Novel inhibitors of IMPDH
Watterson, Scott H., Carlsen, Marianne, Murali Dhar, T.G., Shen, Zhongqi, Pitts, William J., Guo, Junqing, Gu, Henry H., Norris, Derek, Chorba, John, Chen, Ping, Cheney, Daniel, Witmer, Mark, Fleener, Catherine A., Rouleau, Katherine, Townsend, Robert, Hollenbaugh, Diane L., Iwanowicz, Edwin J.
Published in Bioorganic & medicinal chemistry letters (01.02.2003)
Published in Bioorganic & medicinal chemistry letters (01.02.2003)
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Discovery and initial SAR of 2-amino-5-carboxamidothiazoles as inhibitors of the Src-family kinase p56 Lck
Wityak, John, Das, Jagabandhu, Moquin, Robert V., Shen, Zhongqi, Lin, James, Chen, Ping, Doweyko, Arthur M., Pitt, Sidney, Pang, Suhong, Shen, Ding Ren, Fang, Qiong, de Fex, Henry F., Schieven, Gary L., Kanner, Steven B., Barrish, Joel C.
Published in Bioorganic & medicinal chemistry letters (2003)
Published in Bioorganic & medicinal chemistry letters (2003)
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Molecular design, synthesis, and structure–Activity relationships leading to the potent and selective p56 lck inhibitor BMS-243117
Das, Jagabandhu, Lin, James, Moquin, Robert V., Shen, Zhongqi, Spergel, Steven H., Wityak, John, Doweyko, Arthur M., DeFex, Henry F., Fang, Qiong, Pang, Suhong, Pitt, Sidney, Shen, Ding Ren, Schieven, Gary L., Barrish, Joel C.
Published in Bioorganic & medicinal chemistry letters (2003)
Published in Bioorganic & medicinal chemistry letters (2003)
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A biomimetic-like radical approach to furanoditerpenes
Zoretic, Phillip A., Shen, Zhongqi, Wang, Ming, Ribeiro, Anthony A.
Published in Tetrahedron letters (24.04.1995)
Published in Tetrahedron letters (24.04.1995)
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Discovery and initial SAR of imidazoquinoxalines as inhibitors of the Src-family kinase p56 Lck
Chen, Ping, Norris, Derek, Iwanowicz, Edwin J., Spergel, Steven H., Lin, James, Gu, Henry H., Shen, Zhongqi, Wityak, John, Lin, Tai-An, Pang, Suhong, De Fex, Henry F., Pitt, Sidney, Shen, Ding Ren, Doweyko, Arthur M., Bassolino, Donna A., Roberge, Jacques Y., Poss, Michael A., Chen, Bang-Chi, Schieven, Gary L., Barrish, Joel C.
Published in Bioorganic & medicinal chemistry letters (2002)
Published in Bioorganic & medicinal chemistry letters (2002)
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Discovery of N-[2-[2-[[3-Methoxy-4-(5-oxazolyl)phenyl]amino]-5-oxazolyl]phenyl]-N-methyl-4-morpholineacetamide as a Novel and Potent Inhibitor of Inosine Monophosphate Dehydrogenase (IMPDH) with Excellent in Vivo Activity
Murali Dhar, T. G, Shen, Zhongqi, Guo, Junqing, Liu, Chunjian, Watterson, Scott H, Gu, Henry H, Pitts, William J, Fleener, Catherine A, Rouleau, Katherine A, Sherbina, N. Z, McIntyre, Kim W, Shuster, David J, Witmer, Mark R, Tredup, Jeffrey A, Chen, Bang-Chi, Zhao, Rulin, Bednarz, Mark S, Cheney, Daniel L, MacMaster, John F, Miller, Laura M, Berry, Karen K, Harper, Timothy W, Barrish, Joel C, Hollenbaugh, Diane L, Iwanowicz, Edwin J
Published in Journal of medicinal chemistry (07.11.2002)
Published in Journal of medicinal chemistry (07.11.2002)
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