A novel CDK7 inhibitor of the Pyrazolotriazine class exerts broad-spectrum antiviral activity at nanomolar concentrations
Hutterer, Corina, Eickhoff, Jan, Milbradt, Jens, Korn, Klaus, Zeitträger, Isabel, Bahsi, Hanife, Wagner, Sabrina, Zischinsky, Gunther, Wolf, Alexander, Degenhart, Carsten, Unger, Anke, Baumann, Matthias, Klebl, Bert, Marschall, Manfred
Published in Antimicrobial agents and chemotherapy (01.04.2015)
Published in Antimicrobial agents and chemotherapy (01.04.2015)
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Journal Article
Dual Inhibition of GSK3β and CDK5 Protects the Cytoskeleton of Neurons from Neuroinflammatory-Mediated Degeneration In Vitro and In Vivo
Reinhardt, Lydia, Kordes, Susanne, Reinhardt, Peter, Glatza, Michael, Baumann, Matthias, Drexler, Hannes C.A., Menninger, Sascha, Zischinsky, Gunther, Eickhoff, Jan, Fröb, Claudia, Bhattarai, Prabesh, Arulmozhivarman, Guruchandar, Marrone, Lara, Janosch, Antje, Adachi, Kenjiro, Stehling, Martin, Anderson, Eric N., Abo-Rady, Masin, Bickle, Marc, Pandey, Udai Bhan, Reimer, Michell M., Kizil, Caghan, Schöler, Hans R., Nussbaumer, Peter, Klebl, Bert, Sterneckert, Jared L.
Published in Stem cell reports (05.03.2019)
Published in Stem cell reports (05.03.2019)
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In vivo proof-of-concept for two experimental antiviral drugs, both directed to cellular targets, using a murine cytomegalovirus model
Sonntag, Eric, Hahn, Friedrich, Bertzbach, Luca D., Seyler, Lisa, Wangen, Christina, Müller, Regina, Tannig, Pierre, Grau, Benedikt, Baumann, Matthias, Zent, Eldar, Zischinsky, Gunther, Eickhoff, Jan, Kaufer, Benedikt B., Bäuerle, Tobias, Tsogoeva, Svetlana B., Marschall, Manfred
Published in Antiviral research (01.01.2019)
Published in Antiviral research (01.01.2019)
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Journal Article
Abstract 5936: A novel class of orally bioavailable small molecules induces potent and sustained tumor growth inhibition and T cell infiltration in various solid tumor mouse models
Gapp, Bianca, Zischinsky, Gunther, Urban, Maria, Birnbacher, Nora, Schwarzböck, Alice, Grünaug, Sabine, Gastaldi, Tommaso, Stütz, Anton, Nussbaumer, Peter, Stranner, Stefan, Buchberger, Julia, Birbach, Andreas, Schögl, Daniela, Kuttke, Mario, Dohnal, Alexander, Gugenberger, Romana
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Journal Article
Chemical Validation of DegS As a Target for the Development of Antibiotics with a Novel Mode of Action
Bongard, Jens, Schmitz, Anna Laura, Wolf, Alex, Zischinsky, Gunther, Pieren, Michel, Schellhorn, Birgit, Bravo‐Rodriguez, Kenny, Schillinger, Jasmin, Koch, Uwe, Nussbaumer, Peter, Klebl, Bert, Steinmann, Jörg, Buer, Jan, Sanchez‐Garcia, Elsa, Ehrmann, Michael, Kaiser, Markus
Published in ChemMedChem (05.06.2019)
Published in ChemMedChem (05.06.2019)
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Journal Article
Design and Synthesis of a New Class of Selective Integrin α5β1 Antagonists
Stragies, Roland, Osterkamp, Frank, Zischinsky, Gunther, Vossmeyer, Doerte, Kalkhof, Holger, Reimer, Ulf, Zahn, Grit
Published in Journal of medicinal chemistry (09.08.2007)
Published in Journal of medicinal chemistry (09.08.2007)
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Journal Article
Abstract 416: A novel non-covalent and rapidly reversible proteasome inhibitor for multiple myeloma and various solid cancers
Ahn, Won-Gyun, Jeon, Yeejin, Yang, Yeong-In, Kim, Jaeseung, Lee, Seung-Joo, Koch, Uwe, Zischinsky, Gunther, Choidas, Axel, Pasha, Ayesha, Klebl, Bert, Huber, Robert, Hamacher, Michael, Nam, Kiyean
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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약학적으로 유효한 피라졸로-트리아진 및/또는 피라졸로-피리미딘 유도체
PARK DONGSIK, KOCH UWE, EICKHOFF JAN, KIM JAESEUNG, SEO MOOYOUNG, ZISCHINSKY GUNTHER, JEON YEEJIN, NAM KIYEAN, YU DONGHOON
Year of Publication 23.12.2020
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Year of Publication 23.12.2020
Patent
사이클린 의존성 키나아제의 선택적 억제제로서의 피라졸로-트리아진 및/또는 피라졸로피리미딘 유도체
PARK DONGSIK, EICKHOFF JAN, KIM JAESEUNG, SEO MOOYOUNG, ZISCHINSKY GUNTHER, JEON YEEJIN, NAM KIYEAN, YU DONGHOON
Year of Publication 18.12.2020
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Year of Publication 18.12.2020
Patent
Abstract 2997: Dynarrestin, a novel dynein inhibitor that does not block ciliogenesis
Baumann, Matthias, Höing, Susanne, Yeh, Ting-Yu, Martinez, Nancy, Habenberger, Peter, Kremer, Lea, Drexler, Hannes CA, Küchler, Philipp, Reinhardt, Peter, Choidas, Axel, Zischinsky, Mia-Lisa, Zischinsky, Gunther, Ketcham, Stephanie A., Wagner, Lydia, Nussbaumer, Peter, Ziegler, Slava, Klebl, Bert, Schroer, Trina, Schöler, Hans R., Waldmann, Herbert, Sterneckert, Jared L.
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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Journal Article
α5β1 Integrin Blockade Inhibits Lymphangiogenesis in Airway Inflammation
Okazaki, Tatsuma, Ni, Amy, Ayeni, Oluwasheyi A, Baluk, Peter, Yao, Li-Chin, Vossmeyer, Doerte, Zischinsky, Gunther, Zahn, Grit, Knolle, Jochen, Christner, Claudia, McDonald, Donald M
Published in The American journal of pathology (2009)
Published in The American journal of pathology (2009)
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Journal Article
Dynarrestin, a Novel Inhibitor of Cytoplasmic Dynein
Höing, Susanne, Yeh, Ting-Yu, Baumann, Matthias, Martinez, Nancy E., Habenberger, Peter, Kremer, Lea, Drexler, Hannes C.A., Küchler, Philipp, Reinhardt, Peter, Choidas, Axel, Zischinsky, Mia-Lisa, Zischinsky, Gunther, Nandini, Swaran, Ledray, Aaron P., Ketcham, Stephanie A., Reinhardt, Lydia, Abo-Rady, Masin, Glatza, Michael, King, Stephen J., Nussbaumer, Peter, Ziegler, Slava, Klebl, Bert, Schroer, Trina A., Schöler, Hans R., Waldmann, Herbert, Sterneckert, Jared
Published in Cell chemical biology (19.04.2018)
Published in Cell chemical biology (19.04.2018)
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Journal Article
Abstract 695: The generation of a mono-selective CDK7 inhibitor
Eickhoff, Jan E., Zischinsky, Gunther, Choidas, Axel, Habenberger, Peter, Wolf, Alexander, Degenhardt, Carsten, Baumann, Matthias, Unger, Anke, Ghallab, Ahmad, Werchau, Doreen, Hengstler, Jan, Nussbaumer, Peter, Klebl, Bert M.
Published in Cancer research (Chicago, Ill.) (15.04.2013)
Published in Cancer research (Chicago, Ill.) (15.04.2013)
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Journal Article
SAR of N-phenyl piperidine based oral integrin a5b1 antagonists
Zischinsky, Gunther, Osterkamp, Frank, Vossmeyer, Doerte, Zahn, Grit, Scharn, Dirk, Zwintscher, Ariane, Stragies, Roland
Published in Bioorganic & medicinal chemistry letters (01.01.2010)
Published in Bioorganic & medicinal chemistry letters (01.01.2010)
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Journal Article
Discovery of orally available integrin a5b1 antagonists
Zischinsky, Gunther, Osterkamp, Frank, Vossmeyer, Doerte, Zahn, Grit, Scharn, Dirk, Zwintscher, Ariane, Stragies, Roland
Published in Bioorganic & medicinal chemistry letters (01.01.2010)
Published in Bioorganic & medicinal chemistry letters (01.01.2010)
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