Invention of novel 3-aminopiperidin-2-ones as calcitonin gene-related peptide receptor antagonists
Staas, Donnette D., Bell, Ian M., Burgey, Christopher S., Deng, James Z., Gallicchio, Steven N., Lim, John J., Paone, Daniel V., Potteiger, Craig M., Shaw, Anthony W., Stevenson, Heather, Stump, Craig A., Blair Zartman, C., Moore, Eric L., Bruno, Joseph G., Mosser, Scott D., White, Rebecca B., Kane, Stefanie A., Salvatore, Christopher A., Graham, Samuel L., Williams, Theresa M., Selnick, Harold G., Fraley, Mark E.
Published in Bioorganic & medicinal chemistry letters (01.11.2024)
Published in Bioorganic & medicinal chemistry letters (01.11.2024)
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Journal Article
MK-8825: A potent and selective CGRP receptor antagonist with good oral activity in rats
Bell, Ian M., Stump, Craig A., Gallicchio, Steven N., Staas, Donnette D., Zartman, C. Blair, Moore, Eric L., Sain, Nova, Urban, Mark, Bruno, Joseph G., Calamari, Amy, Kemmerer, Amanda L., Mosser, Scott D., Fandozzi, Christine, White, Rebecca B., Zrada, Matthew M., Selnick, Harold G., Graham, Samuel L., Vacca, Joseph P., Kane, Stefanie A., Salvatore, Christopher A.
Published in Bioorganic & medicinal chemistry letters (15.06.2012)
Published in Bioorganic & medicinal chemistry letters (15.06.2012)
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Journal Article
The discovery of highly potent CGRP receptor antagonists
Stump, Craig A., Bell, Ian M., Bednar, Rodney A., Bruno, Joseph G., Fay, John F., Gallicchio, Steven N., Johnston, Victor K., Moore, Eric L., Mosser, Scott D., Quigley, Amy G., Salvatore, Christopher A., Theberge, Cory R., Blair Zartman, C., Zhang, Xu-Fang, Kane, Stefanie A., Graham, Samuel L., Vacca, Joseph P., Williams, Theresa M.
Published in Bioorganic & medicinal chemistry letters (2009)
Published in Bioorganic & medicinal chemistry letters (2009)
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Journal Article
Identification of a novel RAMP-independent CGRP receptor antagonist
Zartman, C. Blair, Bell, Ian M., Gallicchio, Steven N., Graham, Samuel L., Kane, Stefanie A., Mallee, John J., Rutledge, Ruth Z., Salvatore, Christopher A., Vacca, Joseph P., Williams, Theresa M.
Published in Bioorganic & medicinal chemistry letters (15.11.2011)
Published in Bioorganic & medicinal chemistry letters (15.11.2011)
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Journal Article
Identification and Pharmacological Characterization of Domains Involved in Binding of CGRP Receptor Antagonists to the Calcitonin-like Receptor
Salvatore, Christopher A, Mallee, John J, Bell, Ian M, Zartman, C. Blair, Williams, Theresa M, Koblan, Kenneth S, Kane, Stefanie A
Published in Biochemistry (Easton) (14.02.2006)
Published in Biochemistry (Easton) (14.02.2006)
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Journal Article
The identification of potent, orally bioavailable tricyclic CGRP receptor antagonists
Bell, Ian M., Bednar, Rodney A., Corcoran, Halea A., Fay, John F., Gallicchio, Steven N., Johnston, Victor K., Hershey, James C., Miller-Stein, Cynthia M., Moore, Eric L., Mosser, Scott D., Roller, Shane A., Salvatore, Christopher A., Theberge, Cory R., Wong, Bradley K., Blair Zartman, C., Kane, Stefanie A., Williams, Theresa M., Graham, Samuel L., Vacca, Joseph P.
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
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Journal Article
Discovery of MK-3207: A Highly Potent, Orally Bioavailable CGRP Receptor Antagonist
Bell, Ian M, Gallicchio, Steven N, Wood, Michael R, Quigley, Amy G, Stump, Craig A, Zartman, C. Blair, Fay, John F, Li, Chi-Chung, Lynch, Joseph J, Moore, Eric L, Mosser, Scott D, Prueksaritanont, Thomayant, Regan, Christopher P, Roller, Shane, Salvatore, Christopher A, Kane, Stefanie A, Vacca, Joseph P, Selnick, Harold G
Published in ACS medicinal chemistry letters (08.04.2010)
Published in ACS medicinal chemistry letters (08.04.2010)
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Journal Article
[11C]MK-4232: The First Positron Emission Tomography Tracer for the Calcitonin Gene-Related Peptide Receptor
Bell, Ian M, Gallicchio, Steven N, Stump, Craig A, Bruno, Joseph G, Fan, Hong, Gantert, Liza T, Hostetler, Eric D, Kemmerer, Amanda L, McWherter, Melody, Moore, Eric L, Mosser, Scott D, Purcell, Mona L, Riffel, Kerry, Salvatore, Christopher A, Sanabria-Bohórquez, Sandra, Staas, Donnette D, White, Rebecca B, Williams, Mangay, Zartman, C. Blair, Cook, Jacquelynn J, Hargreaves, Richard J, Kane, Stefanie A, Graham, Samuel L, Selnick, Harold G
Published in ACS medicinal chemistry letters (12.09.2013)
Published in ACS medicinal chemistry letters (12.09.2013)
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Journal Article
Non-peptide calcitonin gene-related peptide receptor antagonists from a benzodiazepinone lead
Williams, Theresa M., Stump, Craig A., Nguyen, Diem N., Quigley, Amy G., Bell, Ian M., Gallicchio, Steven N., Zartman, C. Blair, Wan, Bang-Lin, Penna, Kimberly Della, Kunapuli, Priya, Kane, Stefanie A., Koblan, Ken S., Mosser, Scott D., Rutledge, Ruth Z., Salvatore, Christopher, Fay, John F., Vacca, Joseph P., Graham, Samuel L.
Published in Bioorganic & medicinal chemistry letters (15.05.2006)
Published in Bioorganic & medicinal chemistry letters (15.05.2006)
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Journal Article
Identification of novel, orally bioavailable spirohydantoin CGRP receptor antagonists
Bell, Ian M., Bednar, Rodney A., Fay, John F., Gallicchio, Steven N., Hochman, Jerome H., McMasters, Daniel R., Miller-Stein, Cynthia, Moore, Eric L., Mosser, Scott D., Pudvah, Nicole T., Quigley, Amy G., Salvatore, Christopher A., Stump, Craig A., Theberge, Cory R., Wong, Bradley K., Zartman, C. Blair, Zhang, Xu-Fang, Kane, Stefanie A., Graham, Samuel L., Vacca, Joseph P., Williams, Theresa M.
Published in Bioorganic & medicinal chemistry letters (15.12.2006)
Published in Bioorganic & medicinal chemistry letters (15.12.2006)
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Journal Article
3-Aminopyrrolidinone Farnesyltransferase Inhibitors: Design of Macrocyclic Compounds with Improved Pharmacokinetics and Excellent Cell Potency
Bell, Ian M, Gallicchio, Steven N, Abrams, Marc, Beese, Lorena S, Beshore, Douglas C, Bhimnathwala, Hema, Bogusky, Michael J, Buser, Carolyn A, Culberson, J. Christopher, Davide, Joseph, Ellis-Hutchings, Michelle, Fernandes, Christine, Gibbs, Jackson B, Graham, Samuel L, Hamilton, Kelly A, Hartman, George D, Heimbrook, David C, Homnick, Carl F, Huber, Hans E, Huff, Joel R, Kassahun, Kelem, Koblan, Kenneth S, Kohl, Nancy E, Lobell, Robert B, Lynch, Joseph J, Robinson, Ronald, Rodrigues, A. David, Taylor, Jeffrey S, Walsh, Eileen S, Williams, Theresa M, Zartman, C. Blair
Published in Journal of medicinal chemistry (06.06.2002)
Published in Journal of medicinal chemistry (06.06.2002)
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Journal Article
Potent benzimidazolone-based CGRP receptor antagonists
THEBERGE, Cory R, BEDNAR, Rodney A, WILLIAMS, Theresa M, ZARTMAN, C. Blair, ZHANG, Xu-Fang, GRAHAM, Samuel L, VACCA, Joseph P, BELL, Ian M, CORCORAN, Halea A, FAY, John F, HERSHEY, James C, JOHNSTON, Victor K, KANE, Stefanie A, MOSSER, Scott, SALVATORE, Christopher A
Published in Bioorganic & medicinal chemistry (01.12.2008)
Published in Bioorganic & medicinal chemistry (01.12.2008)
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Journal Article
Identification of potent, highly constrained CGRP receptor antagonists
Stump, Craig A., Bell, Ian M., Bednar, Rodney A., Fay, John F., Gallicchio, Steven N., Hershey, James C., Jelley, Richard, Kreatsoulas, Constantine, Moore, Eric L., Mosser, Scott D., Quigley, Amy G., Roller, Shane A., Salvatore, Christopher A., Sharik, Steven S., Theberge, Cory R., Zartman, C. Blair, Kane, Stefanie A., Graham, Samuel L., Selnick, Harold G., Vacca, Joseph P., Williams, Theresa M.
Published in Bioorganic & medicinal chemistry letters (15.04.2010)
Published in Bioorganic & medicinal chemistry letters (15.04.2010)
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Journal Article
Biochemical and Structural Characterization of a Novel Class of Inhibitors of the Type 1 Insulin-like Growth Factor and Insulin Receptor Kinases
Bell, Ian M, Stirdivant, Steven M, Ahern, Janet, Culberson, J. Christopher, Darke, Paul L, Dinsmore, Christopher J, Drakas, Robert A, Gallicchio, Steven N, Graham, Samuel L, Heimbrook, David C, Hall, Dawn L, Hua, Jin, Kett, Nathan R, Kim, Annette S, Kornienko, Maria, Kuo, Lawrence C, Munshi, Sanjeev K, Quigley, Amy G, Reid, John C, Trotter, B. Wesley, Waxman, Lloyd H, Williams, Theresa M, Zartman, C. Blair
Published in Biochemistry (Easton) (12.07.2005)
Published in Biochemistry (Easton) (12.07.2005)
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Journal Article
Selective electrolytic fluorinations in 70% HF/30% pyridine
Lee, Sarah M., Roseman, Jamie M., Blair Zartman, C., Morrison, Eamonn P., Harrison, Sean J., Stankiewicz, Corrie A., Middleton, W.J.
Published in Journal of fluorine chemistry (01.03.1996)
Published in Journal of fluorine chemistry (01.03.1996)
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Journal Article
N-Arylpiperazinone Inhibitors of Farnesyltransferase: Discovery and Biological Activity
Williams, Theresa M, Bergman, Jeffrey M, Brashear, Karen, Breslin, Michael J, Dinsmore, Christopher J, Hutchinson, John H, MacTough, Suzanne C, Stump, Craig A, Wei, Donna D, Zartman, C. Blair, Bogusky, Michael J, Culberson, J. Christopher, Buser-Doepner, Carolyn, Davide, Joseph, Greenberg, Ian B, Hamilton, Kelly A, Koblan, Kenneth S, Kohl, Nancy E, Liu, Dongming, Lobell, Robert B, Mosser, Scott D, O'Neill, Timothy J, Rands, Elaine, Schaber, Michael D, Wilson, Francine, Senderak, Edith, Motzel, Sherri L, Gibbs, Jackson B, Graham, Samuel L, Heimbrook, David C, Hartman, George D, Oliff, Allen I, Huff, Joel R
Published in Journal of medicinal chemistry (23.09.1999)
Published in Journal of medicinal chemistry (23.09.1999)
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Journal Article
Acetonitrile/water gas-phase reaction products observed by use of atmospheric pressure chemical ionization: adducts formed with sulfonamides
Ross III, Charles W., Coddington, Arthur B., Murphy, Joan S., Wisnoski, David D., Zartman, C. Blair, Ramjit, Harri G.
Published in Rapid communications in mass spectrometry (01.01.2005)
Published in Rapid communications in mass spectrometry (01.01.2005)
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Journal Article
Macrocyclic piperazinones as potent dual inhibitors of farnesyltransferase and geranylgeranyltransferase-I
Dinsmore, Christopher J, Zartman, C.Blair, Bergman, Jeffrey M, Abrams, Marc T, Buser, Carolyn A, Culberson, J.Christopher, Davide, Joseph P, Ellis-Hutchings, Michelle, Fernandes, Christine, Graham, Samuel L, Hartman, George D, Huber, Hans E, Lobell, Robert B, Mosser, Scott D, Robinson, Ronald G, Williams, Theresa M
Published in Bioorganic & medicinal chemistry letters (09.02.2004)
Published in Bioorganic & medicinal chemistry letters (09.02.2004)
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Journal Article
Conformational Restriction of Flexible Ligands Guided by the Transferred NOE Experiment: Potent Macrocyclic Inhibitors of Farnesyltransferase
Dinsmore, Christopher J, Bogusky, Michael J, Culberson, J. Christopher, Bergman, Jeffrey M, Homnick, Carl F, Zartman, C. Blair, Mosser, Scott D, Schaber, Michael D, Robinson, Ronald G, Koblan, Kenneth S, Huber, Hans E, Graham, Samuel L, Hartman, George D, Huff, Joel R, Williams, Theresa M
Published in Journal of the American Chemical Society (07.03.2001)
Published in Journal of the American Chemical Society (07.03.2001)
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