Three-Dimensional Quantitative Structure−Activity Relationships of Cyclo-oxygenase-2 (COX-2) Inhibitors: A Comparative Molecular Field Analysis
Chavatte, Philippe, Yous, Saïd, Marot, Christophe, Baurin, Nicolas, Lesieur, Daniel
Published in Journal of medicinal chemistry (27.09.2001)
Published in Journal of medicinal chemistry (27.09.2001)
Get full text
Journal Article
Determination of ionization constants of N-imidazole derivatives, aromatase inhibitors, using capillary electrophoresis and influence of substituents on pKa shifts
FOULON, C, DANEL, C, VACCHER, C, YOUS, S, BONTE, J.-P, GOOSSENS, J.-F
Published in Journal of Chromatography A (30.04.2004)
Published in Journal of Chromatography A (30.04.2004)
Get full text
Journal Article
Antioxidant activity of melatonin and a pinoline derivative on linoleate model system
Mekhloufi, J., Bonnefont-Rousselot, D., Yous, S., Lesieur, D., Couturier, M., Thérond, P., Legrand, A., Jore, D., Gardès-Albert, M.
Published in Journal of pineal research (01.08.2005)
Published in Journal of pineal research (01.08.2005)
Get full text
Journal Article
Novel naphthalenic ligands with high affinity for the melatonin receptor
Yous, S, Andrieux, J, Howell, H. E, Morgan, P. J, Renard, P, Pfeiffer, B, Lesieur, D, Guardiola-Lemaitre, B
Published in Journal of medicinal chemistry (01.04.1992)
Published in Journal of medicinal chemistry (01.04.1992)
Get full text
Journal Article
Exposure to glycol ethers in a population of French men evaluated by measurement of urinary alkoxycarboxylic acids
BEN-BRIK, E, JEROME, L, ARNAUD, I, YOUS, S, LABAT, L, HAGUENOER, J. M, MULTIGNER, Luc
Published in International archives of occupational and environmental health (01.06.2004)
Published in International archives of occupational and environmental health (01.06.2004)
Get full text
Journal Article
Chiral resolution of the enantiomers of new aromatase inhibitors by liquid chromatography on amylose stationary phases
DANEL, C, FOULON, C, PARK, C, YOUS, S, BONTE, J.-P, VACCHER, C
Published in Chromatographia (01.02.2004)
Published in Chromatographia (01.02.2004)
Get full text
Journal Article
Synthesis and Evaluation of Benzoxazolinonic Imidazoles and Derivatives as Non-steroidal Aromatase Inhibitors
Nativelle-Serpentini, Celine, Moslemi, Safa, Yous, Said, Ha Park, Chang, Lesieur, Daniel, Sourdaine, Pascal, Séralini, Gilles-Eric
Published in Journal of enzyme inhibition and medicinal chemistry (01.04.2004)
Published in Journal of enzyme inhibition and medicinal chemistry (01.04.2004)
Get full text
Journal Article
Synthesis of 6-Cycloalkyl-2(3H)-benzoxazolones and Benzoxathiazolones via 6-Tri-N-butyltin Intermediates
Carato, P., Moussavi, Z., Yous, S., Poupaert, J.-H., Lebegue, N., Berthelot, P.
Published in Synthetic communications (01.01.2004)
Published in Synthetic communications (01.01.2004)
Get full text
Journal Article
Direct separation of the stereoisomers of methoxytetrahydronaphthalene derivatives, new agonist and antagonist ligands for melatonin receptors, by liquid chromatography on cellulose chiral stationary phases
Belloli, E., Foulon, C., Yous, S., Vaccher, M.-P., Bonte, J.-P., Vaccher, C.
Published in Journal of Chromatography A (12.01.2001)
Published in Journal of Chromatography A (12.01.2001)
Get full text
Journal Article
Design, Synthesis and In Vitro Evaluation of Novel Benzo[b]thiophene Derivatives as Serotonin N-acetyltransferase (AANAT) Inhibitors
Mesangeau, C., Yous, S., Chavatte, P., Ferry, G., Audinot, V., Boutin, J.A., Delagrange, P., Bennejean, C., Renard, P., Lesieur, D.
Published in Journal of enzyme inhibition and medicinal chemistry (01.04.2003)
Published in Journal of enzyme inhibition and medicinal chemistry (01.04.2003)
Get full text
Journal Article
Design, Synthesis and In Vitro Evaluation of Novel Derivatives as Serotonin N -Acetyltransferase Inhibitors
Beaurain, N., Mésangeau, C., Chavatte, P., Ferry, G., Audinot, V., Boutin, J.A., Delagrange, P., Bennejean, C., Yous, S.
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2002)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2002)
Get full text
Journal Article
Conformational analysis of tripeptide Ac-Lys-Pro-Val-NH2, COOH-terminal sequence of alpha-MSH
Chavatte, P, Yous, S, Lesieur, D, Hénichart, J P
Published in Journal of pharmacy and pharmacology (01.07.2001)
Published in Journal of pharmacy and pharmacology (01.07.2001)
Get more information
Journal Article
2(3H)-Benzoxazolone and Bioisosters as "Privileged Scaffold" in the Design of Pharmacological Probes
POUPAERT, Jacques, CARATO, Pascal, COLACINO, Evelina
Published in Current medicinal chemistry (01.01.2005)
Published in Current medicinal chemistry (01.01.2005)
Get full text
Journal Article
Synthesis of 2(3H)-benzoxazolinone derivatives as potential beta-3-adrenergic receptor ligands
Delhomel, JF, Yous, S, Depreux, P, Lesieur, D
Published in Journal of heterocyclic chemistry (01.09.1999)
Published in Journal of heterocyclic chemistry (01.09.1999)
Get more information
Journal Article
Rexinoid Bexarotene Modulates Triglyceride but not Cholesterol Metabolism via Gene-Specific Permissivity of the RXR/LXR Heterodimer in the Liver
Lalloyer, Fanny, Pedersen, Thomas Åskov, Gross, Barbara, Lestavel, Sophie, Yous, Saïd, Vallez, Emmanuelle, Gustafsson, Jan-Åke, Mandrup, Susanne, Fiévet, Catherine, Staels, Bart, Tailleux, Anne
Published in Arteriosclerosis, thrombosis, and vascular biology (01.10.2009)
Published in Arteriosclerosis, thrombosis, and vascular biology (01.10.2009)
Get full text
Journal Article
Characterization of the melatoninergic MT3 binding site on the NRH:quinone oxidoreductase 2 enzyme
MAILLIET, Francois, FERRY, Gilles, YOUS, Said, DELAGRANGE, Philippe, BOUTIN, Jean A, VELLA, Fanny, BERGER, Syluie, COGE, Francis, CHOMARAT, Pascale, MALLET, Catherine, GUENIN, Sophie-Pénélope, GUILLAUMET, Gérald, VIAUD-MASSUARD, Marie-Claude
Published in Biochemical pharmacology (19.12.2005)
Published in Biochemical pharmacology (19.12.2005)
Get full text
Journal Article
New radioligands for describing the molecular pharmacology of MT1 and MT2 melatonin receptors
Legros, Céline, Matthey, Ulrich, Grelak, Teresa, Pedragona-Moreau, Sandrine, Hassler, Werner, Yous, Saïd, Thomas, Emmanuel, Suzenet, Franck, Folleas, Benoît, Lefoulon, François, Berthelot, Pascal, Caignard, Daniel-Henri, Guillaumet, Gérald, Delagrange, Philippe, Brayer, Jean-Louis, Nosjean, Olivier, Boutin, Jean A
Published in International journal of molecular sciences (25.04.2013)
Published in International journal of molecular sciences (25.04.2013)
Get full text
Journal Article
The RXR Agonist Bexarotene Improves Cholesterol Homeostasis and Inhibits Atherosclerosis Progression in a Mouse Model of Mixed Dyslipidemia
Lalloyer, Fanny, Fiévet, Catherine, Lestavel, Sophie, Torpier, Gérard, van der Veen, Jelske, Touche, Véronique, Bultel, Stéphanie, Yous, Saïd, Kuipers, Folkert, Paumelle, Réjane, Fruchart, Jean-Charles, Staels, Bart, Tailleux, Anne
Published in Arteriosclerosis, thrombosis, and vascular biology (01.12.2006)
Published in Arteriosclerosis, thrombosis, and vascular biology (01.12.2006)
Get full text
Journal Article
Pictet–Spengler heterocyclizations via microwave-assisted degradation of DMSO
Mésangeau, Christophe, Yous, Saïd, Pérès, Basile, Lesieur, Daniel, Besson, Thierry
Published in Tetrahedron letters (04.04.2005)
Published in Tetrahedron letters (04.04.2005)
Get full text
Journal Article