Cathepsin B Is Dispensable for Cellular Processing of Cathepsin B-Cleavable Antibody-Drug Conjugates
Caculitan, Niña G, Dela Cruz Chuh, Josefa, Ma, Yong, Zhang, Donglu, Kozak, Katherine R, Liu, Yichin, Pillow, Thomas H, Sadowsky, Jack, Cheung, Tommy K, Phung, Qui, Haley, Benjamin, Lee, Byoung-Chul, Akita, Robert W, Sliwkowski, Mark X, Polson, Andrew G
Published in Cancer research (Chicago, Ill.) (15.12.2017)
Published in Cancer research (Chicago, Ill.) (15.12.2017)
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Journal Article
Preclinical experimental models of drug metabolism and disposition in drug discovery and development
Zhang, Donglu, Luo, Gang, Ding, Xinxin, Lu, Chuang
Published in Acta pharmaceutica Sinica. B (01.12.2012)
Published in Acta pharmaceutica Sinica. B (01.12.2012)
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Journal Article
Effect of ketoconazole and diltiazem on the pharmacokinetics of apixaban, an oral direct factor Xa inhibitor
Frost, Charles E., Byon, Wonkyung, Song, Yan, Wang, Jessie, Schuster, Alan E., Boyd, Rebecca A., Zhang, Donglu, Yu, Zhigang, Dias, Clapton, Shenker, Andrew, LaCreta, Frank
Published in British journal of clinical pharmacology (01.05.2015)
Published in British journal of clinical pharmacology (01.05.2015)
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Journal Article
Drug Concentration Asymmetry in Tissues and Plasma for Small Molecule-Related Therapeutic Modalities
Zhang, Donglu, Hop, Cornelis E C A, Patilea-Vrana, Gabriela, Gampa, Gautham, Seneviratne, Herana Kamal, Unadkat, Jashvant D, Kenny, Jane R, Nagapudi, Karthik, Di, Li, Zhou, Lian, Zak, Mark, Wright, Matthew R, Bumpus, Namandjé N, Zang, Richard, Liu, Xingrong, Lai, Yurong, Khojasteh, S Cyrus
Published in Drug metabolism and disposition (01.10.2019)
Published in Drug metabolism and disposition (01.10.2019)
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Journal Article
Apixaban Metabolism and Pharmacokinetics after Oral Administration to Humans
RAGHAVAN, Nirmala, FROST, Charles E, DONGLU ZHANG, ZHIGANG YU, KAN HE, HAIYING ZHANG, HUMPHREYS, W. Griffith, PINTO, Donald, CHEN, Shiangyuan, BONACORSI, Samuel, WONG, Pancras C
Published in Drug metabolism and disposition (01.01.2009)
Published in Drug metabolism and disposition (01.01.2009)
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Journal Article
Effect of Activated Charcoal on Apixaban Pharmacokinetics in Healthy Subjects
Wang, Xiaoli, Mondal, Sabiha, Wang, Jessie, Tirucherai, Giridhar, Zhang, Donglu, Boyd, Rebecca A., Frost, Charles
Published in American journal of cardiovascular drugs : drugs, devices, and other interventions (01.04.2014)
Published in American journal of cardiovascular drugs : drugs, devices, and other interventions (01.04.2014)
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Journal Article
Targeted drug delivery through the traceless release of tertiary and heteroaryl amines from antibody–drug conjugates
Staben, Leanna R., Koenig, Stefan G., Lehar, Sophie M., Vandlen, Richard, Zhang, Donglu, Chuh, Josefa, Yu, Shang-Fan, Ng, Carl, Guo, Jun, Liu, Yanzhou, Fourie-O'Donohue, Aimee, Go, MaryAnn, Linghu, Xin, Segraves, Nathaniel L., Wang, Tao, Chen, Jinhua, Wei, BinQing, Phillips, Gail D. Lewis, Xu, Keyang, Kozak, Katherine R., Mariathasan, Sanjeev, Flygare, John A., Pillow, Thomas H.
Published in Nature chemistry (01.12.2016)
Published in Nature chemistry (01.12.2016)
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Journal Article
Characterization of efflux transporters involved in distribution and disposition of apixaban
Zhang, Donglu, He, Kan, Herbst, John J, Kolb, Janet, Shou, Wilson, Wang, Lifei, Balimane, Praveen V, Han, Yong-Hae, Gan, Jinping, Frost, Charles E, Humphreys, W Griffith
Published in Drug metabolism and disposition (01.04.2013)
Published in Drug metabolism and disposition (01.04.2013)
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Journal Article
Preclinical discovery of apixaban, a direct and orally bioavailable factor Xa inhibitor
Wong, Pancras C., Pinto, Donald J. P., Zhang, Donglu
Published in Journal of thrombosis and thrombolysis (01.05.2011)
Published in Journal of thrombosis and thrombolysis (01.05.2011)
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Journal Article
The HER2-directed antibody-drug conjugate DHES0815A in advanced and/or metastatic breast cancer: preclinical characterization and phase 1 trial results
Lewis, Gail D., Li, Guangmin, Guo, Jun, Yu, Shang-Fan, Fields, Carter T., Lee, Genee, Zhang, Donglu, Dragovich, Peter S., Pillow, Thomas, Wei, BinQing, Sadowsky, Jack, Leipold, Douglas, Wilson, Tim, Kamath, Amrita, Mamounas, Michael, Lee, M. Violet, Saad, Ola, Choeurng, Voleak, Ungewickell, Alexander, Monemi, Sharareh, Crocker, Lisa, Kalinsky, Kevin, Modi, Shanu, Jung, Kyung Hae, Hamilton, Erika, LoRusso, Patricia, Krop, Ian, Schutten, Melissa M., Commerford, Renee, Sliwkowski, Mark X., Cho, Eunpi
Published in Nature communications (11.01.2024)
Published in Nature communications (11.01.2024)
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Journal Article
Effect of Rifampin on the Pharmacokinetics of Apixaban, an Oral Direct Inhibitor of Factor Xa
Vakkalagadda, Blisse, Frost, Charles, Byon, Wonkyung, Boyd, Rebecca A., Wang, Jessie, Zhang, Donglu, Yu, Zhigang, Dias, Clapton, Shenker, Andrew, LaCreta, Frank
Published in American journal of cardiovascular drugs : drugs, devices, and other interventions (01.04.2016)
Published in American journal of cardiovascular drugs : drugs, devices, and other interventions (01.04.2016)
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Journal Article
In Vitro Assessment of Metabolic Drug-Drug Interaction Potential of Apixaban through Cytochrome P450 Phenotyping, Inhibition, and Induction Studies
LIFEI WANG, DONGLU ZHANG, HUMPHREYS, W. Griffith, GROSSMAN, Scott J, RAGHAVAN, Nirmala, MING YAO, LI MA, FROST, Charles A, MAXWELL, Brad D, CHEN, Shiang-Yuan, KAN HE, GOOSEN, Theunis C
Published in Drug metabolism and disposition (01.03.2010)
Published in Drug metabolism and disposition (01.03.2010)
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Journal Article
Modulating Therapeutic Activity and Toxicity of Pyrrolobenzodiazepine Antibody-Drug Conjugates with Self-Immolative Disulfide Linkers
Pillow, Thomas H, Schutten, Melissa, Yu, Shang-Fan, Ohri, Rachana, Sadowsky, Jack, Poon, Kirsten Achilles, Solis, Willy, Zhong, Fiona, Del Rosario, Geoffrey, Go, Mary Ann T, Lau, Jeffrey, Yee, Sharon, He, Jintang, Liu, Luna, Ng, Carl, Xu, Keyang, Leipold, Douglas D, Kamath, Amrita V, Zhang, Donglu, Masterson, Luke, Gregson, Stephen J, Howard, Philip W, Fang, Fan, Chen, Jinhua, Gunzner-Toste, Janet, Kozak, Katherine K, Spencer, Susan, Polakis, Paul, Polson, Andrew G, Flygare, John A, Junutula, Jagath R
Published in Molecular cancer therapeutics (01.05.2017)
Published in Molecular cancer therapeutics (01.05.2017)
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Journal Article
Intratumoral Payload Concentration Correlates with the Activity of Antibody-Drug Conjugates
Zhang, Donglu, Yu, Shang-Fan, Khojasteh, S Cyrus, Ma, Yong, Pillow, Thomas H, Sadowsky, Jack D, Su, Dian, Kozak, Katherine R, Xu, Keyang, Polson, Andrew G, Dragovich, Peter S, Hop, Cornelis E C A
Published in Molecular cancer therapeutics (01.03.2018)
Published in Molecular cancer therapeutics (01.03.2018)
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