Identification of a Benzoisoxazoloazepine Inhibitor (CPI-0610) of the Bromodomain and Extra-Terminal (BET) Family as a Candidate for Human Clinical Trials
Albrecht, Brian K, Gehling, Victor S, Hewitt, Michael C, Vaswani, Rishi G, Côté, Alexandre, Leblanc, Yves, Nasveschuk, Christopher G, Bellon, Steve, Bergeron, Louise, Campbell, Robert, Cantone, Nico, Cooper, Michael R, Cummings, Richard T, Jayaram, Hariharan, Joshi, Shivangi, Mertz, Jennifer A, Neiss, Adrianne, Normant, Emmanuel, O’Meara, Michael, Pardo, Eneida, Poy, Florence, Sandy, Peter, Supko, Jeffrey, Sims, Robert J, Harmange, Jean-Christophe, Taylor, Alexander M, Audia, James E
Published in Journal of medicinal chemistry (25.02.2016)
Published in Journal of medicinal chemistry (25.02.2016)
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Solvent effects on differentiation of mouse brain tissue using laser microdissection ‘cut and drop’ sampling with direct mass spectral analysis
Cahill, John F., Kertesz, Vilmos, Porta, Tiffany, LeBlanc, J.C. Yves, Heeren, Ron M.A., Van Berkel, Gary J.
Published in Rapid communications in mass spectrometry (15.03.2018)
Published in Rapid communications in mass spectrometry (15.03.2018)
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Fragment-Based Discovery of a Selective and Cell-Active Benzodiazepinone CBP/EP300 Bromodomain Inhibitor (CPI-637)
Taylor, Alexander M, Côté, Alexandre, Hewitt, Michael C, Pastor, Richard, Leblanc, Yves, Nasveschuk, Christopher G, Romero, F. Anthony, Crawford, Terry D, Cantone, Nico, Jayaram, Hariharan, Setser, Jeremy, Murray, Jeremy, Beresini, Maureen H, de Leon Boenig, Gladys, Chen, Zhongguo, Conery, Andrew R, Cummings, Richard T, Dakin, Leslie A, Flynn, E. Megan, Huang, Oscar W, Kaufman, Susan, Keller, Patricia J, Kiefer, James R, Lai, Tommy, Li, Yingjie, Liao, Jiangpeng, Liu, Wenfeng, Lu, Henry, Pardo, Eneida, Tsui, Vickie, Wang, Jian, Wang, Yongyun, Xu, Zhaowu, Yan, Fen, Yu, Dong, Zawadzke, Laura, Zhu, Xiaoqin, Zhu, Xiaoyu, Sims, Robert J, Cochran, Andrea G, Bellon, Steve, Audia, James E, Magnuson, Steven, Albrecht, Brian K
Published in ACS medicinal chemistry letters (12.05.2016)
Published in ACS medicinal chemistry letters (12.05.2016)
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Discovery, Design, and Optimization of Isoxazole Azepine BET Inhibitors
Gehling, Victor S, Hewitt, Michael C, Vaswani, Rishi G, Leblanc, Yves, Côté, Alexandre, Nasveschuk, Christopher G, Taylor, Alexander M, Harmange, Jean-Christophe, Audia, James E, Pardo, Eneida, Joshi, Shivangi, Sandy, Peter, Mertz, Jennifer A, Sims, Robert J, Bergeron, Louise, Bryant, Barbara M, Bellon, Steve, Poy, Florence, Jayaram, Hariharan, Sankaranarayanan, Ravichandran, Yellapantula, Sreegouri, Bangalore Srinivasamurthy, Nandana, Birudukota, Swarnakumari, Albrecht, Brian K
Published in ACS medicinal chemistry letters (12.09.2013)
Published in ACS medicinal chemistry letters (12.09.2013)
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Chemical Noise Reduction via Mass Spectrometry and Ion/Ion Charge Inversion: Amino Acids
Hassell, Kerry M, LeBlanc, Yves C, McLuckey, Scott A
Published in Analytical chemistry (Washington) (01.05.2011)
Published in Analytical chemistry (Washington) (01.05.2011)
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Discovery of Benzotriazolo[4,3‑d][1,4]diazepines as Orally Active Inhibitors of BET Bromodomains
Taylor, Alexander M, Vaswani, Rishi G, Gehling, Victor S, Hewitt, Michael C, Leblanc, Yves, Audia, James E, Bellon, Steve, Cummings, Richard T, Côté, Alexandre, Harmange, Jean-Christophe, Jayaram, Hari, Joshi, Shivangi, Lora, Jose M, Mertz, Jennifer A, Neiss, Adrianne, Pardo, Eneida, Nasveschuk, Christopher G, Poy, Florence, Sandy, Peter, Setser, Jeremy W, Sims, Robert J, Tang, Yong, Albrecht, Brian K
Published in ACS medicinal chemistry letters (11.02.2016)
Published in ACS medicinal chemistry letters (11.02.2016)
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Kinetic Size-Exclusion Chromatography with Mass Spectrometry Detection: An Approach for Solution-Based Label-Free Kinetic Analysis of Protein–Small Molecule Interactions
Bao, Jiayin, Krylova, Svetlana M, Cherney, Leonid T, LeBlanc, J. C. Yves, Pribil, Patrick, Johnson, Philip E, Wilson, Derek J, Krylov, Sergey N
Published in Analytical chemistry (Washington) (21.10.2014)
Published in Analytical chemistry (Washington) (21.10.2014)
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Identification of prostaglandin D2 receptor antagonists based on a tetrahydropyridoindole scaffold
BEAULIEU, Christian, GUAY, Daniel, DENIS, Danielle, GREIG, Gillian, MATHIEU, Marie-Claude, O'NEILL, Gary, ZHAOYIN WANG, LEBLANC, Yves, ROY, Patrick, DUFRESNE, Claude, ZAMBONI, Robert, BERTHELETTE, Carl, DAY, Stephen, TSOU, Nancy
Published in Bioorganic & medicinal chemistry letters (15.04.2008)
Published in Bioorganic & medicinal chemistry letters (15.04.2008)
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Conformation-assisted Inhibition of Protein-tyrosine Phosphatase-1B Elicits Inhibitor Selectivity over T-cell Protein-tyrosine Phosphatase
Asante-Appiah, Ernest, Patel, Sangita, Desponts, Caroline, Taylor, Jillian M., Lau, Cheuk, Dufresne, Claude, Therien, Michel, Friesen, Rick, Becker, Joseph W., Leblanc, Yves, Kennedy, Brian P., Scapin, Giovanna
Published in The Journal of biological chemistry (24.03.2006)
Published in The Journal of biological chemistry (24.03.2006)
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The development of potent non-peptidic PTP-1B inhibitors
DUFRESNE, Claude, ROY, Patrick, WADDLETON, Deena, RAMACHANDRAN, Chidambaram, KENNEDY, Brian P, LIJING XU, GORDON, Robert, CHI CHUNG CHAN, LEBLANC, Yves, ZHAOYIN WANG, ASANTE-APPIAH, Ernest, CROMLISH, Wanda, BOIE, Yves, FORGHANI, Farnaz, DESMARAIS, Sylvie, QINGPING WANG, SKOREY, Kathryn
Published in Bioorganic & medicinal chemistry letters (23.02.2004)
Published in Bioorganic & medicinal chemistry letters (23.02.2004)
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Modeling of Groundwater Flow and Drawdown Evolution Simulation of Abidjan Aquifer (Cote D'ivoire)
Jean, Kouame Kan, Patrice, Jourda Jean, Bachir, Saley Mahaman, Kouakou, Deh Serges, Tawa, Anani Abenan, Yves, Leblanc, Vincent, Cloutier, Jean, Biemi
Published in Journal of Asian scientific research (Online) (01.04.2013)
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Published in Journal of Asian scientific research (Online) (01.04.2013)
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Scout-multiple reaction monitoring: A liquid chromatography tandem mass spectrometry approach for multi-residue pesticide analysis without time scheduling
Salvador, Arnaud, Carrière, Romain, Ayciriex, Sophie, Margoum, Christelle, Leblanc, Yves, Lemoine, Jérôme
Published in Journal of Chromatography A (21.06.2020)
Published in Journal of Chromatography A (21.06.2020)
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Determination of Pentachlorophenol and Its Oil Solvent in Wood Pole Samples by SFE and GC with Postcolumn Flow Splitting for Simultaneous Detection of the Species
Leblanc, Yves G, Gilbert, Roland, Hubert, Joseph
Published in Analytical chemistry (Washington) (01.01.1999)
Published in Analytical chemistry (Washington) (01.01.1999)
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Detection of Opioids on Mail/Packages Using Open Port Interface Mass Spectrometry (OPI-MS)
Metwally, Haidy, Agrawal, Prashant, Smith, Rachael, Liu, Chang, LeBlanc, Yves, Covey, Thomas R, Oleschuk, Richard
Published in Journal of the American Society for Mass Spectrometry (04.11.2020)
Published in Journal of the American Society for Mass Spectrometry (04.11.2020)
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SpectraX: A Straightforward Tool for Principal Component Analysis-Based Spectral Analysis
Yu, Jian, Metwally, Haidy, Kolwich, Jennifer, Tomm, Hailey, Klotz, Rachel, Liu, Chang, LeBlanc, J. C. Yves, Covey, Thomas R., Ross, Avena C., Oleschuk, Richard D.
Published in Journal of the American Society for Mass Spectrometry (07.02.2024)
Published in Journal of the American Society for Mass Spectrometry (07.02.2024)
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Synthesis and biological evaluation of 2,3-diarylthiophenes as selective Cox-2 and Cox-1 inhibitors
Leblanc, Yves, Gauthier, JacquesYves, Ethier, Diane, Guay, Jocelyne, Mancini, Joseph, Riendeau, Denis, Tagari, Philip, Vickers, Philip, Wong, Elizabeth, Prasit, Petpiboon
Published in Bioorganic & medicinal chemistry letters (21.09.1995)
Published in Bioorganic & medicinal chemistry letters (21.09.1995)
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The Integrated Psychological Treatment for Individuals With Schizophrenia in Correctional and Forensic Psychiatric Settings: An Implementation Study
Dumont, Mathieu, Briand, Catherine, Leblanc, Yves, Aubin, Ginette, Potvin, Stéphane, Dumais, Alexandre
Published in International journal of offender therapy and comparative criminology (01.07.2020)
Published in International journal of offender therapy and comparative criminology (01.07.2020)
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Integrating community-based nonprofit organizations into the cancer care journey: how do connections and coordination take shape?
Tremblay, Dominique, Usher, Susan, Gentil, Barbara, Courval, Marie-Josée, Leblanc, Yves, Cournoyer, Johanne
Published in International journal of integrated care (04.11.2022)
Published in International journal of integrated care (04.11.2022)
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