Eco-friendly methods of synthesis and preliminary biological evaluation of sulfonamide derivatives of cyclic arylguanidines
Zaręba, Przemysław, Drabczyk, Anna K., Wnorowski, Artur, Pindelska, Edyta, Latacz, Gniewomir, Jaśkowska, Jolanta
Published in Ultrasonics sonochemistry (01.11.2022)
Published in Ultrasonics sonochemistry (01.11.2022)
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Journal Article
Design, synthesis and molecular modelling of new bulky Fananserin derivatives with altered pharmacological profile as potential antidepressants
Zaręba, Przemysław, Jaśkowska, Jolanta, Czekaj, Izabela, Satała, Grzegorz
Published in Bioorganic & medicinal chemistry (01.08.2019)
Published in Bioorganic & medicinal chemistry (01.08.2019)
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Journal Article
New, Eco-Friendly Method for Synthesis of 3-Chlorophenyl and 1,1′-Biphenyl Piperazinylhexyl Trazodone Analogues with Dual 5-HT1A/5-HT7 Affinity and Its Antidepressant-like Activity
Zaręba, Przemysław, Partyka, Anna, Latacz, Gniewomir, Satała, Grzegorz, Zajdel, Paweł, Jaśkowska, Jolanta
Published in Molecules (Basel, Switzerland) (26.10.2022)
Published in Molecules (Basel, Switzerland) (26.10.2022)
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Journal Article
Microwave-Assisted Synthesis of Trazodone and Its Derivatives as New 5-HT1A Ligands: Binding and Docking Studies
Jaśkowska, Jolanta, Zaręba, Przemysław, Śliwa, Paweł, Pindelska, Edyta, Satała, Grzegorz, Majka, Zbigniew
Published in Molecules (Basel, Switzerland) (23.04.2019)
Published in Molecules (Basel, Switzerland) (23.04.2019)
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Journal Article
New N-aryl-N′-aryl-/(thio)ureido-/sulfamoylamino-derivatives of alkyl/alkylcarbamoyl piperazines: Effect of structural modifications on selectivity over 5-HT1A receptor
Zaręba, Przemysław, Śliwa, Paweł, Satała, Grzegorz, Zajdel, Paweł, Latacz, Gniewomir, Jaśkowska, Jolanta
Published in European journal of medicinal chemistry (05.05.2022)
Published in European journal of medicinal chemistry (05.05.2022)
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Journal Article
New Pharmaceutical Salts of Trazodone
Jaśkowska, Jolanta, Zaręba, Przemysław, Drabczyk, Anna, Kozak, Agnieszka, Madura, Izabela D, Majka, Zbigniew, Pindelska, Edyta
Published in Molecules (Basel, Switzerland) (02.02.2021)
Published in Molecules (Basel, Switzerland) (02.02.2021)
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Journal Article
Ultrasound assisted one-pot synthesis and preliminary in vitro studies of salicylamide arylpiperazines as dual 5-HT1A/5-HT7 ligands
Jaśkowska, Jolanta, Drabczyk, Anna Karolina, Śliwa, Paweł, Jodłowski, Przemysław, Pindelska, Edyta, Kułaga, Damian, Zaręba, Przemysław, Majka, Zbigniew, Siwek, Agata, Wolak, Małgorzata, Kołaczkowski, Marcin
Published in Journal of molecular structure (05.03.2023)
Published in Journal of molecular structure (05.03.2023)
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Journal Article
Green synthesis of 1,3,5-triazine derivatives using a sonochemical protocol
Kułaga, Damian, Drabczyk, Anna K., Zaręba, Przemysław, Jaśkowska, Jolanta, Chrzan, Julia, Ewa Greber, Katarzyna, Ciura, Krzesimir, Plażuk, Damian, Wielgus, Ewelina
Published in Ultrasonics sonochemistry (01.08.2024)
Published in Ultrasonics sonochemistry (01.08.2024)
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Journal Article
A new synthetic ultrasound-assisted method for dibenzoepines
Jaśkowska, Jolanta, Drabczyk, Anna Karolina, Kułaga, Damian, Zaręba, Przemysław, Majka, Zbigniew, Jodłowski, Przemysław
Published in Heliyon (01.07.2023)
Published in Heliyon (01.07.2023)
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Journal Article
Eco-friendly synthesis of new olanzapine derivatives and evaluation of their anticancer potential
Drabczyk, Anna K, Ku aga, Damian, Zar ba, Przemys aw, Tyli ska, Wiktoria, Bachowski, Wojciech, Archa a, Aneta, Wnorowski, Artur, Tzani, Andromachi, Detsi, Anastasia, Ja kowska, Jolanta
Published in RSC advances (07.07.2023)
Published in RSC advances (07.07.2023)
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Journal Article
Mechanochemical Synthesis Method for Drugs Used in the Treatment of CNS Diseases under PTC Conditions
Jaśkowska, Jolanta, Drabczyk, Anna Karolina, Michorczyk, Piotr, Kułaga, Damian, Zaręba, Przemysław, Jodłowski, Przemysław, Majka, Zbigniew, Jakubski, Jarosław, Pindelska, Edyta
Published in Catalysts (21.04.2022)
Published in Catalysts (21.04.2022)
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Journal Article
Solvent-free microwave-assisted synthesis of aripiprazole
Jaśkowska, Jolanta, Drabczyk, Anna K., Kułaga, Damian, Zaręba, Przemysław, Majka, Zbigniew
Published in Current chemistry letters (2018)
Published in Current chemistry letters (2018)
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Journal Article
New, Eco-Friendly Method for Synthesis of 3-Chlorophenyl and 1,1′-Biphenyl Piperazinylhexyl Trazodone Analogues with Dual 5-HT[sub.1A]/5-HT[sub.7] Affinity and Its Antidepressant-like Activity
Zaręba, Przemysław, Partyka, Anna, Latacz, Gniewomir, Satała, Grzegorz, Zajdel, Paweł, Jaśkowska, Jolanta
Published in Molecules (Basel, Switzerland) (01.10.2022)
Published in Molecules (Basel, Switzerland) (01.10.2022)
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Journal Article
New N-aryl-N'-aryl-/(thio)ureido-/sulfamoylamino-derivatives of alkyl/alkylcarbamoyl piperazines: Effect of structural modifications on selectivity over 5-HT 1A receptor
Zaręba, Przemysław, Śliwa, Paweł, Satała, Grzegorz, Zajdel, Paweł, Latacz, Gniewomir, Jaśkowska, Jolanta
Published in European journal of medicinal chemistry (05.05.2022)
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Published in European journal of medicinal chemistry (05.05.2022)
Journal Article
Microwave-Assisted Synthesis of Trazodone and Its Derivatives as New 5-HT 1A Ligands: Binding and Docking Studies
Jaśkowska, Jolanta, Zaręba, Przemysław, Śliwa, Paweł, Pindelska, Edyta, Satała, Grzegorz, Majka, Zbigniew
Published in Molecules (Basel, Switzerland) (23.04.2019)
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Published in Molecules (Basel, Switzerland) (23.04.2019)
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