Confirmation and Characterization of the Eccentric, Warm Jupiter TIC 393818343 b with a Network of Citizen Scientists
Sgro, Lauren A., Dalba, Paul A., Esposito, Thomas M., Marchis, Franck, Dragomir, Diana, Villanueva, Steven, Fulton, Benjamin, Billiani, Mario, Loose, Margaret, Meneghelli, Nicola, Rivett, Darren, Saibi, Fadi, Saibi, Sophie, Martin, Bryan, Lekkas, Georgios, Zaharevitz, Daniel, Zellem, Robert T., Terentev, Ivan A., Gagliano, Robert, Jacobs, Thomas Lee, Kristiansen, Martti H., LaCourse, Daryll M., Omohundro, Mark, Schwengeler, Hans M.
Published in The Astronomical journal (01.07.2024)
Published in The Astronomical journal (01.07.2024)
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A Common Pharmacophore for a Diverse Set of Colchicine Site Inhibitors Using a Structure-Based Approach
Nguyen, Tam Luong, McGrath, Connor, Hermone, Ann R, Burnett, James C, Zaharevitz, Daniel W, Day, Billy W, Wipf, Peter, Hamel, Ernest, Gussio, Rick
Published in Journal of medicinal chemistry (22.09.2005)
Published in Journal of medicinal chemistry (22.09.2005)
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A Common Pharmacophore for Epothilone and Taxanes: Molecular Basis for Drug Resistance Conferred by Tubulin Mutations in Human Cancer Cells
Giannakakou, P, Gussio, R, Nogales, E, Downing, K H, Zaharevitz, D, Bollbuck, B, Poy, G, Sackett, D, Nicolaou, K C, Fojo, T
Published in Proceedings of the National Academy of Sciences - PNAS (14.03.2000)
Published in Proceedings of the National Academy of Sciences - PNAS (14.03.2000)
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Identification of a Potent and Selective Pharmacophore for Cdc25 Dual Specificity Phosphatase Inhibitors
Lazo, John S, Nemoto, Kaoru, Pestell, Katharine E, Cooley, Kathleen, Southwick, Eileen C, Mitchell, Douglas A, Furey, William, Gussio, Rick, Zaharevitz, Daniel W, Joo, Beomjun, Wipf, Peter
Published in Molecular pharmacology (01.04.2002)
Published in Molecular pharmacology (01.04.2002)
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Paullones, a Series of Cyclin-Dependent Kinase Inhibitors: Synthesis, Evaluation of CDK1/Cyclin B Inhibition, and in Vitro Antitumor Activity
Schultz, Christiane, Link, Andreas, Leost, Maryse, Zaharevitz, Daniel W, Gussio, Rick, Sausville, Edward A, Meijer, Laurent, Kunick, Conrad
Published in Journal of medicinal chemistry (29.07.1999)
Published in Journal of medicinal chemistry (29.07.1999)
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Identification of small molecule inhibitors of anthrax lethal factor
Panchal, Rekha G, Bavari, Sina, Hermone, Ann R, Nguyen, Tam Luong, Wong, Thiang Yian, Schwarzenbacher, Robert, Schmidt, James, Lane, Douglas, McGrath, Connor, Turk, Benjamin E, Burnett, James, Aman, M Javad, Little, Stephen, Sausville, Edward A, Zaharevitz, Daniel W, Cantley, Lewis C, Liddington, Robert C, Gussio, Rick
Published in Nature structural & molecular biology (01.01.2004)
Published in Nature structural & molecular biology (01.01.2004)
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Novel small molecule inhibitors of botulinum neurotoxin A metalloprotease activity
Burnett, James C, Schmidt, James J, Stafford, Robert G, Panchal, Rekha G, Nguyen, Tam L, Hermone, Ann R, Vennerstrom, Jonathan L, McGrath, Connor F, Lane, Douglas J, Sausville, Edward A, Zaharevitz, Daniel W, Gussio, Rick, Bavari, Sina
Published in Biochemical and biophysical research communications (10.10.2003)
Published in Biochemical and biophysical research communications (10.10.2003)
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Journal Article
Homology model of RSK2 N-terminal kinase domain, structure-based identification of novel RSK2 inhibitors, and preliminary common pharmacophore
Nguyen, Tam Luong, Gussio, Rick, Smith, Jeffrey A., Lannigan, Deborah A., Hecht, Sidney M., Scudiero, Dominic A., Shoemaker, Robert H., Zaharevitz, Daniel W.
Published in Bioorganic & medicinal chemistry (01.09.2006)
Published in Bioorganic & medicinal chemistry (01.09.2006)
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Conformational sampling of the botulinum neurotoxin serotype a light chain: implications for inhibitor binding
Burnett, James C., Schmidt, James J., McGrath, Connor F., Nguyen, Tam L., Hermone, Ann R., Panchal, Rekha G., Vennerstrom, Jonathan L., Kodukula, Krishna, Zaharevitz, Daniel W., Gussio, Rick, Bavari, Sina
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Published in Bioorganic & medicinal chemistry (17.01.2005)
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2-Substituted paullones : CDK1/cyclin B-inhibiting property and in vitro antiproliferative activity
KUNICK, C, SCHULTZ, C, LEMCKE, T, ZAHAREVITZ, D. W, GUSSIO, R, JALLURI, R. K, SAUSVILLE, E. A, LEOST, M, MEIJER, L
Published in Bioorganic & medicinal chemistry letters (20.03.2000)
Published in Bioorganic & medicinal chemistry letters (20.03.2000)
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Poly(ethylene glycol) Prodrugs of the CDK Inhibitor, Alsterpaullone (NSC 705701): Synthesis and Pharmacokinetic Studies
Greenwald, Richard B, Zhao, Hong, Xia, Jing, Wu, Dechun, Nervi, Stephen, Stinson, Sherman F, Majerova, Eva, Bramhall, Chris, Zaharevitz, Daniel W
Published in Bioconjugate chemistry (01.09.2004)
Published in Bioconjugate chemistry (01.09.2004)
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A Common Pharmacophore for a Diverse Set of Colchicine Site Inhibitors Using a Structure-Based Approach
Nguyen, Tam Luong, McGrath, Connor, Hermone, Ann R, Burnett, James C, Zaharevitz, Daniel W, Day, Billy W, Wipf, Peter, Hamel, Ernest, Gussio, Rick
Published in Journal of medicinal chemistry (01.12.2005)
Published in Journal of medicinal chemistry (01.12.2005)
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Synthesis of Paullones with Aminoalkyl Side Chains
Wieking, Karen, Knockaert, Marie, Leost, Maryse, Zaharevitz, Daniel W., Meijer, Laurent, Kunick, Conrad
Published in Archiv der Pharmazie (Weinheim) (01.07.2002)
Published in Archiv der Pharmazie (Weinheim) (01.07.2002)
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The Discovery of Novel, Structurally Diverse Protein Kinase C Agonists through Computer 3D-Database Pharmacophore Search. Molecular Modeling Studies
Wang, Shaomeng, Zaharevitz, Daniel W, Sharma, Rajiv, Marquez, Victor E, Lewin, Nancy E, Du, Linh, Blumberg, Peter M, Milne, G. W. A
Published in Journal of medicinal chemistry (01.12.1994)
Published in Journal of medicinal chemistry (01.12.1994)
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All-Atom Models for the Non-Nucleoside Binding Site of HIV-1 Reverse Transcriptase Complexed with Inhibitors: A 3D QSAR Approach
Gussio, Rick, Pattabiraman, Nagarajan, Zaharevitz, Daniel W, Kellogg, Glen E, Topol, Igor A, Rice, William G, Schaeffer, Catherine A, Erickson, John W, Burt, Stanley K
Published in Journal of medicinal chemistry (12.04.1996)
Published in Journal of medicinal chemistry (12.04.1996)
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Identification of small-molecule inhibitors of the colorectal cancer oncogene Krüppel-like factor 5 expression by ultrahigh-throughput screening
Bialkowska, Agnieszka B, Crisp, Melissa, Bannister, Thomas, He, Yuanjun, Chowdhury, Sarwat, Schürer, Stephan, Chase, Peter, Spicer, Timothy, Madoux, Franck, Tian, Chenlu, Hodder, Peter, Zaharevitz, Daniel, Yang, Vincent W
Published in Molecular cancer therapeutics (01.11.2011)
Published in Molecular cancer therapeutics (01.11.2011)
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