Drug Concentration Asymmetry in Tissues and Plasma for Small Molecule-Related Therapeutic Modalities
Zhang, Donglu, Hop, Cornelis E C A, Patilea-Vrana, Gabriela, Gampa, Gautham, Seneviratne, Herana Kamal, Unadkat, Jashvant D, Kenny, Jane R, Nagapudi, Karthik, Di, Li, Zhou, Lian, Zak, Mark, Wright, Matthew R, Bumpus, Namandjé N, Zang, Richard, Liu, Xingrong, Lai, Yurong, Khojasteh, S Cyrus
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Structure-Based Discovery of Novel Amide-Containing Nicotinamide Phosphoribosyltransferase (Nampt) Inhibitors
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Identification of 2,3-dihydro-1H-pyrrolo[3,4-c]pyridine-derived ureas as potent inhibitors of human nicotinamide phosphoribosyltransferase (NAMPT)
Dragovich, Peter S., Bair, Kenneth W., Baumeister, Timm, Ho, Yen-Ching, Liederer, Bianca M., Liu, Xiongcai, Liu, Yongbo, O’Brien, Thomas, Oeh, Jason, Sampath, Deepak, Skelton, Nicholas, Wang, Leslie, Wang, Weiru, Wu, Hongxing, Xiao, Yang, Yuen, Po-wai, Zak, Mark, Zhang, Lei, Zheng, Xiaozhang
Published in Bioorganic & medicinal chemistry letters (01.09.2013)
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Total Synthesis of Thiostrepton. Retrosynthetic Analysis and Construction of Key Building Blocks
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Published in Journal of the American Chemical Society (10.08.2005)
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Zheng, Xiaozhang, Baumeister, Timm, Buckmelter, Alexandre J., Caligiuri, Maureen, Clodfelter, Karl H., Han, Bingsong, Ho, Yen-Ching, Kley, Nikolai, Lin, Jian, Reynolds, Dominic J., Sharma, Geeta, Smith, Chase C., Wang, Zhongguo, Dragovich, Peter S., Oh, Angela, Wang, Weiru, Zak, Mark, Wang, Yunli, Yuen, Po-wai, Bair, Kenneth W.
Published in Bioorganic & medicinal chemistry letters (01.01.2014)
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Nicolaou, K. C, Zak, Mark, Rahimipour, Shai, Estrada, Anthony A, Lee, Sang Hyup, O'Brate, Aurora, Giannakakou, Paraskevi, Ghadiri, M. Reza
Published in Journal of the American Chemical Society (02.11.2005)
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Zak, Mark, Dengler, Hart S., Rajapaksa, Naomi S.
Published in Bioorganic & medicinal chemistry letters (15.10.2019)
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Measuring Nad + Levels in Mouse Blood and Tissue Samples Via A Surrogate Matrix Approach Using LC–MS/MS
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Inhaled JAK inhibitor GDC-0214 reduces exhaled nitric oxide in patients with mild asthma: A randomized, controlled, proof-of-activity trial
Braithwaite, Irene E., Cai, Fang, Tom, Jennifer A., Galanter, Joshua M., Owen, Ryan P., Zhu, Rui, Williams, Mathew, McGregor, Anna G., Eliahu, Avi, Durk, Matthew R., Dengler, Hart S., Zak, Mark, Kenny, Jane R., Wilson, Maria E., Beasley, Richard, Chen, Hubert
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Nonfatal Occupational Injuries and Illnesses Among Older Workers — United States, 2009
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Published in MMWR. Morbidity and mortality weekly report (29.04.2011)
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Year of Publication 02.07.2024
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Retinal toxicity, in vivo and in vitro, associated with inhibition of nicotinamide phosphoribosyltransferase
Zabka, Tanja S, Singh, Jatinder, Dhawan, Preeti, Liederer, Bianca M, Oeh, Jason, Kauss, Mara A, Xiao, Yang, Zak, Mark, Lin, Tori, McCray, Bobbi, La, Nghi, Nguyen, Trung, Beyer, Joseph, Farman, Cynthia, Uppal, Hirdesh, Dragovich, Peter S, O'Brien, Thomas, Sampath, Deepak, Misner, Dinah L
Published in Toxicological sciences (01.03.2015)
Published in Toxicological sciences (01.03.2015)
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A Mild and Selective Method for the Hydrolysis of Esters with Trimethyltin Hydroxide
Nicolaou, K. C., Estrada, Anthony A., Zak, Mark, Lee, Sang Hyup, Safina, Brian S.
Published in Angewandte Chemie (International ed.) (18.02.2005)
Published in Angewandte Chemie (International ed.) (18.02.2005)
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Published in Bioorganic & medicinal chemistry letters (15.06.2019)
Published in Bioorganic & medicinal chemistry letters (15.06.2019)
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