Discovery of Orally Active Inhibitors of Brahma Homolog (BRM)/SMARCA2 ATPase Activity for the Treatment of Brahma Related Gene 1 (BRG1)/SMARCA4-Mutant Cancers
Papillon, Julien P. N, Nakajima, Katsumasa, Adair, Christopher D, Hempel, Jonathan, Jouk, Andriana O, Karki, Rajeshri G, Mathieu, Simon, Möbitz, Henrik, Ntaganda, Rukundo, Smith, Troy, Visser, Michael, Hill, Susan E, Hurtado, Felipe Kellermann, Chenail, Gregg, Bhang, Hyo-Eun C, Bric, Anka, Xiang, Kay, Bushold, Geoffrey, Gilbert, Tamara, Vattay, Anthony, Dooley, Julie, Costa, Emily A, Park, Isabel, Li, Ailing, Farley, David, Lounkine, Eugen, Yue, Q. Kimberley, Xie, Xiaoling, Zhu, Xiaoping, Kulathila, Raviraj, King, Daniel, Hu, Tiancen, Vulic, Katarina, Cantwell, John, Luu, Catherine, Jagani, Zainab
Published in Journal of medicinal chemistry (21.11.2018)
Published in Journal of medicinal chemistry (21.11.2018)
Get full text
Journal Article
Discovery and Characterization of Allosteric WNK Kinase Inhibitors
Yamada, Ken, Zhang, Ji-Hu, Xie, Xiaoling, Reinhardt, Juergen, Xie, Amy Qiongshu, LaSala, Daniel, Kohls, Darcy, Yowe, David, Burdick, Debra, Yoshisue, Hajime, Wakai, Hiromichi, Schmidt, Isabel, Gunawan, Jason, Yasoshima, Kayo, Yue, Q. Kimberley, Kato, Mitsunori, Mogi, Muneto, Idamakanti, Neeraja, Kreder, Natasha, Drueckes, Peter, Pandey, Pramod, Kawanami, Toshio, Huang, Waanjeng, Yagi, Yukiko I, Deng, Zhan, Park, Hyi-Man
Published in ACS chemical biology (16.12.2016)
Published in ACS chemical biology (16.12.2016)
Get full text
Journal Article
Reporter Enzyme Inhibitor Study To Aid Assembly of Orthogonal Reporter Gene Assays
Ho, Pei-i, Yue, Kimberley, Pandey, Pramod, Breault, Lyne, Harbinski, Fred, McBride, Aaron J, Webb, Brian, Narahari, Janaki, Karassina, Natasha, Wood, Keith V, Hill, Adam, Auld, Douglas S
Published in ACS chemical biology (17.05.2013)
Published in ACS chemical biology (17.05.2013)
Get full text
Journal Article
Identifying initiation and elongation inhibitors of dengue virus RNA polymerase in a high-throughput lead-finding campaign
Smith, Thomas M, Lim, Siew Pheng, Yue, Kimberley, Busby, Scott A, Arora, Rishi, Seh, Cheah Chen, Wright, S Kirk, Nutiu, Razvan, Niyomrattanakit, Pornwaratt, Wan, Kah Fei, Beer, David, Shi, Pei-Yong, Benson, Timothy E
Published in Journal of biomolecular screening (01.01.2015)
Published in Journal of biomolecular screening (01.01.2015)
Get full text
Journal Article
Oxygen Access to the Active Site of Cholesterol Oxidase through a Narrow Channel Is Gated by an Arg-Glu Pair
Coulombe, R, Yue, K Q, Ghisla, S, Vrielink, A
Published in The Journal of biological chemistry (10.08.2001)
Published in The Journal of biological chemistry (10.08.2001)
Get full text
Journal Article
Two RNA Tunnel Inhibitors Bind in Highly Conserved Sites in Dengue Virus NS5 Polymerase: Structural and Functional Studies
Arora, Rishi, Liew, Chong Wai, Soh, Tingjin Sherryl, Otoo, Dorcas Adobea, Seh, Cheah Chen, Yue, Kimberley, Nilar, Shahul, Wang, Gang, Yokokawa, Fumiaki, Noble, Christian G, Chen, Yen Liang, Shi, Pei-Yong, Lescar, Julien, Smith, Thomas M, Benson, Timothy E, Lim, Siew Pheng
Published in Journal of virology (23.11.2020)
Published in Journal of virology (23.11.2020)
Get full text
Journal Article
Matrix-Based Activity Pattern Classification as a Novel Method for the Characterization of Enzyme Inhibitors Derived from High-Throughput Screening
Auld, Douglas S, Jimenez, Marta, Yue, Kimberley, Busby, Scott, Chen, Yu-Chi, Bowes, Scott, Wendel, Greg, Smith, Thomas, Zhang, Ji-Hu
Published in Journal of biomolecular screening (01.12.2016)
Published in Journal of biomolecular screening (01.12.2016)
Get full text
Journal Article
Drug-induced hypersensitivity syndrome in pediatric patients
Carroll, M C, Yueng-Yue, K A, Esterly, N B, Drolet, B A
Published in Pediatrics (Evanston) (01.08.2001)
Published in Pediatrics (Evanston) (01.08.2001)
Get more information
Journal Article