Discovery of non-peptide small molecular CXCR4 antagonists as anti-HIV agents: Recent advances and future opportunities
Zhang, Heng, Kang, Dongwei, Huang, Boshi, Liu, Na, Zhao, Fabao, Zhan, Peng, Liu, Xinyong
Published in European journal of medicinal chemistry (23.05.2016)
Published in European journal of medicinal chemistry (23.05.2016)
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Journal Article
Facilitation of GluN2C-containing NMDA receptors in the external globus pallidus increases firing of fast spiking neurons and improves motor function in a hemiparkinsonian mouse model
Liu, Jinxu, Shelkar, Gajanan P., Sarode, Lopmudra P., Gawande, Dinesh Y., Zhao, Fabao, Clausen, Rasmus Praetorius, Ugale, Rajesh R., Dravid, Shashank Manohar
Published in Neurobiology of disease (01.03.2021)
Published in Neurobiology of disease (01.03.2021)
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Journal Article
Discovery of GluN2A subtype-selective N -methyl-d-aspartate (NMDA) receptor ligands
Jiang, Liyang, Liu, Na, Zhao, Fabao, Huang, Boshi, Kang, Dongwei, Zhan, Peng, Liu, Xinyong
Published in Acta pharmaceutica Sinica. B (01.05.2024)
Published in Acta pharmaceutica Sinica. B (01.05.2024)
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Journal Article
Covalently Targeted Highly Conserved Tyr318 to Improve the Drug Resistance Profiles of HIV-1 NNRTIs: A Proof-of-Concept Study
Zhou, Zhenzhen, Meng, Bairu, An, Jiaqi, Zhao, Fabao, Sun, Yanying, Zeng, Dan, Wang, Wenna, Gao, Shenghua, Xia, Yu, Dun, Caiyun, De Clercq, Erik, Pannecouque, Christophe, Zhan, Peng, Kang, Dongwei, Liu, Xinyong
Published in International journal of molecular sciences (07.01.2023)
Published in International journal of molecular sciences (07.01.2023)
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Journal Article
Identification of Polyphenol Derivatives as Novel SARS-CoV-2 and DENV Non-Nucleoside RdRp Inhibitors
Gao, Shenghua, Song, Letian, Xu, Hongtao, Fikatas, Antonios, Oeyen, Merel, De Jonghe, Steven, Zhao, Fabao, Jing, Lanlan, Jochmans, Dirk, Vangeel, Laura, Cheng, Yusen, Kang, Dongwei, Neyts, Johan, Herdewijn, Piet, Schols, Dominique, Zhan, Peng, Liu, Xinyong
Published in Molecules (Basel, Switzerland) (25.12.2022)
Published in Molecules (Basel, Switzerland) (25.12.2022)
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Discovery and Mechanistic Investigation of Piperazinone Phenylalanine Derivatives with Terminal Indole or Benzene Ring as Novel HIV-1 Capsid Modulators
Xu, Shujing, Sun, Lin, Zalloum, Waleed A, Huang, Tianguang, Zhang, Xujie, Ding, Dang, Shao, Xiaoyu, Jiang, Xiangyi, Zhao, Fabao, Cocklin, Simon, De Clercq, Erik, Pannecouque, Christophe, Dick, Alexej, Liu, Xinyong, Zhan, Peng
Published in Molecules (Basel, Switzerland) (01.12.2022)
Published in Molecules (Basel, Switzerland) (01.12.2022)
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Journal Article
Identification of Novel Diarylpyrimidines as Potent HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors by Exploring the Primer Grip Region
Zhang, Tao, Zhou, Zhongxia, Zhao, Fabao, Sang, Zihao, De Clercq, Erik, Pannecouque, Christophe, Kang, Dongwei, Zhan, Peng, Liu, Xinyong
Published in Pharmaceuticals (Basel, Switzerland) (01.11.2022)
Published in Pharmaceuticals (Basel, Switzerland) (01.11.2022)
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Journal Article
Discovery of novel sulfonamide substituted indolylarylsulfones as potent HIV-1 inhibitors with better safety profiles
Gao, Shenghua, Song, Letian, Cheng, Yusen, Zhao, Fabao, Kang, Dongwei, Song, Shu, Yang, Mianling, Ye, Bing, Zhao, Wei, Tang, Yajie, De Clercq, Erik, Pannecouque, Christophe, Zhan, Peng, Liu, Xinyong
Published in Acta pharmaceutica Sinica. B (01.06.2023)
Published in Acta pharmaceutica Sinica. B (01.06.2023)
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Journal Article
Design and optimization of piperidine-substituted thiophene[3,2-d]pyrimidine-based HIV-1 NNRTIs with improved drug resistance and pharmacokinetic profiles
Sun, Yanying, Zhou, Zhenzhen, Shi, Zhongling, Zhao, Fabao, Xie, Minghui, Zhuo, Zongji, De Clercq, Erik, Pannecouque, Christophe, Kang, Dongwei, Zhan, Peng, Liu, Xinyong
Published in Acta pharmaceutica Sinica. B (01.07.2024)
Published in Acta pharmaceutica Sinica. B (01.07.2024)
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Journal Article
Discovery of ( R )-2-amino-3-triazolpropanoic acid derivatives as NMDA receptor glycine site agonists with GluN2 subunit-specific activity
Zhao, Fabao, Mazis, Georgios, Yi, Feng, Lotti, James S, Layeux, Michael S, Schultz, Eric P, Bunch, Lennart, Hansen, Kasper B, Clausen, Rasmus P
Published in Frontiers in chemistry (17.11.2022)
Published in Frontiers in chemistry (17.11.2022)
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Journal Article
Discovery of diarylpyrimidine derivatives bearing piperazine sulfonyl as potent HIV-1 nonnucleoside reverse transcriptase inhibitors
Jiang, Xiangyi, Huang, Boshi, Rumrill, Shawn, Pople, David, Zalloum, Waleed A., Kang, Dongwei, Zhao, Fabao, Ji, Xiangkai, Gao, Zhen, Hu, Lide, Wang, Zhao, Xie, Minghui, De Clercq, Erik, Ruiz, Francesc X., Arnold, Eddy, Pannecouque, Christophe, Liu, Xinyong, Zhan, Peng
Published in Communications chemistry (29.04.2023)
Published in Communications chemistry (29.04.2023)
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Journal Article
Preparation and properties of optically active poly( N-methacryloyl l-leucine methyl ester)
Feng, Liang, Hu, Jiwen, Liu, Zhilei, Zhao, Fabao, Liu, Guojun
Published in Polymer (Guilford) (15.06.2007)
Published in Polymer (Guilford) (15.06.2007)
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Journal Article
Review of small synthetic molecules targeting HBV capsid assembly
Liu, Na, Zhao, Fabao, Zhan, Peng, Liu, Xinyong
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.01.2015)
Published in Medicinal chemistry (Shp-sariqah, United Arab Emirates) (01.01.2015)
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Journal Article
Non-nucleoside anti-HBV agents: advances in structural optimization and mechanism of action investigations
Liu, Na, Zhao, Fabao, Jia, Haiyong, Rai, Diwakar, Zhan, Peng, Jiang, Xuemei, Liu, Xinyong
Published in MedChemComm (01.01.2015)
Published in MedChemComm (01.01.2015)
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Journal Article
Multiple morphologies of the aggregates from self-assembly of diblock copolymer with relatively long corona-forming block in dilute aqueous solution
Zhao, Fabao, Sun, Jianping, Liu, Zhilei, Feng, Liang, Hu, Jiwen
Published in Journal of polymer science. Part B, Polymer physics (01.02.2010)
Published in Journal of polymer science. Part B, Polymer physics (01.02.2010)
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Journal Article
Improved synthetic route for the GluN2-specific NMDA receptor glycine site agonist AICP
Zhao, Fabao, Rouzbeh, Nirvan, Hansen, Kasper B., Clausen, Rasmus P.
Published in Tetrahedron letters (19.03.2020)
Published in Tetrahedron letters (19.03.2020)
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Journal Article
The nucleotide receptor STING translocates to the phagosomes to negatively regulate anti-fungal immunity
Chen, Tian, Feng, Yiting, Sun, Wanwei, Zhao, Guimin, Wu, Han, Cheng, Xiaochen, Zhao, Fabao, Zhang, Lei, Zheng, Yi, Zhan, Peng, Zhao, Wei, Liu, Bingyu, Gao, Chengjiang
Published in Immunity (Cambridge, Mass.) (08.08.2023)
Published in Immunity (Cambridge, Mass.) (08.08.2023)
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Journal Article
Structure-Based Optimization of Novel Sterol 24-C-Methyltransferase Inhibitors for the Treatment of Candida albicans Infections
Wang, Xue, Jin, Xueyang, Zhao, Fabao, Xu, Zejun, Tan, Wenzhuo, Zhang, Jiaozhen, Xu, Yuliang, Luan, Xiaoyi, Fang, Min, Xie, Zhiyu, Chang, Wenqiang, Lou, Hongxiang
Published in Journal of medicinal chemistry (13.06.2024)
Published in Journal of medicinal chemistry (13.06.2024)
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