Repeat oral dosing of prasugrel, a novel P2Y12 receptor inhibitor, results in cumulative and potent antiplatelet and antithrombotic activity in several animal species
NIITSU, Yoichi, SUGIDACHI, Atsuhiro, OGAWA, Taketoshi, JAKUBOWSKI, Joseph A, HASHIMOTO, Masami, ISOBE, Takashi, OTSUGURO, Ken-Ichi, ASAI, Fumitoshi
Published in European journal of pharmacology (28.01.2008)
Published in European journal of pharmacology (28.01.2008)
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Journal Article
Selective blockade of P2Y12 receptors by prasugrel inhibits myocardial infarction induced by thrombotic coronary artery occlusion in rats
Sugidachi, Atsuhiro, Yamaguchi, Shinji, Jakubowski, Joseph A, Ohno, Kosaku, Tomizawa, Atsuyuki, Hashimoto, Masami, Niitsu, Yoichi
Published in Journal of cardiovascular pharmacology (01.09.2011)
Published in Journal of cardiovascular pharmacology (01.09.2011)
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Journal Article
The influence of P2Y12 receptor deficiency on the platelet inhibitory activities of prasugrel in a mouse model: Evidence for specific inhibition of P2Y12 receptors by prasugrel
Hashimoto, Masami, Sugidachi, Atsuhiro, Isobe, Takashi, Niitsu, Yoichi, Ogawa, Taketoshi, Jakubowski, Joseph A., Asai, Fumitoshi
Published in Biochemical pharmacology (01.10.2007)
Published in Biochemical pharmacology (01.10.2007)
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Journal Article
Effects of prasugrel, a novel P2Y12 inhibitor, in rat models of cerebral and peripheral artery occlusive diseases
OGAWA, Taketoshi, HASHIMOTO, Masami, NIITSU, Yoichi, JAKUBOWSKI, Joseph A, TANI, Yoshiro, OTSUGURO, Ken-Ichi, ASAI, Fumitoshi, SUGIDACHI, Atsuhiro
Published in European journal of pharmacology (01.06.2009)
Published in European journal of pharmacology (01.06.2009)
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Journal Article
Discovery of R-142086 as a Factor Xa (FXa) Inhibitor: Syntheses and Structure–Activity Relationships of Cinnamyl Derivatives
Noguchi, Tetsuji, Tanaka, Naoki, Nishimata, Toyoki, Goto, Riki, Hayakawa, Miho, Sugidachi, Atsuhiro, Ogawa, Taketoshi, Niitsu, Yoichi, Asai, Fumitoshi, Ishizuka, Tomoko, Fujimoto, Koichi
Published in Chemical & pharmaceutical bulletin (01.01.2009)
Published in Chemical & pharmaceutical bulletin (01.01.2009)
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Journal Article
Discovery of DS-1093a: An oral hypoxia-inducible factor prolyl hydroxylase inhibitor for the treatment of renal anemia
Tanaka, Naoki, Fukuda, Takeshi, Takano, Rieko, Sasaki, Koji, Tsuji, Takashi, Goto, Riki, Kuribayashi, Takeshi, Yamaguchi, Kyoji, Niitsu, Yoichi, Ishii, Ken, Hashimoto, Masami, Takahashi, Shinichi, Obayashi, Hisakuni
Published in Bioorganic & medicinal chemistry letters (01.10.2024)
Published in Bioorganic & medicinal chemistry letters (01.10.2024)
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Journal Article
Discovery of DS44470011: An oral hypoxia-inducible factor prolyl hydroxylase inhibitor for the treatment of renal anemia
Fukuda, Takeshi, Kuribayashi, Takeshi, Takano, Rieko, Sasaki, Koji, Tsuji, Takashi, Niitsu, Yoichi, Ishii, Ken, Hashimoto, Masami, Baba, Daichi, Ito, Shuichiro, Tanaka, Naoki
Published in Bioorganic & medicinal chemistry letters (01.08.2024)
Published in Bioorganic & medicinal chemistry letters (01.08.2024)
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Journal Article
Pharmacology of CS-747 (prasugrel, LY640315), a novel, potent antiplatelet agent with in vivo P2Y12 receptor antagonist activity
Niitsu, Yoichi, Jakubowski, Joseph A, Sugidachi, Atsuhiro, Asai, Fumitoshi
Published in Seminars in thrombosis and hemostasis (01.04.2005)
Published in Seminars in thrombosis and hemostasis (01.04.2005)
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Ministrokes in channelrhodopsin-2 transgenic mice reveal widespread deficits in motor output despite maintenance of cortical neuronal excitability
Anenberg, Eitan, Arstikaitis, Pamela, Niitsu, Yoichi, Harrison, Thomas C, Boyd, Jamie D, Hilton, Brett J, Tetzlaff, Wolfram, Murphy, Timothy H
Published in The Journal of neuroscience (22.01.2014)
Published in The Journal of neuroscience (22.01.2014)
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Journal Article
Effects of prasugrel, a novel P2Y(12) inhibitor, in rat models of cerebral and peripheral artery occlusive diseases
Ogawa, Taketoshi, Hashimoto, Masami, Niitsu, Yoichi, Jakubowski, Joseph A, Tani, Yoshiro, Otsuguro, Ken-Ichi, Asai, Fumitoshi, Sugidachi, Atsuhiro
Published in European journal of pharmacology (10.06.2009)
Published in European journal of pharmacology (10.06.2009)
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Journal Article
Effects of prasugrel, a novel P2Y sub(12) inhibitor, in rat models of cerebral and peripheral artery
Ogawa, Taketoshi, Hashimoto, Masami, Niitsu, Yoichi, Jakubowski, Joseph A, Tani, Yoshiro, Otsuguro, Ken-Ichi, Asai, Fumitoshi, Sugidachi, Atsuhiro
Published in European journal of pharmacology (01.06.2009)
Published in European journal of pharmacology (01.06.2009)
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Journal Article
Effects of prasugrel, a novel P2Y 12 inhibitor, in rat models of cerebral and peripheral artery occlusive diseases
Ogawa, Taketoshi, Hashimoto, Masami, Niitsu, Yoichi, Jakubowski, Joseph A., Tani, Yoshiro, Otsuguro, Ken-ichi, Asai, Fumitoshi, Sugidachi, Atsuhiro
Published in European journal of pharmacology (2009)
Published in European journal of pharmacology (2009)
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Journal Article
Evaluation of MCAO stroke models in normotensive rats: standardized neocortical infarction by the 3VO technique
Yanamoto, Hiroji, Nagata, Izumi, Niitsu, Yoichi, Xue, Jing-Hui, Zhang, Zhiwen, Kikuchi, Haruhiko
Published in Experimental Neurology (01.08.2003)
Published in Experimental Neurology (01.08.2003)
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Journal Article
Repeat oral dosing of prasugrel, a novel P2Y 12 receptor inhibitor, results in cumulative and potent antiplatelet and antithrombotic activity in several animal species
Niitsu, Yoichi, Sugidachi, Atsuhiro, Ogawa, Taketoshi, Jakubowski, Joseph A., Hashimoto, Masami, Isobe, Takashi, Otsuguro, Ken-ichi, Asai, Fumitoshi
Published in European journal of pharmacology (2008)
Published in European journal of pharmacology (2008)
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Journal Article
Discovery of R-142086 as a Factor Xa (FXa) Inhibitor
Noguchi, Tetsuji, Tanaka, Naoki, Nishimata, Toyoki, Goto, Riki, Hayakawa, Miho, Sugidachi, Atsuhiro, Ogawa, Taketoshi, Niitsu, Yoichi, Asai, Fumitoshi, Ishizuka, Tomoko, Fujimoto, Koichi
Published in Chemical & pharmaceutical bulletin (01.01.2009)
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Published in Chemical & pharmaceutical bulletin (01.01.2009)
Journal Article
Prasugrel (CS-747, LY640315) Hydrochloride, a Novel Thienopyridine Prodrug, Shows Potent Antiplatelet and Antithrombotic Effects with Rapid Onset of Action in Rats
Niitsu, Yoichi, Ogawa, Taketoshi, Sugidachi, Atsuhiro, Jakubowski, Joseph A., Yokouchi, Yuki, Kakusaka, Mayumi, Hasegawa, Michihiro, Asai, Fumitoshi
Published in Blood (16.11.2005)
Published in Blood (16.11.2005)
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