Novel diamide-Based inhibitors of IMPDH
Gu, Henry H., Iwanowicz, Edwin J., Guo, Junqing, Watterson, Scott H., Shen, Zhongqi, Pitts, William J., Dhar, T.G.Murali, Fleener, Catherine A., Rouleau, Katherine, Sherbina, N.Z., Witmer, Mark, Tredup, Jeffrey, Hollenbaugh, Diane
Published in Bioorganic & medicinal chemistry letters (06.05.2002)
Published in Bioorganic & medicinal chemistry letters (06.05.2002)
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Quinolone-Based IMPDH inhibitors: introduction of basic residues on ring D and SAR of the corresponding mono, di and benzofused analogues
Dhar, T.G.Murali, Watterson, Scott H., Chen, Ping, Shen, Zhongqi, Gu, Henry H., Norris, Derek, Carlsen, Marianne, Haslow, Kristin D., Pitts, William J., Guo, Junqing, Chorba, John, Fleener, Catherine A., Rouleau, Katherine A., Townsend, Robert, Hollenbaugh, Diane, Iwanowicz, Edwin J.
Published in Bioorganic & medicinal chemistry letters (10.02.2003)
Published in Bioorganic & medicinal chemistry letters (10.02.2003)
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Molecular design, synthesis, and structure-activity relationships leading to the potent and selective p56lck inhibitor BMS-243117
DAS, Jagabandhu, LIN, James, PITT, Sidney, DING REN SHEN, SCHIEVEN, Gary L, BARRISH, Joel C, MOQUIN, Robert V, ZHONGQI SHEN, SPERGEL, Steven H, WITYAK, John, DOWEYKO, Arthur M, DEFEX, Henry F, QIONG FANG, SUHONG PANG
Published in Bioorganic & medicinal chemistry letters (01.07.2003)
Published in Bioorganic & medicinal chemistry letters (01.07.2003)
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Discovery and initial SAR of imidazoquinoxalines as inhibitors of the Src-family kinase p56Lck
PING CHEN, NORRIS, Derek, DE FEX, Henry F, PITT, Sidney, DING REN SHEN, DOWEYKO, Arthur M, BASSOLINO, Donna A, ROBERGE, Jacques Y, POSS, Michael A, CHEN, Bang-Chi, SCHIEVEN, Gary L, BARRISH, Joel C, IWANOWICZ, Edwin J, SPERGEL, Steven H, LIN, James, GU, Henry H, ZHONGQI SHEN, WITYAK, John, LIN, Tai-An, SUHONG PANG
Published in Bioorganic & medicinal chemistry letters (01.05.2002)
Published in Bioorganic & medicinal chemistry letters (01.05.2002)
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The Synthesis and Biological Evaluation of Quinolyl-piperazinyl Piperidines as Potent Serotonin 5-HT1A Antagonists
Childers, Wayne E, Havran, Lisa M, Asselin, Magda, Bicksler, James J, Chong, Dan C, Grosu, George T, Shen, Zhongqi, Abou-Gharbia, Magid, A, Bach, Alvin C, Harrison, Boyd L, Kagan, Natasha, Kleintop, Teresa, Magolda, Ronald, Marathias, Vasilios, Robichaud, Albert J, Sabb, Annmarie L, Zhang, Mei-Yi, Andree, Terrance H, Aschmies, Susan H, Beyer, Chad, Comery, Thomas A, Day, Mark, Grauer, Steven M, Hughes, Zoe A, Rosenzweig-Lipson, Sharon, Platt, Brian, Pulicicchio, Claudine, Smith, Deborah E, Sukoff-Rizzo, Stacy J, Sullivan, Kelly M, Adedoyin, Adedayo, Huselton, Christine, Hirst, Warren D
Published in Journal of medicinal chemistry (27.05.2010)
Published in Journal of medicinal chemistry (27.05.2010)
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Synthesis and structure-activity relationship of novel lactam-fused chroman derivatives having dual affinity at the 5-HT sub(1A) receptor and the serotonin transporter
Shen, Zhongqi, Ramamoorthy, PSiva, Hatzenbuhler, Nicole T, Evrard, Deborah A, Childers, Wayne, Harrison, Boyd L, Chlenov, Michael, Hornby, Geoffrey, Smith, Deborah L, Sullivan, Kelly M, Schechter, Lee E, Andree, Terrance H
Published in Bioorganic & medicinal chemistry letters (01.01.2010)
Published in Bioorganic & medicinal chemistry letters (01.01.2010)
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Journal Article
Synthesis and structure–activity relationship of novel lactam-fused chroman derivatives having dual affinity at the 5-HT 1A receptor and the serotonin transporter
Shen, Zhongqi, Siva Ramamoorthy, P., Hatzenbuhler, Nicole T., Evrard, Deborah A., Childers, Wayne, Harrison, Boyd L., Chlenov, Michael, Hornby, Geoffrey, Smith, Deborah L., Sullivan, Kelly M., Schechter, Lee E., Andree, Terrance H.
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Journal Article
Molecular design, synthesis, and structure-Activity relationships leading to the potent and selective p56(lck) inhibitor BMS-243117
Das, Jagabandhu, Lin, James, Moquin, Robert V, Shen, Zhongqi, Spergel, Steven H, Wityak, John, Doweyko, Arthur M, DeFex, Henry F, Fang, Qiong, Pang, Suhong, Pitt, Sidney, Shen, Ding Ren, Schieven, Gary L, Barrish, Joel C
Published in Bioorganic & medicinal chemistry letters (07.07.2003)
Published in Bioorganic & medicinal chemistry letters (07.07.2003)
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Journal Article
The Synthesis and Biological Evaluation of Quinolyl-piperazinyl Piperidines as Potent Serotonin 5-HT 1A Antagonists
Childers, Wayne E., Havran, Lisa M., Asselin, Magda, Bicksler, James J., Chong, Dan C., Grosu, George T., Shen, Zhongqi, Abou-Gharbia, Magid, A., Bach, Alvin C., Harrison, Boyd L., Kagan, Natasha, Kleintop, Teresa, Magolda, Ronald, Marathias, Vasilios, Robichaud, Albert J., Sabb, Annmarie L., Zhang, Mei-Yi, Andree, Terrance H., Aschmies, Susan H., Beyer, Chad, Comery, Thomas A., Day, Mark, Grauer, Steven M., Hughes, Zoe A., Rosenzweig-Lipson, Sharon, Platt, Brian, Pulicicchio, Claudine, Smith, Deborah E., Sukoff-Rizzo, Stacy J., Sullivan, Kelly M., Adedoyin, Adedayo, Huselton, Christine, Hirst, Warren D.
Published in Journal of medicinal chemistry (27.05.2010)
Published in Journal of medicinal chemistry (27.05.2010)
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Journal Article
Discovery and initial SAR of 2-amino-5-carboxamidothiazoles as inhibitors of the Src-family kinase p56(Lck)
Wityak, John, Das, Jagabandhu, Moquin, Robert V, Shen, Zhongqi, Lin, James, Chen, Ping, Doweyko, Arthur M, Pitt, Sidney, Pang, Suhong, Shen, Ding Ren, Fang, Qiong, de Fex, Henry F, Schieven, Gary L, Kanner, Steven B, Barrish, Joel C
Published in Bioorganic & medicinal chemistry letters (17.11.2003)
Published in Bioorganic & medicinal chemistry letters (17.11.2003)
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