Sirt5 Is a NAD-Dependent Protein Lysine Demalonylase and Desuccinylase
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Published in Science (American Association for the Advancement of Science) (11.11.2011)
Published in Science (American Association for the Advancement of Science) (11.11.2011)
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The Cac1 subunit of histone chaperone CAF-1 organizes CAF-1-H3/H4 architecture and tetramerizes histones
Liu, Wallace H, Roemer, Sarah C, Zhou, Yeyun, Shen, Zih-Jie, Dennehey, Briana K, Balsbaugh, Jeremy L, Liddle, Jennifer C, Nemkov, Travis, Ahn, Natalie G, Hansen, Kirk C, Tyler, Jessica K, Churchill, Mair Ea
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Published in eLife (30.09.2016)
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Prenylation and Membrane Localization of Cdc42 Are Essential for Activation by DOCK7
Zhou, Yeyun, Johnson, Jared L, Cerione, Richard A, Erickson, Jon W
Published in Biochemistry (Easton) (25.06.2013)
Published in Biochemistry (Easton) (25.06.2013)
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The Bicyclic Intermediate Structure Provides Insights into the Desuccinylation Mechanism of Human Sirtuin 5 (SIRT5)
Zhou, Yeyun, Zhang, Hongmin, He, Bin, Du, Jintang, Lin, Hening, Cerione, Richard A., Hao, Quan
Published in The Journal of biological chemistry (17.08.2012)
Published in The Journal of biological chemistry (17.08.2012)
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Flexible Tethering of ASPP Proteins Facilitates PP-1c Catalysis
Zhou, Yeyun, Millott, Robyn, Kim, Hyeong Jin, Peng, Shiyun, Edwards, Ross A., Skene-Arnold, Tamara, Hammel, Michal, Lees-Miller, Susan P., Tainer, John A., Holmes, Charles F.B., Glover, J. N. Mark
Published in Structure (London) (01.10.2019)
Published in Structure (London) (01.10.2019)
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Plasmodium falciparum Sir2A Preferentially Hydrolyzes Medium and Long Chain Fatty Acyl Lysine
Zhu, Anita Y., Zhou, Yeyun, Khan, Saba, Deitsch, Kirk W., Hao, Quan, Lin, Hening
Published in ACS chemical biology (20.01.2012)
Published in ACS chemical biology (20.01.2012)
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Flexible tethering of ASPP proteins facilitates PP-1c catalysis
Glover, Mark, Zhou, Yeyun, Millott, Robyn, Kim, Hyeong Jin, Peng, Shiyun, Edwards, Ross A., Skene-Arnold, Tamara, Hammel, Michal, Tainer, John A., Holmes, Charles F. B.
Published in Acta crystallographica. Section A, Foundations and advances (20.07.2019)
Published in Acta crystallographica. Section A, Foundations and advances (20.07.2019)
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Discovery of 5‑Azaquinoxaline Derivatives as Potent and Orally Bioavailable Allosteric SHP2 Inhibitors
Elsayed, Mohamed S. A., Blake, James F., Boys, Mark L., Brown, Eric, Chapsal, Bruno D., Chicarelli, Mark J., Cook, Adam W., Fell, Jay B., Fischer, John P., Hanson, Lauren, Lemieux, Christine, Martinson, Matthew C., McCown, Joseph, McNulty, Oren T., Mejia, Macedonio J., Neitzel, Nickolas A., Otten, Jennifer N., Rodriguez, Martha E., Wilcox, Daniel, Wong, Christina E., Zhou, Yeyun, Hinklin, Ronald J.
Published in ACS medicinal chemistry letters (14.12.2023)
Published in ACS medicinal chemistry letters (14.12.2023)
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Abstract 1439: In vivo characterization of a selective FGFR2 inhibitor with potency against gatekeeper and molecular brake mutations
Fischer, John, Bouhana, Karyn, Chicarelli, Mark, Fell, Brad, Fulton, Jennifer, Guarnieri, Anna, Haygood, Leyla, Jalluri, Ravi, Johnson, Amber, Mclean, Brent, Mejia, Max, Rieger, Rob, Robinson, John, Rodriguez, Mareli, Sullivan, Francis, Wang, Yang, Winski, Shannon, Zhou, YeYun
Published in Cancer research (Chicago, Ill.) (04.04.2023)
Published in Cancer research (Chicago, Ill.) (04.04.2023)
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Abstract PO3-26-02: Identification of a novel, brain penetrant, EGFR sparing, ErbB2 inhibitor with activity against oncogenic ErbB2 mutations
Chicarelli, Mark J., Arwood-Levine, Ben, Bettendorf, Tanna, Bouhana, Karyn, Brizendine, Richard, Cable, LouAnn, Crow, Michelle, Fell, Brad, Fischer, John, Fulton, Jennifer, Guarnieri, Anna, Hillman, Madison, Jalluri, Ravi, Krischlunas, Daniel, Koch, Keith, Kumar, Vijay, Malinky, Cori, Rieger, Rob, Robinson, John, Stunkard, Lee, Sullivan, Francis, Turton, Roy, Vine, Logan, Winski, Shannon, Zhou, Yeyun
Published in Cancer research (Chicago, Ill.) (02.05.2024)
Published in Cancer research (Chicago, Ill.) (02.05.2024)
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Abstract PO3-26-01: Preclinical in vitro and in vivo characterization of a novel, wild-type-sparing, PI3Kα H1047R mutant-selective inhibitor
Smith, Aaron C., Arwood-Levine, Ben, Born, Alexandra, Brizendine, Richard, Chatterjee, Payal, Chicarelli, Mark J., Conner, Michael L., Fell, Brad, Fulton, Jennifer, Guarnieri, Anna, Jalluri, Ravi, Knox, Hailey, Koch, Keith, Krischlunas, Daniel, Kumar, Vijay, McHugh, Colin, Mclean, Brent, Nassar, Kelsey, Newhouse, Brad, Rieger, Rob, Robinson, John, Rodriguez, Marelí, Salituro, Leah, Stunkard, Lee, Sullivan, Francis, Turton, Roy, Winski, Shannon, Zhou, Yeyun
Published in Cancer research (Chicago, Ill.) (02.05.2024)
Published in Cancer research (Chicago, Ill.) (02.05.2024)
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Abstract 4486: Characterization of a novel mutant selective, EGFR sparing, ErbB2 inhibitor with activity across activating mutations in systemic and CNS tumors
Fulton, Jennifer, Bettendorf, Tanna, Blandon, Abiezer, Bouhana, Karyn, Brizendine, Richard K., Cable, LouAnn, Chicarelli, Mark J., Crow, Michelle, Fell, Brad, Fischer, John, Guarnieri, Anna, Hillman, Madison, Jalluri, Ravi, Kumar, Vijay, Malinky, Cori A., Rieger, Rob, Robinson, John, Stunkard, Lee, Sullivan, Francis, Trujillo, John I., Winski, Shannon, Zhou, Yeyun
Published in Cancer research (Chicago, Ill.) (22.03.2024)
Published in Cancer research (Chicago, Ill.) (22.03.2024)
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Abstract C161: Identification of a reversible selective FGFR2 clinical development candidate with potency against gatekeeper and molecular brake mutations
Fischer, John, Bouhana, Karyn, Brizendine, Richard, Chicarelli, Mark, Fell, Brad, Fulton, Jennifer, Guarnieri, Anna, Haygood, Leyla, Jalluri, Ravi, Johnson, Amber, Koch, Keith, Koslov-Davino, Erika, Mejia, Max, Rieger, Rob, Robinson, John, Rodriguez, Mareli, Sullivan, Francis, Wang, Yang, Winski, Shannon, Wood, Silas, Zhou, Yeyun
Published in Molecular cancer therapeutics (01.12.2023)
Published in Molecular cancer therapeutics (01.12.2023)
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Abstract 167: Pre-clinical characterization of a novel series of FGFR2 selective inhibitors with potency against clinically relevant mutations
Fischer, John, Bouhana, Karyn, Chicarelli, Mark J., Dahlke, Josh, Fell, Brad, Fulton, Jennifer, Guarnieri, Anna, Jalluri, Ravi, Johnson, Amber, Mclean, Brent, Mejia, Max, Rieger, Rob, Robinson, John, Rodriguez, Mareli, Sullivan, Francis, Wang, Yang, Winski, Shannon, Zhou, Yeyun
Published in Cancer research (Chicago, Ill.) (15.06.2022)
Published in Cancer research (Chicago, Ill.) (15.06.2022)
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Abstract 1440: Identification of a novel EGFR sparing brain penetrant ErbB2 inhibitor with activity against oncogenic ErbB2 mutations
Chicarelli, Mark J, Bouhana, Karyn, Brizendine, Richard K., Cable, LouAnn, Crow, Michelle, Fell, Brad, Fischer, John, Fulton, Jennifer, Guarnieri, Anna, Jalluri, Ravi, Knox, Hailey, Koch, Keith A., Rieger, Rob, Robinson, John, Stunkard, Lee M., Sullivan, Francis, Turton, Roy, Winski, Shannon, Zhou, Yeyun
Published in Cancer research (Chicago, Ill.) (04.04.2023)
Published in Cancer research (Chicago, Ill.) (04.04.2023)
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Design, synthesis and biological characterization of novel inhibitors of CD38
Dong, Min, Si, Yuan-Qi, Sun, Shuang-Yong, Pu, Xiao-Ping, Yang, Zhen-Jun, Zhang, Liang-Ren, Zhang, Li-He, Leung, Fung Ping, Lam, Connie Mo Ching, Kwong, Anna Ka Yee, Yue, Jianbo, Zhou, Yeyun, Kriksunov, Irina A., Hao, Quan, Lee, Hon Cheung
Published in Organic & biomolecular chemistry (07.05.2011)
Published in Organic & biomolecular chemistry (07.05.2011)
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Crystal structure of Saccharomyces cerevisiae glutamine synthetase Gln1 suggests a nanotube-like supramolecular assembly
He, Yong-Xing, Gui, Long, Liu, Yin-Zi, Du, Yang, Zhou, Yeyun, Li, Ping, Zhou, Cong-Zhao
Published in Proteins, structure, function, and bioinformatics (01.07.2009)
Published in Proteins, structure, function, and bioinformatics (01.07.2009)
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Prenylation and Membrane Localization of Cdc42 Are Essential for Activation by DOCK7
Zhou, Yeyun, Johnson Jared L.author, Cerione Richard A.author, Erickson Jon W.author
Year of Publication 2015
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Year of Publication 2015
Journal Article
Tubular oil well pump
ZHAO XIAOLIANG, MU LINGYU, ZHOU XINGZE, ZHAO NING, ZHANG FENGYUAN, LIAO XINWEI, ZHOU YEYUN
Year of Publication 13.01.2016
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Year of Publication 13.01.2016
Patent
Pipe type oil well pump
ZHAO XIAOLIANG, MU LINGYU, ZHOU XINGZE, ZHAO NING, ZHANG FENGYUAN, LIAO XINWEI, ZHOU YEYUN
Year of Publication 09.12.2015
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Year of Publication 09.12.2015
Patent