Structure-Based Design of a Potent and Selective YTHDC1 Ligand
Zálešák, František, Nai, Francesco, Herok, Marcin, Bochenkova, Elena, Bedi, Rajiv K., Li, Yaozong, Errani, Francesco, Caflisch, Amedeo
Published in Journal of medicinal chemistry (13.06.2024)
Published in Journal of medicinal chemistry (13.06.2024)
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Fragment Ligands of the m6A‑RNA Reader YTHDF2
Nai, Francesco, Nachawati, Raed, Zálešák, František, Wang, Xiang, Li, Yaozong, Caflisch, Amedeo
Published in ACS medicinal chemistry letters (08.09.2022)
Published in ACS medicinal chemistry letters (08.09.2022)
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Unified Approach to Benzo[d]thiazol-2-yl-Sulfonamides
Zálešák, František, Kováč, Ondřej, Lachetová, Eliška, Št’astná, Nikola, Pospíšil, Jiří
Published in Journal of organic chemistry (03.09.2021)
Published in Journal of organic chemistry (03.09.2021)
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Heteroaryl sulfonamide synthesis: scope and limitations
Iakovenko, Roman O, Chrenko, Daniel, Kristek, Jozef, Desmedt, Eline, Zálešák, František, De Vleeschouwer, Freija, Pospíšil, Ji í
Published in Organic & biomolecular chemistry (13.04.2022)
Published in Organic & biomolecular chemistry (13.04.2022)
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Proteolysis Targeting Chimera Degraders of the METTL3–14 m6A‑RNA Methyltransferase
Errani, Francesco, Invernizzi, Annalisa, Herok, Marcin, Bochenkova, Elena, Stamm, Fiona, Corbeski, Ivan, Romanucci, Valeria, Di Fabio, Giovanni, Zálešák, František, Caflisch, Amedeo
Published in JACS Au (26.02.2024)
Published in JACS Au (26.02.2024)
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Julia‐Kocienski‐Like Connective C−C and C=C Bond‐Forming Reaction
Bon, David J.‐Y. D., Chrenko, Daniel, Kováč, Ondřej, Ferugová, Vendula, Lasák, Pavel, Fuksová, Markéta, Zálešák, František, Pospíšil, Jiří
Published in Advanced synthesis & catalysis (19.02.2024)
Published in Advanced synthesis & catalysis (19.02.2024)
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One and Two-Carbon Homologation of Primary and Secondary Alcohols to Corresponding Carboxylic Esters Using β‑Carbonyl BT Sulfones as a Common Intermediate
Bon, David J.-Y. D, Kováč, Ondřej, Ferugová, Vendula, Zálešák, František, Pospíšil, Jiří
Published in Journal of organic chemistry (04.05.2018)
Published in Journal of organic chemistry (04.05.2018)
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Trisubstituted Highly Activated Benzo[d]thiazol-2-yl-sulfone-Containing Olefins as Building Blocks in Organic Synthesis
Kovac, Ondrej, Zalesak, Frantisek, Bon, David J-Y D., Roiser, Lukas, Baar, Lubomir, Waser, Mario, Pospisil, Jiri
Published in Journal of organic chemistry (05.06.2020)
Published in Journal of organic chemistry (05.06.2020)
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Journal Article
Structure-based design of ligands of the m6A-RNA reader YTHDC1
Li, Yaozong, Bedi, Rajiv Kumar, Nai, Francesco, von Roten, Valentin, Dolbois, Aymeric, Zálešák, František, Nachawati, Raed, Huang, Danzhi, Caflisch, Amedeo
Published in European journal of medicinal chemistry reports (01.08.2022)
Published in European journal of medicinal chemistry reports (01.08.2022)
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General approach to neolignan-core of the boehmenan natural product family
Barbuscakova, Zuzana, Kozubikova, Hana, Zalesak, Frantisek, Dolezal, Karel, Pospisil, Jiri
Published in Monatshefte für Chemie (01.04.2018)
Published in Monatshefte für Chemie (01.04.2018)
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Journal Article
Fragment Ligands of the m 6 A-RNA Reader YTHDF2
Nai, Francesco, Nachawati, Raed, Zálešák, František, Wang, Xiang, Li, Yaozong, Caflisch, Amedeo
Published in ACS medicinal chemistry letters (08.09.2022)
Published in ACS medicinal chemistry letters (08.09.2022)
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Journal Article
Proteolysis Targeting Chimera Degraders of the METTL3-14 m 6 A-RNA Methyltransferase
Errani, Francesco, Invernizzi, Annalisa, Herok, Marcin, Bochenkova, Elena, Stamm, Fiona, Corbeski, Ivan, Romanucci, Valeria, Di Fabio, Giovanni, Zálešák, František, Caflisch, Amedeo
Published in JACS Au (26.02.2024)
Published in JACS Au (26.02.2024)
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Journal Article
Structure-based design of ligands of the m 6 A-RNA reader YTHDC1
Li, Yaozong, Bedi, Rajiv Kumar, Nai, Francesco, von Roten, Valentin, Dolbois, Aymeric, Zálešák, František, Nachawati, Raed, Huang, Danzhi, Caflisch, Amedeo
Published in European journal of medicinal chemistry reports (2022)
Published in European journal of medicinal chemistry reports (2022)
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Journal Article
N6-ADENOSINE-METHYLTRANSFERASE INHIBITORS IN CANCER TREATMENT
CAFLISCH, Amedeo, DOLBOIS, Aymeric, HUANG, Danzhi, ZALESAK, Frantisek
Year of Publication 02.05.2024
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Year of Publication 02.05.2024
Patent
N6-ADENOSINE-METHYLTRANSFERASE INHIBITORS IN CANCER TREATMENT
CAFLISCH, Amedeo, DOLBOIS, Aymeric, HUANG, Danzhi, ZALESAK, Frantisek
Year of Publication 27.03.2024
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Year of Publication 27.03.2024
Patent
N6-ADENOSINE-METHYLTRANSFERASE INHIBITORS IN CANCER TREATMENT
DOLBOIS, AYMERIC, HUANG, DANZHI, ZALESAK, FRANTISEK, CAFLISCH, AMEDEO
Year of Publication 24.11.2022
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Year of Publication 24.11.2022
Patent
N6-ADENOSINE-METHYLTRANSFERASE INHIBITORS IN CANCER TREATMENT
CAFLISCH, Amedeo, DOLBOIS, Aymeric, HUANG, Danzhi, ZALESAK, Frantisek
Year of Publication 24.11.2022
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Year of Publication 24.11.2022
Patent
LIGANDS OF THE M6A-RNA READERS
IVERNIZZI, Annalisa, ERRANI, Francesco, CAFLISCH, Amedeo, HEROK, Marcin, NAI, Francesco, LI, Yaozong, BEDI, Rajiv, ZALESAK, Frantisek
Year of Publication 13.11.2024
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Year of Publication 13.11.2024
Patent