A novel prognostic signature based on smoking-associated genes for predicting prognosis and immune microenvironment in NSCLC smokers
Li, Qixuan, Wang, Tianyi, Tang, Yijie, Zou, Xian, Shen, Zhongqi, Tang, Zixin, Zhou, Youlang, Shi, Jiahai
Published in Cancer cell international (15.05.2024)
Published in Cancer cell international (15.05.2024)
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The active components of Erzhi wan and their anti-Alzheimer's disease mechanisms determined by an integrative approach of network pharmacology, bioinformatics, molecular docking, and molecular dynamics simulation
Yu, Meng, Shen, Zhongqi, Zhang, Shaozhi, Zhang, Yang, Zhao, Hongwei, Zhang, Longfei
Published in Heliyon (15.07.2024)
Published in Heliyon (15.07.2024)
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2-Aminothiazole as a Novel Kinase Inhibitor Template. Structure−Activity Relationship Studies toward the Discovery of N-(2-Chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyethyl)-1- piperazinyl)]-2-methyl-4-pyrimidinyl]amino)]-1,3-thiazole-5-carboxamide (Dasatinib, BMS-354825) as a Potent pan-Src Kinase Inhibitor
Das, Jagabandhu, Chen, Ping, Norris, Derek, Padmanabha, Ramesh, Lin, James, Moquin, Robert V, Shen, Zhongqi, Cook, Lynda S, Doweyko, Arthur M, Pitt, Sidney, Pang, Suhong, Shen, Ding Ren, Fang, Qiong, de Fex, Henry F, McIntyre, Kim W, Shuster, David J, Gillooly, Kathleen M, Behnia, Kamelia, Schieven, Gary L, Wityak, John, Barrish, Joel C
Published in Journal of medicinal chemistry (16.11.2006)
Published in Journal of medicinal chemistry (16.11.2006)
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Regulatory effects of galanin system on development of several age-related chronic diseases
Fang, Penghua, Yu, Mei, Wan, Dang, Zhang, Lei, Han, Long, Shen, Zhongqi, Shi, Mingyi, Zhu, Yan, Zhang, Zhenwen, Bo, Ping
Published in Experimental gerontology (01.09.2017)
Published in Experimental gerontology (01.09.2017)
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TCM considering EIZs' integration
Liu, Yangyang, Lian, Hongbo, Tang, Xiaowei, Shen, Zhongqi, Li, Jiarui, Liu, Lian
Published in Journal of engineering (Stevenage, England) (01.03.2019)
Published in Journal of engineering (Stevenage, England) (01.03.2019)
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A new facile method for the synthesis of 1-arylimidazole-5-carboxylates
Chen, Bang-Chi, Bednarz, Mark S, Zhao, Rulin, Sundeen, Joseph E, Chen, Ping, Shen, Zhongqi, Skoumbourdis, Amanda P, Barrish, Joel C
Published in Tetrahedron letters (15.07.2000)
Published in Tetrahedron letters (15.07.2000)
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Acridone-Based Inhibitors of Inosine 5‘-Monophosphate Dehydrogenase: Discovery and SAR Leading to the Identification of N-(2-(6-(4-Ethylpiperazin-1-yl)pyridin-3-yl)propan-2-yl)-2- fluoro-9-oxo-9,10-dihydroacridine-3-carboxamide (BMS-566419)
Watterson, Scott H, Chen, Ping, Zhao, Yufen, Gu, Henry H, Dhar, T. G. Murali, Xiao, Zili, Ballentine, Shelley K, Shen, Zhongqi, Fleener, Catherine A, Rouleau, Katherine A, Obermeier, Mary, Yang, Zheng, McIntyre, Kim W, Shuster, David J, Witmer, Mark, Dambach, Donna, Chao, Sam, Mathur, Arvind, Chen, Bang-Chi, Barrish, Joel C, Robl, Jeffrey A, Townsend, Robert, Iwanowicz, Edwin J
Published in Journal of medicinal chemistry (26.07.2007)
Published in Journal of medicinal chemistry (26.07.2007)
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Synthesis and structure-activity relationship of novel lactam-fused chroman derivatives having dual affinity at the 5-HT1A receptor and the serotonin transporter
ZHONGQI SHEN, SIVA RAMAMOORTHY, P, SCHECHTER, Lee E, ANDREE, Terrance H, HATZENBUHLER, Nicole T, EVRARD, Deborah A, CHILDERS, Wayne, HARRISON, Boyd L, CHLENOV, Michael, HORNBY, Geoffrey, SMITH, Deborah L, SULLIVAN, Kelly M
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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3-Cyanoindole-based inhibitors of inosine monophosphate dehydrogenase: Synthesis and initial structure-activity relationships
MURALI DHAR, T. G, ZHONGQI SHEN, TOWNSEND, Robert, HOLLENBAUGH, Diane L, IWANOWICZ, Edwin J, GU, Henry H, PING CHEN, NORRIS, Derek, WATTERSON, Scott H, BALLENTINE, Shelley K, FLEENER, Catherine A, ROULEAU, Katherine A, BARRISH, Joel C
Published in Bioorganic & medicinal chemistry letters (20.10.2003)
Published in Bioorganic & medicinal chemistry letters (20.10.2003)
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Novel indole-based inhibitors of IMPDH: introduction of hydrogen bond acceptors at indole C-3
Watterson, Scott H., Dhar, T.G.Murali, Ballentine, Shelley K., Shen, Zhongqi, Barrish, Joel C., Cheney, Daniel, Fleener, Catherine A., Rouleau, Katherine A., Townsend, Robert, Hollenbaugh, Diane L., Iwanowicz, Edwin J.
Published in Bioorganic & medicinal chemistry letters (07.04.2003)
Published in Bioorganic & medicinal chemistry letters (07.04.2003)
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Discovery of N-[2-[2-[[3-Methoxy-4-(5-oxazolyl)phenyl]amino]-5-oxazolyl]phenyl]-N-methyl-4- morpholineacetamide as a Novel and Potent Inhibitor of Inosine Monophosphate Dehydrogenase with Excellent in Vivo Activity
Dhar, T. G. Murali, Shen, Zhongqi, Guo, Junqing, Liu, Chunjian, Watterson, Scott H, Gu, Henry H, Pitts, William J, Fleener, Catherine A, Rouleau, Katherine A, Sherbina, N. Z, McIntyre, Kim W, Witmer, Mark R, Tredup, Jeffrey A, Chen, Bang-Chi, Zhao, Rulin, Bednarz, Mark S, Cheney, Daniel L, MacMaster, John F, Miller, Laura M, Berry, Karen K, Harper, Timothy W, Barrish, Joel C, Hollenbaugh, Diane L, Iwanowicz, Edwin J
Published in Journal of medicinal chemistry (23.05.2002)
Published in Journal of medicinal chemistry (23.05.2002)
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Journal Article
Rapid synthesis of triazine inhibitors of inosine monophosphate dehydrogenase
Pitts, William J., Guo, Junqing, Dhar, T.G.Murali, Shen, Zhongqi, Gu, Henry H., Watterson, Scott H., Bednarz, Mark S., Chen, Bang-Chi, Barrish, Joel C., Bassolino, Donna, Cheney, Daniel, Fleener, Catherine A., Rouleau, Katherine A., Hollenbaugh, Diane L., Iwanowicz, Edwin J.
Published in Bioorganic & medicinal chemistry letters (19.08.2002)
Published in Bioorganic & medicinal chemistry letters (19.08.2002)
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Journal Article
The TosMIC approach to 3-(Oxazol-5-yl) indoles: application to the synthesis of indole-based IMPDH inhibitors
Dhar, T.G.Murali, Shen, Zhongqi, Fleener, Catherine A., Rouleau, Katherine A., Barrish, Joel C., Hollenbaugh, Diane L., Iwanowicz, Edwin J.
Published in Bioorganic & medicinal chemistry letters (18.11.2002)
Published in Bioorganic & medicinal chemistry letters (18.11.2002)
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Journal Article
Inhibitors of inosine monophosphate dehydrogenase: SARs about the N-[3-Methoxy-4-(5-oxazolyl)phenyl moiety
Iwanowicz, Edwin J., Watterson, Scott H., Guo, Junqing, Pitts, William J., Murali Dhar, T.G., Shen, Zhongqi, Chen, Ping, Gu, Henry H., Fleener, Catherine A., Rouleau, Katherine A., Cheney, Daniel L., Townsend, Robert M., Hollenbaugh, Diane L.
Published in Bioorganic & medicinal chemistry letters (16.06.2003)
Published in Bioorganic & medicinal chemistry letters (16.06.2003)
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Journal Article
Novel inhibitors of IMPDH: a highly potent and selective quinolone-based series
Watterson, Scott H., Carlsen, Marianne, Murali Dhar, T.G., Shen, Zhongqi, Pitts, William J., Guo, Junqing, Gu, Henry H., Norris, Derek, Chorba, John, Chen, Ping, Cheney, Daniel, Witmer, Mark, Fleener, Catherine A., Rouleau, Katherine, Townsend, Robert, Hollenbaugh, Diane L., Iwanowicz, Edwin J.
Published in Bioorganic & medicinal chemistry letters (10.02.2003)
Published in Bioorganic & medicinal chemistry letters (10.02.2003)
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