Discovery and Optimization of Potent GPR40 Full Agonists Containing Tricyclic Spirocycles
Wang, Yingcai, Liu, Jiwen (Jim), Dransfield, Paul J, Zhu, Liusheng, Wang, Zhongyu, Du, Xiaohui, Jiao, Xianyun, Su, Yongli, Li, An-rong, Brown, Sean P, Kasparian, Annie, Vimolratana, Marc, Yu, Ming, Pattaropong, Vatee, Houze, Jonathan B, Swaminath, Gayathri, Tran, Thanhvien, Nguyen, Khanh, Guo, Qi, Zhang, Jane, Zhuang, Run, Li, Frank, Miao, Lynn, Bartberger, Michael D, Correll, Tiffany L, Chow, David, Wong, Simon, Luo, Jian, Lin, Daniel C.-H, Medina, Julio C
Published in ACS medicinal chemistry letters (13.06.2013)
Published in ACS medicinal chemistry letters (13.06.2013)
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Discovery and optimization of a series of quinazolinone-derived antagonists of CXCR3
Johnson, Michael, Li, An-Rong, Liu, Jiwen, Fu, Zice, Zhu, Liusheng, Miao, Shichang, Wang, Xuemei, Xu, Qingge, Huang, Alan, Marcus, Andrew, Xu, Feng, Ebsworth, Karen, Sablan, Emmanuel, Danao, Jay, Kumer, Jeff, Dairaghi, Dan, Lawrence, Chris, Sullivan, Tim, Tonn, George, Schall, Thomas, Collins, Tassie, Medina, Julio
Published in Bioorganic & medicinal chemistry letters (15.06.2007)
Published in Bioorganic & medicinal chemistry letters (15.06.2007)
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AMG 837: A potent, orally bioavailable GPR40 agonist
Houze, Jonathan B., Zhu, Liusheng, Sun, Ying, Akerman, Michelle, Qiu, Wei, Zhang, Alex J., Sharma, Rajiv, Schmitt, Michael, Wang, Yingcai, Liu, Jiwen, Liu, Jinqian, Medina, Julio C., Reagan, Jeff D., Luo, Jian, Tonn, George, Zhang, Jane, Lu, Jenny Ying-Lin, Chen, Michael, Lopez, Edwin, Nguyen, Kathy, Yang, Li, Tang, Liang, Tian, Hui, Shuttleworth, Steven J., Lin, Daniel C.-H.
Published in Bioorganic & medicinal chemistry letters (15.01.2012)
Published in Bioorganic & medicinal chemistry letters (15.01.2012)
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Journal Article
Optimization of a series of quinazolinone-derived antagonists of CXCR3
Liu, Jiwen, Fu, Zice, Li, An-Rong, Johnson, Michael, Zhu, Liusheng, Marcus, Andrew, Danao, Jay, Sullivan, Tim, Tonn, George, Collins, Tassie, Medina, Julio
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
Published in Bioorganic & medicinal chemistry letters (01.09.2009)
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Discovery and optimization of a novel series of liver X receptor-α agonists
Li, Leping, Liu, Jiwen, Zhu, Liusheng, Cutler, Serena, Hasegawa, Hirohiko, Shan, Bei, Medina, Julio C.
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
Published in Bioorganic & medicinal chemistry letters (15.03.2006)
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Optimization of the heterocyclic core of the quinazolinone-derived CXCR3 antagonists
Li, An-Rong, Johnson, Michael G., Liu, Jiwen, Chen, Xiaoqi, Du, Xiaohui, Mihalic, Jeffrey T., Deignan, Jeffrey, Gustin, Darin J., Duquette, Jason, Fu, Zice, Zhu, Liusheng, Marcus, Andrew P., Bergeron, Phillipe, McGee, Lawrence R., Danao, Jay, Lemon, Bryan, Carabeo, Teresa, Sullivan, Timothy, Ma, Ji, Tang, Liang, Tonn, George, Collins, Tassie L., Medina, Julio C.
Published in Bioorganic & medicinal chemistry (15.01.2008)
Published in Bioorganic & medicinal chemistry (15.01.2008)
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Optimization of 2-aminothiazole derivatives as CCR4 antagonists
Wang, Xuemei, Xu, Feng, Xu, Qingge, Mahmud, Hossen, Houze, Jonathan, Zhu, Liusheng, Akerman, Michelle, Tonn, George, Tang, Liang, McMaster, Brian E., Dairaghi, Daniel J., Schall, Thomas J., Collins, Tassie L., Medina, Julio C.
Published in Bioorganic & medicinal chemistry letters (15.05.2006)
Published in Bioorganic & medicinal chemistry letters (15.05.2006)
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AMG 176, a Selective MCL1 Inhibitor, Is Effective in Hematologic Cancer Models Alone and in Combination with Established Therapies
Caenepeel, Sean, Brown, Sean P, Belmontes, Brian, Moody, Gordon, Keegan, Kathleen S, Chui, Danny, Whittington, Douglas A, Huang, Xin, Poppe, Leszek, Cheng, Alan C, Cardozo, Mario, Houze, Jonathan, Li, Yunxiao, Lucas, Brian, Paras, Nick A, Wang, Xianghong, Taygerly, Joshua P, Vimolratana, Marc, Zancanella, Manuel, Zhu, Liusheng, Cajulis, Elaina, Osgood, Tao, Sun, Jan, Damon, Leah, Egan, Regina K, Greninger, Patricia, McClanaghan, Joseph D, Gong, Jianan, Moujalled, Donia, Pomilio, Giovanna, Beltran, Pedro, Benes, Cyril H, Roberts, Andrew W, Huang, David C, Wei, Andrew, Canon, Jude, Coxon, Angela, Hughes, Paul E
Published in Cancer discovery (01.12.2018)
Published in Cancer discovery (01.12.2018)
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Discovery of a Potent and Selective Steroidal Glucocorticoid Receptor Antagonist (ORIC-101)
Rew, Yosup, Du, Xiaohui, Eksterowicz, John, Zhou, Haiying, Jahchan, Nadine, Zhu, Liusheng, Yan, Xuelei, Kawai, Hiroyuki, McGee, Lawrence R, Medina, Julio C, Huang, Tom, Chen, Chelsea, Zavorotinskaya, Tatiana, Sutimantanapi, Dena, Waszczuk, Joanna, Jackson, Erica, Huang, Elizabeth, Ye, Qiuping, Fantin, Valeria R, Sun, Daqing
Published in Journal of medicinal chemistry (13.09.2018)
Published in Journal of medicinal chemistry (13.09.2018)
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SARM1 억제제로서 치환된 피리딘 유도체
ZHU LIUSHENG, REYNOLDS CHARLES HOWARD, BROWN SEAN POMEROY, GRICE CHERYL A, KOLLURI RAO, TEGLEY CHRISTOPHER MICHAEL, TASKER ANDREW STEWART
Year of Publication 01.04.2024
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Year of Publication 01.04.2024
Patent
Abstract A133: Development of murine models to evaluate the impact of glucocorticoid receptor (GR) inhibition on chemotherapy response
Jahchan, Nadine, Zhou, Haiying, Stice, James, Kong, Wayne, McWeeney, Dan, Sun, Daqing, Rew, Yosup, Du, Xiaohui, Zhu, Liusheng, Ye, Qiuping, Jackson, Erica L., Fantin, Valeria
Published in Molecular cancer therapeutics (01.01.2018)
Published in Molecular cancer therapeutics (01.01.2018)
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Discovery of a Potent Steroidal Glucocorticoid Receptor Antagonist with Enhanced Selectivity against the Progesterone and Androgen Receptors (OP-3633)
Du, Xiaohui, Eksterowicz, John, Zhou, Haiying, Rew, Yosup, Zhu, Liusheng, Yan, Xuelei, Medina, Julio C, Huang, Tom, Chen, Xi, Sutimantanapi, Dena, Jahchan, Nadine, Kong, Wayne, Sun, Jessica, Zavorotinskaya, Tatiana, Ye, Qiuping, Fantin, Valeria R, Sun, Daqing
Published in Journal of medicinal chemistry (25.07.2019)
Published in Journal of medicinal chemistry (25.07.2019)
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Abstract 4172: Activation of AR signaling by mifepristone enhances prostate cancer growth and impairs enzalutamide response
Zhou, Haiying, Jachan, Nadine, Singh, Mallika, Tran, Chris, McWeeney, Dan, Balbas, Minna, Schenkein, Emily, Zovorotinskaya, Tatiana, Jackson, Erica L., Medina, Julio, Sun, Daqing, Rew, Yosup, Du, Xiaohui, Eksterowicz, John, Yan, Xuelei, Zhu, Liusheng, Ye, Qiuping, Fantin, Valeria
Published in Cancer research (Chicago, Ill.) (01.07.2017)
Published in Cancer research (Chicago, Ill.) (01.07.2017)
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CD73 CD73 INHIBITORS
EKSTEROWICZ JOHN, YEH CHIEN HUNG, SUN DAQING, PHAM JOHNNY, FANTIN VALERIA R, ZAVOROTINSKAYA TATIANA, DU XIAOHUI, BLANK BRIAN R, WU KEJIA, KAWAI HIROYUKI, YE QIUPING, ZHU LIUSHENG, MOORE JARED, REW YOSUP
Year of Publication 02.04.2024
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Year of Publication 02.04.2024
Patent
Discovery of AM-1638: A Potent and Orally Bioavailable GPR40/FFA1 Full Agonist
Brown, Sean P, Dransfield, Paul J, Vimolratana, Marc, Jiao, XianYun, Zhu, Liusheng, Pattaropong, Vatee, Sun, Ying, Liu, Jinqian, Luo, Jian, Zhang, Jane, Wong, Simon, Zhuang, Run, Guo, Qi, Li, Frank, Medina, Julio C, Swaminath, Gayathri, Lin, Daniel C.-H, Houze, Jonathan B
Published in ACS medicinal chemistry letters (13.09.2012)
Published in ACS medicinal chemistry letters (13.09.2012)
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Discovery of the imidazole-derived GPR40 agonist AM-3189
Ma, Zhihua, Lin, Daniel C.-H., Sharma, Rajiv, Liu, Jinqian, Zhu, Liusheng, Li, An-Rong, Kohn, Todd, Wang, Yingcai, Liu, Jiwen (Jim), Bartberger, Michael D., Medina, Julio C., Zhuang, Run, Li, Frank, Zhang, Jane, Luo, Jian, Wong, Simon, Tonn, George R., Houze, Jonathan B.
Published in Bioorganic & medicinal chemistry letters (01.01.2016)
Published in Bioorganic & medicinal chemistry letters (01.01.2016)
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Journal Article
INHIBITORS OF GLUCOCORTICOID RECEPTOR
MINNA DELARAE BALBAS, JOHN EKSTEROWICZ, ZHOU HAIYING, SUN DAQING, JULIO C MEDINA, ZHU LIUSHENG, VALERIA R FANTIN, DU XIAOHUI, YAN XUELEI, LAWRENCE R MCGEE, REW YOSUP
Year of Publication 11.01.2022
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Year of Publication 11.01.2022
Patent
Discovery of AM-6226: A Potent and Orally Bioavailable GPR40 Full Agonist That Displays Efficacy in Nonhuman Primates
Brown, Sean P., Dransfield, Paul, Vimolratana, Marc, Zhu, Liusheng, Luo, Jian, Zhang, Jane, Jiao, XianYun, Pattaropong, Vatee, Wong, Simon, Zhuang, Run, Swaminath, Gayathri, Houze, Jonathan B., Lin, Daniel C.-H.
Published in ACS medicinal chemistry letters (12.07.2018)
Published in ACS medicinal chemistry letters (12.07.2018)
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Journal Article
INHIBITORS OF GLUCOCORTICOID RECEPTOR
MINNA DELARAE BALBAS, JOHN EKSTEROWICZ, ZHOU HAIYING, SUN DAQING, JULIO C MEDINA, ZHU LIUSHENG, VALERIA R FANTIN, DU XIAOHUI, YAN XUELEI, LAWRENCE R MCGEE, REW YOSUP
Year of Publication 21.10.2021
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Year of Publication 21.10.2021
Patent