Human Immunodeficiency Virus Type 1 cDNA Integration: New Aromatic Hydroxylated Inhibitors and Studies of the Inhibition Mechanism
FARNET, C. M, WANG, B, HANSEN, M, LIPFORD, J. R, ZALKOW, L, ROBINSON, W. E, SIEGEL, J, BUSHMAN, F
Published in Antimicrobial Agents and Chemotherapy (01.09.1998)
Published in Antimicrobial Agents and Chemotherapy (01.09.1998)
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Syntheses and Biological Activities of a Novel Group of Steroidal Derived Inhibitors for Human CDC25A Protein Phosphatase
Peng, Hairuo, Xie, Wenge, Otterness, Diane M, Cogswell, John P, McConnell, Randy T, Carter, H. Luke, Powis, Garth, Abraham, Robert T, Zalkow, Leon H
Published in Journal of medicinal chemistry (01.03.2001)
Published in Journal of medicinal chemistry (01.03.2001)
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Steroidal derived acids as inhibitors of human Cdc25A protein phosphatase
HAIRUO PENG, WENGE XIE, KIM, D.-I, ZALKOW, L. H, POWIS, G, OTTERNESS, D. M, ABRAHAM, R. T
Published in Bioorganic & medicinal chemistry (01.02.2000)
Published in Bioorganic & medicinal chemistry (01.02.2000)
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A multiwell assay for inhibitors of phosphatidylinositol-3-kinase and the identification of natural product inhibitors
Frew, T, Powis, G, Berggren, M, Abraham, R T, Ashendel, C L, Zalkow, L H, Hudson, C, Qazia, S, Gruszecka-Kowalik, E, Merriman, R
Published in Anticancer research (01.11.1994)
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Published in Anticancer research (01.11.1994)
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Antiviral activity of a derivative of the photosensitive compound Hypericin
Yip, L., Hudson, J.B., Gruszecka-Kowalik, E., Zalkow, L.H., Neil Towers, G.H.
Published in Phytomedicine (Stuttgart) (01.09.1996)
Published in Phytomedicine (Stuttgart) (01.09.1996)
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Synthesis of 2-Methyl-(Z)-4-(phenylimino)naphth[2,3-d]oxazol-9-one, a Monoimine Quinone with Selective Cytotoxicity toward Cancer Cells
Benedetti-Doctorovich, Violeta, Burgess, Edward M, Lambropoulos, John, Lednicer, Daniel, Van Derveer, Donald, Zalkow, Leon H
Published in Journal of medicinal chemistry (01.03.1994)
Published in Journal of medicinal chemistry (01.03.1994)
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Structure–activity relationship of Aza-steroids as PI-PLC inhibitors
Xie, Wenge, Peng, Hairuo, Kim, Deog-Il, Kunkel, Mark, Powis, Garth, Zalkow, Leon H.
Published in Bioorganic & medicinal chemistry (01.05.2001)
Published in Bioorganic & medicinal chemistry (01.05.2001)
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Novel anthraquinone inhibitors of human leukocyte elastase and cathepsin G
Zembower, David E, Kam, Chih Min, Powers, James C, Zalkow, Leon H
Published in Journal of medicinal chemistry (01.05.1992)
Published in Journal of medicinal chemistry (01.05.1992)
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Inhibition of intracellular Ca2+ signalling, cytotoxicity and antitumor activity of the herbicide oryzalin and its analogues
POWIS, G, GALLEGOS, A, ABRAHAM, R. T, ASHENDEL, C. L, ZALKOW, L. H, DORR, R, DVORAKOVA, K, SALMON, S, HARRISON, S, WORZALLA, J
Published in Cancer chemotherapy and pharmacology (1997)
Published in Cancer chemotherapy and pharmacology (1997)
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Quinobene, a new potent anti-HIV agent
Gruszecka-Kowalik, Ewa, Haugwitz, Rudiger D., Zalkow, Leon H.
Published in Biochemical and biophysical research communications (30.09.1992)
Published in Biochemical and biophysical research communications (30.09.1992)
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A multisample assay for inhibitors of phosphatidylinositol phospholipase C: identification of naturally occurring peptide inhibitors with antiproliferative activity
Hill, S R, Bonjouklian, R, Powis, G, Abraham, R T, Ashendel, C L, Zalkow, L H
Published in Anti-cancer drug design (01.08.1994)
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Published in Anti-cancer drug design (01.08.1994)
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Advances with phospholipid signalling as a target for anticancer drug development
Powis, G, Berggren, M, Gallegos, A, Frew, T, Hill, S, Kozikowski, A, Bonjouklian, R, Zalkow, L, Abraham, R, Ashendel, C
Published in Acta biochimica polonica (01.01.1995)
Published in Acta biochimica polonica (01.01.1995)
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Novel quinone antiproliferative inhibitors of phosphatidylinositol-3-kinase
Frew, T, Powis, G, Berggren, M, Gallegos, A, Abraham, R T, Ashendel, C L, Zalkow, L H, Hudson, C, Gruszecka-Kowalik, E, Burgess, E M
Published in Anti-cancer drug design (01.06.1995)
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Published in Anti-cancer drug design (01.06.1995)
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