Novel Endomorphin Analogs Are More Potent and Longer-Lasting Analgesics in Neuropathic, Inflammatory, Postoperative, and Visceral Pain Relative to Morphine
Feehan, Amy K., Morgenweck, Jenny, Zhang, Xing, Amgott-Kwan, Ariel T., Zadina, James E.
Published in The journal of pain (01.12.2017)
Published in The journal of pain (01.12.2017)
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Opioidergic projections to sleep-active neurons in the ventrolateral preoptic nucleus
Greco, Mary-Ann, Fuller, Patrick M, Jhou, Thomas C, Martin-Schild, S, Zadina, James E, Hu, Zhian, Shiromani, Priyattam, Lu, Jun
Published in Brain research (15.12.2008)
Published in Brain research (15.12.2008)
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Rewarding and Psychomotor Stimulant Effects of Endomorphin-1: Anteroposterior Differences within the Ventral Tegmental Area and Lack of Effect in Nucleus Accumbens
Zangen, Abraham, Ikemoto, Satoshi, Zadina, James E, Wise, Roy A
Published in The Journal of neuroscience (15.08.2002)
Published in The Journal of neuroscience (15.08.2002)
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Endomorphin analog analgesics with reduced abuse liability, respiratory depression, motor impairment, tolerance, and glial activation relative to morphine
Zadina, James E., Nilges, Mark R., Morgenweck, Jenny, Zhang, Xing, Hackler, Laszlo, Fasold, Melita B.
Published in Neuropharmacology (01.06.2016)
Published in Neuropharmacology (01.06.2016)
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Discriminative Stimulus and Low Abuse Liability Effects of Novel Endomorphin Analogs Suggest a Potential Treatment Indication for Opioid Use Disorder
Nilges, Mark R, Laurent, Morgan, Cable, Chloe, Arens, Louis, Vafiades, James, Zadina, James E
Published in The Journal of pharmacology and experimental therapeutics (01.09.2019)
Published in The Journal of pharmacology and experimental therapeutics (01.09.2019)
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Differential antinociceptive effects induced by intrathecally administered endomorphin-1 and endomorphin-2 in the mouse
Sakurada, Shinobu, Hayashi, Takafumi, Yuhki, Masayuki, Orito, Tohru, Zadina, James E, Kastin, Abba J, Fujimura, Tsutomu, Murayama, Kimie, Sakurada, Chikai, Sakurada, Tsukasa, Narita, Minoru, Suzuki, Tsutomu, Tan-no, Koichi, Tseng, Leon F
Published in European journal of pharmacology (21.09.2001)
Published in European journal of pharmacology (21.09.2001)
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Differential antagonism of endomorphin-1 and endomorphin-2 spinal antinociception by naloxonazine and 3-methoxynaltrexone
Sakurada, Shinobu, Hayashi, Takafumi, Yuhki, Masayuki, Fujimura, Tsutomu, Murayama, Kimie, Yonezawa, Akihiko, Sakurada, Chikai, Takeshita, Mitsuhiro, Zadina, James E., Kastin, Abba J., Sakurada, Tsukasa
Published in Brain research (20.10.2000)
Published in Brain research (20.10.2000)
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Endomorphins, Met-Enkephalin, Tyr-MIF-1, and the P-glycoprotein Efflux System
KASTIN, Abba J, FASOLD, Melita B, ZADINA, James E
Published in Drug metabolism and disposition (01.03.2002)
Published in Drug metabolism and disposition (01.03.2002)
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Journal Article
Dissociation of analgesic and rewarding effects of endomorphin-1 in rats
Wilson, Aimee M, Soignier, R.Denis, Zadina, James E, Kastin, Abba J, Nores, William L, Olson, Richard D, Olson, Gayle A
Published in Peptides (New York, N.Y. : 1980) (01.12.2000)
Published in Peptides (New York, N.Y. : 1980) (01.12.2000)
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Pleiotropic opioid regulation of spinal endomorphin 2 release and its adaptations to opioid withdrawal are sexually dimorphic
Chakrabarti, Sumita, Liu, Nai-Jiang, Zadina, James E, Sharma, Tarak, Gintzler, Alan R
Published in The Journal of pharmacology and experimental therapeutics (01.01.2012)
Published in The Journal of pharmacology and experimental therapeutics (01.01.2012)
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A potent and selective endogenous agonist for the µ-opiate receptor
Zadina, James E, Hackler, Laszlo, Ge, Lin-Jun, Kastin, Abba J
Published in Nature (London) (03.04.1997)
Published in Nature (London) (03.04.1997)
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Differential antagonism of endomorphin-1 and endomorphin-2 supraspinal antinociception by naloxonazine and 3-methylnaltrexone
Sakurada, Shinobu, Hayashi, Takafumi, Yuhki, Masayuki, Fujimura, Tsutomu, Murayama, Kimie, Yonezawa, Akihiko, Sakurada, Chikai, Takeshita, Mitsuhiro, Sato, Takumi, Zadina, James E, Kastin, Abba J, Sakurada, Tsukasa
Published in Peptides (New York, N.Y. : 1980) (01.05.2002)
Published in Peptides (New York, N.Y. : 1980) (01.05.2002)
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