research (30.03.1998)
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