Search Results - "ZSOLT SZOMBATHELYI" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Effects of RGH-237 [N-{4-[4-(3-Aminocarbonyl-phenyl)-piperazin-1-yl]-butyl}-4-bromo-benzamide], an Orally Active, Selective Dopamine D3 Receptor Partial Agonist in Animal Models of Cocaine Abuse

Effects of RGH-237 [N-{4-[4-(3-Aminocarbonyl-phenyl)-piperazin-1-yl]-butyl}-4-bromo-benzamide], an Orally Active, Selective Dopamine D3 Receptor Partial Agonist in Animal Models of Cocaine Abuse

by IstvÃ¡n GyertyÃ¡n, BÃ©la Kiss, Krisztina GÃ¡l, IstvÃ¡n Laszlovszky, Attila HorvÃ¡th, Larisza I. GÃ©mesi, Katalin SÃ¡ghy, Gabriella PÃ¡sztor, MÃ¡ria ZÃ¡jer, Margit KapÃ¡s, Ãva Ãgai Csongor, GyÃ¶rgy DomÃ¡ny, KÃ¡roly Tihanyi, Zsolt Szombathelyi
Published in The Journal of pharmacology and experimental therapeutics (01.03.2007)

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Synthesis and Evaluation of 2′-Hydroxyethyl trans-Apovincaminate Derivatives as Antioxidant and Cognitive Enhancer Agents

Synthesis and Evaluation of 2′-Hydroxyethyl trans-Apovincaminate Derivatives as Antioxidant and Cognitive Enhancer Agents

by Nemes, András, Czibula, László, Szántay, Jr, Csaba, Gere, Anikó, Kiss, Béla, Laszy, Judit, Gyertyán, István, Szombathelyi, Zsolt, Szántay, Csaba
Published in Journal of medicinal chemistry (14.02.2008)

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NR2B containing NMDA receptor dependent windup of single spinal neurons

NR2B containing NMDA receptor dependent windup of single spinal neurons

by Kovács, Gyula, Kocsis, Pál, Tarnawa, István, Horváth, Csilla, Szombathelyi, Zsolt, Farkas, Sándor
Published in Neuropharmacology (2004)

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Identification of Metabolic Pathways Involved in the Biotransformation of Tolperisone by Human Microsomal Enzymes

Identification of Metabolic Pathways Involved in the Biotransformation of Tolperisone by Human Microsomal Enzymes

by DALMADI, Balazs, LEIBINGER, Janos, SZEBERENYI, Szabolcs, BORBAS, Timea, FARKAS, Sandor, SZOMBATHELYI, Zsolt, TIHANYI, Karoly
Published in Drug metabolism and disposition (01.05.2003)

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Participation of AMPA- and NMDA-type excitatory amino acid receptors in the spinal reflex transmission, in rat

Participation of AMPA- and NMDA-type excitatory amino acid receptors in the spinal reflex transmission, in rat

by Kocsis, Pál, Tarnawa, István, Szombathelyi, Zsolt, Farkas, Sándor
Published in Brain research bulletin (15.04.2003)

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Cariprazine (RGH-188), a Dopamine D 3 Receptor-Preferring, D 3 /D 2 Dopamine Receptor Antagonist–Partial Agonist Antipsychotic Candidate: In Vitro and Neurochemical Profile

by Kiss, Béla, Horváth, Attila, Némethy, Zsolt, Schmidt, Éva, Laszlovszky, István, Bugovics, Gyula, Fazekas, Károly, Hornok, Katalin, Orosz, Szabolcs, Gyertyán, István, Ágai-Csongor, Éva, Domány, György, Tihanyi, Károly, Adham, Nika, Szombathelyi, Zsolt
Published in The Journal of pharmacology and experimental therapeutics (01.04.2010)

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Cariprazine (RGH-188), a potent D 3/D 2 dopamine receptor partial agonist, binds to dopamine D 3 receptors in vivo and shows antipsychotic-like and procognitive effects in rodents

Cariprazine (RGH-188), a potent D 3/D 2 dopamine receptor partial agonist, binds to dopamine D 3 receptors in vivo and shows antipsychotic-like and procognitive effects in rodents

by Gyertyán, István, Kiss, Béla, Sághy, Katalin, Laszy, Judit, Szabó, Györgyi, Szabados, Tamás, Gémesi, Larisza I., Pásztor, Gabriella, Zájer-Balázs, Mária, Kapás, Margit, Csongor, Éva Ágai, Domány, György, Tihanyi, Károly, Szombathelyi, Zsolt
Published in Neurochemistry international (01.11.2011)

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Cariprazine (RGH-188), a potent D3/D2 dopamine receptor partial agonist, binds to dopamine D3 receptors in vivo and shows antipsychotic-like and procognitive effects in rodents

Cariprazine (RGH-188), a potent D3/D2 dopamine receptor partial agonist, binds to dopamine D3 receptors in vivo and shows antipsychotic-like and procognitive effects in rodents

by GYERTYAN, Istvan, KISS, Béla, AGAI CSONGOR, Eva, DOMANY, György, TIHANYI, Károly, SZOMBATHELYI, Zsolt, SAGHY, Katalin, LASZY, Judit, SZABO, Györgyi, SZABADOS, Tamás, GEMESI, Larisza I, PASZTOR, Gabriella, ZAJER-BALAZS, Mária, KAPAS, Margit
Published in Neurochemistry international (01.11.2011)

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Discovery of 4-amino-3-arylsulfoquinolines, a novel non-acetylenic chemotype of metabotropic glutamate 5 (mGlu5) receptor negative allosteric modulators

Discovery of 4-amino-3-arylsulfoquinolines, a novel non-acetylenic chemotype of metabotropic glutamate 5 (mGlu5) receptor negative allosteric modulators

by Galambos, János, Bielik, Attila, Wágner, Gábor, Domány, György, Kóti, János, Béni, Zoltán, Szigetvári, Áron, Sánta, Zsuzsanna, Orgován, Zoltán, Bobok, Amrita, Kiss, Béla, Mikó-Bakk, Mónika L., Vastag, Mónika, Sághy, Katalin, Krasavin, Mikhail, Gál, Krisztina, Greiner, István, Szombathelyi, Zsolt, Keserű, György M.
Published in European journal of medicinal chemistry (16.06.2017)

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4-Aryl-3-arylsulfonyl-quinolines as negative allosteric modulators of metabotropic GluR5 receptors: From HTS hit to development candidate

4-Aryl-3-arylsulfonyl-quinolines as negative allosteric modulators of metabotropic GluR5 receptors: From HTS hit to development candidate

by Galambos, János, Domány, György, Nógrádi, Katalin, Wágner, Gábor, Keserű, György M., Bobok, Amrita, Kolok, Sándor, Mikó-Bakk, Mónika L., Vastag, Mónika, Sághy, Katalin, Kóti, János, Szakács, Zoltán, Béni, Zoltán, Gál, Krisztina, Szombathelyi, Zsolt, Greiner, István
Published in Bioorganic & medicinal chemistry letters (15.02.2016)

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Thieno[2,3-b]pyridines as negative allosteric modulators of metabotropic GluR5 receptors: Lead optimization

Thieno[2,3-b]pyridines as negative allosteric modulators of metabotropic GluR5 receptors: Lead optimization

by Nogradi, Katalin, Wagner, Gabor, Domany, Gyorgy, Bobok, Amrita, Magdo, Ildiko, Kolok, Sandor, Miko-Bakk, Monika L., Vastag, Monika, Saghy, Katalin, Gyertyan, Istvan, Koti, Janos, Gal, Krisztina, Farkas, Sandor, Keseru, Gyorgy M., Greiner, Istvan, Szombathelyi, Zsolt
Published in Bioorganic & medicinal chemistry letters (15.04.2015)

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Thieno[2,3-b]pyridines as negative allosteric modulators of metabotropic GluR5 receptors: Hit-to-lead optimization

Thieno[2,3-b]pyridines as negative allosteric modulators of metabotropic GluR5 receptors: Hit-to-lead optimization

by Nógrádi, Katalin, Wágner, Gábor, Domány, György, Bobok, Amrita, Magdó, Ildikó, Kiss, Béla, Kolok, Sándor, Fónagy, Katalin, Gyertyán, István, Háda, Viktor, Kóti, János, Gál, Krisztina, Farkas, Sándor, Keserű, György M., Greiner, István, Szombathelyi, Zsolt
Published in Bioorganic & medicinal chemistry letters (15.08.2014)

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Subnanomolar dopamine D3 receptor antagonism coupled to moderate D2 affinity results in favourable antipsychotic-like activity in rodent models: II. behavioural characterisation of RG-15

Subnanomolar dopamine D3 receptor antagonism coupled to moderate D2 affinity results in favourable antipsychotic-like activity in rodent models: II. behavioural characterisation of RG-15

by Gyertyán, István, Sághy, Katalin, Laszy, Judit, Elekes, Ottilia, Kedves, Rita, Gémesi, Larisza I., Pásztor, Gabriella, Zájer-Balázs, Mária, Kapás, Margit, Ágai Csongor, Éva, Domány, György, Kiss, Béla, Szombathelyi, Zsolt
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.11.2008)

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Subnanomolar dopamine D3 receptor antagonism coupled to moderate D2 affinity results in favourable antipsychotic-like activity in rodent models: I. neurochemical characterisation of RG-15

Subnanomolar dopamine D3 receptor antagonism coupled to moderate D2 affinity results in favourable antipsychotic-like activity in rodent models: I. neurochemical characterisation of RG-15

by Kiss, Béla, Laszlovszky, István, Horváth, Attila, Némethy, Zsolt, Schmidt, Éva, Bugovics, Gyula, Fazekas, Károly, Gyertyán, István, Ágai-Csongor, Éva, Domány, György, Szombathelyi, Zsolt
Published in Naunyn-Schmiedeberg's archives of pharmacology (01.11.2008)

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Neuroprotective Effects of Vinpocetine and its Major Metabolite Cis‐apovincaminic Acid on NMDA‐Induced Neurotoxicity in a Rat Entorhinal Cortex Lesion Model

Neuroprotective Effects of Vinpocetine and its Major Metabolite Cis‐apovincaminic Acid on NMDA‐Induced Neurotoxicity in a Rat Entorhinal Cortex Lesion Model

by Nyakas, Csaba, Felszeghy, Klára, Szabó, Róbert, Keijser, Jan N., Luiten, Paul G.M., Szombathelyi, Zsolt, Tihanyi, Károly
Published in CNS neuroscience & therapeutics (01.06.2009)

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Gene Expression Profiling Identifies Key Estradiol Targets in the Frontal Cortex of the Rat

Gene Expression Profiling Identifies Key Estradiol Targets in the Frontal Cortex of the Rat

by Sárvári, Miklós, Hrabovszky, Erik, Kalló, Imre, Galamb, Orsolya, Solymosi, Norbert, Likó, István, Molnár, Béla, Tihanyi, Károly, Szombathelyi, Zsolt, Liposits, Zsolt
Published in Endocrinology (Philadelphia) (01.03.2010)

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Hit-to-lead optimization of disubstituted oxadiazoles and tetrazoles as mGluR5 NAMs

Hit-to-lead optimization of disubstituted oxadiazoles and tetrazoles as mGluR5 NAMs

by Wágner, Gábor, Wéber, Csaba, Nyéki, Olga, Nógrádi, Katalin, Bielik, Attila, Molnár, László, Bobok, Amrita, Horváth, Attila, Kiss, Béla, Kolok, Sándor, Nagy, József, Kurkó, Dalma, Gál, Krisztina, Greiner, István, Szombathelyi, Zsolt, Keserű, György M., Domány, György
Published in Bioorganic & medicinal chemistry letters (15.06.2010)

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Carbamoyloximes as novel non-competitive mGlu5 receptor antagonists

Carbamoyloximes as novel non-competitive mGlu5 receptor antagonists

by Galambos, János, Wágner, Gábor, Nógrádi, Katalin, Bielik, Attila, Molnár, László, Bobok, Amrita, Horváth, Attila, Kiss, Béla, Kolok, Sándor, Nagy, József, Kurkó, Dalma, Bakk, Mónika L., Vastag, Mónika, Sághy, Katalin, Gyertyán, István, Gál, Krisztina, Greiner, István, Szombathelyi, Zsolt, Keserű, György M., Domány, György
Published in Bioorganic & medicinal chemistry letters (01.08.2010)

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Effects of RGH-237 [ N -{4-[4-(3-Aminocarbonyl-phenyl)-piperazin-1-yl]-butyl}-4-bromo-benzamide], an Orally Active, Selective Dopamine D 3 Receptor Partial Agonist in Animal Models of Cocaine Abuse

Effects of RGH-237 [ N -{4-[4-(3-Aminocarbonyl-phenyl)-piperazin-1-yl]-butyl}-4-bromo-benzamide], an Orally Active, Selective Dopamine D 3 Receptor Partial Agonist in Animal Models of Cocaine Abuse

by Gyertyán, István, Kiss, Béla, Gál, Krisztina, Laszlovszky, István, Horváth, Attila, Gémesi, Larisza I., Sághy, Katalin, Pásztor, Gabriella, Zájer, Mária, Kapás, Margit, Csongor, Éva Ágai, Domány, György, Tihanyi, Károly, Szombathelyi, Zsolt
Published in The Journal of pharmacology and experimental therapeutics (01.03.2007)

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NR2B subunit selective NMDA antagonists inhibit neurotoxic effect of alcohol-withdrawal in primary cultures of rat cortical neurones

NR2B subunit selective NMDA antagonists inhibit neurotoxic effect of alcohol-withdrawal in primary cultures of rat cortical neurones

by Nagy, József, Horváth, Csilla, Farkas, Sándor, Kolok, Sándor, Szombathelyi, Zsolt
Published in Neurochemistry international (2004)

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