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Published in The Journal of biological chemistry (03.06.1994)
Published in The Journal of biological chemistry (03.06.1994)
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Gamma-aminobutyric acid type B receptors with specific heterodimer composition and postsynaptic actions in hippocampal neurons are targets of anticonvulsant gabapentin action
Ng, G Y, Bertrand, S, Sullivan, R, Ethier, N, Wang, J, Yergey, J, Belley, M, Trimble, L, Bateman, K, Alder, L, Smith, A, McKernan, R, Metters, K, O'Neill, G P, Lacaille, J C, Hébert, T E
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Published in Molecular pharmacology (01.01.2001)
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Quinolinic acid in cerebrospinal fluid and serum in HIV-1 infection: relationship to clinical and neurological status
Heyes, M P, Brew, B J, Martin, A, Price, R W, Salazar, A M, Sidtis, J J, Yergey, J A, Mouradian, M M, Sadler, A E, Keilp, J
Published in Annals of neurology (01.02.1991)
Published in Annals of neurology (01.02.1991)
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Description of a 96-Well Plate Assay to Measure Cytochrome P4503A Inhibition in Human Liver Microsomes Using a Selective Fluorescent Probe
Chauret, Nathalie, Tremblay, Nathalie, Lackman, Rebecca L., Gauthier, Jacques-Yves, Silva, José M., Marois, Jean, Yergey, James A., Nicoll-Griffith, Deborah A.
Published in Analytical biochemistry (15.12.1999)
Published in Analytical biochemistry (15.12.1999)
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Refinement of an in Vitro Cell Model for Cytochrome P450 Induction
SILVA, J. M, MORIN, P. E, DAY, S. H, KENNEDY, B. P, PAYETTE, P, RUSHMORE, T, YERGEY, J. A, NICOLL-GRIFFITH, D. A
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Published in Drug metabolism and disposition (01.05.1998)
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Overexpression of human prostaglandin G/H synthase-1 and -2 by recombinant vaccinia virus: inhibition by nonsteroidal anti-inflammatory drugs and biosynthesis of 15-hydroxyeicosatetraenoic acid
O'Neill, G P, Mancini, J A, Kargman, S, Yergey, J, Kwan, M Y, Falgueyret, J P, Abramovitz, M, Kennedy, B P, Ouellet, M, Cromlish, W
Published in Molecular pharmacology (01.02.1994)
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Published in Molecular pharmacology (01.02.1994)
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Mechanism of selective inhibition of human prostaglandin G/H synthase-1 and -2 in intact cells
Kargman, Stacia, Wong, Elizabeth, Greig, Gillian M., Falgueyret, Jean-Pierre, Cromlish, Wanda, Ethier, Diane, Yergey, Jim A., Riendeau, Denis, Evans, Jilly F., Kennedy, Brian, Tagari, Philip, Francis, Donna A., O'Neill, Gary P.
Published in Biochemical pharmacology (11.10.1996)
Published in Biochemical pharmacology (11.10.1996)
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Investigation of the in Vitro Metabolism Profile of a Phosphodiesterase-IV Inhibitor, CDP-840: Leading to Structural Optimization
Li, C, Chauret, N, Trimble, L A, Nicoll-Griffith, D A, Silva, J M, MacDonald, D, Perrier, H, Yergey, J A, Parton, T, Alexander, R P, Warrellow, G J
Published in Drug metabolism and disposition (01.03.2001)
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Published in Drug metabolism and disposition (01.03.2001)
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Enzyme kinetics of cytochrome P450-mediated reactions
Shou, M, Lin, Y, Lu, P, Tang, C, Mei, Q, Cui, D, Tang, W, Ngui, J S, Lin, C C, Singh, R, Wong, B K, Yergey, J A, Lin, J H, Pearson, P G, Baillie, T A, Rodrigues, A D, Rushmore, T H
Published in Current drug metabolism (01.03.2001)
Published in Current drug metabolism (01.03.2001)
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Microsomal metabolism of the 5-lipoxygenase inhibitors L-746,530 and L-739,010 to reactive intermediates that covalently bind to protein: the role of the 6,8-dioxabicyclo[3.2.1]octanyl moiety
Chauret, N, Nicoll-Griffith, D, Friesen, R, Li, C, Trimble, L, Dubé, D, Fortin, R, Girard, Y, Yergey, J
Published in Drug metabolism and disposition (01.12.1995)
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Published in Drug metabolism and disposition (01.12.1995)
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Dioxabicyclooctanyl Naphthalenenitriles as Nonredox 5-Lipoxygenase Inhibitors: Structure−Activity Relationship Study Directed toward the Improvement of Metabolic Stability
Delorme, Daniel, Ducharme, Yves, Brideau, Christine, Chan, Chi-Chung, Chauret, Nathalie, Desmarais, Sylvie, Dubé, Daniel, Falgueyret, Jean-Pierre, Fortin, Réjean, Guay, Jocelyne, Hamel, Pierre, Jones, Tom R, Lépine, Carole, Li, Chun, McAuliffe, Malia, McFarlane, Cyril S, Nicoll-Griffith, Deborah A, Riendeau, Denis, Yergey, James A, Girard, Yves
Published in Journal of medicinal chemistry (27.09.1996)
Published in Journal of medicinal chemistry (27.09.1996)
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In vitro metabolism considerations, including activity testing of metabolites, in the discovery and selection of the COX-2 inhibitor etoricoxib (MK-0663)
Chauret, Nathalie, Yergey, James A, Brideau, Christine, Friesen, Richard W, Mancini, Joseph, Riendeau, Denis, Silva, José, Styhler, Angela, Trimble, Laird A, Nicoll-Griffith, Deborah A
Published in Bioorganic & medicinal chemistry letters (23.04.2001)
Published in Bioorganic & medicinal chemistry letters (23.04.2001)
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Mass spectrometric analysis of arachidonyl-containing phospholipids in human U937 cells
Li, Chun, McClory, Andrew, Wong, Elizabeth, Yergey, James A.
Published in Journal of mass spectrometry. (01.05.1999)
Published in Journal of mass spectrometry. (01.05.1999)
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In vitro and in vivo biotransformations of the naphthalenic lignan lactone 5-lipoxygenase inhibitor, L-702,539
Chauret, N, Li, C, Ducharme, Y, Trimble, L A, Yergey, J A, Ramachandran, C, Nicoll-Griffith, D A
Published in Drug metabolism and disposition (01.01.1995)
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Published in Drug metabolism and disposition (01.01.1995)
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Oxidative Bioactivation of the Lactol Prodrug of A Lactone Cyclooxygenase-2 Inhibitor
NICOLL-GRIFFITH, D. A, FALGUEYRET, J.-P, RIENDEAU, D, SILVA, J. M, MORIN, P.-E, TRIMBLE, L, CHAN, C.-C, CLAS, S, LEGER, S, ZHAOYIN WANG, YERGEY, J. A
Published in Drug metabolism and disposition (01.03.1999)
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Published in Drug metabolism and disposition (01.03.1999)
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Characterization of verlukast metabolites arising from an epoxide intermediate produced with hepatic microsomes from beta-naphthoflavone-treated rodents (P-4501A1)
Nicoll-Griffith, D A, Chauret, N, Yergey, J A, Trimble, L A, Favreau, L, Zamboni, R, Grossman, S J, Drey, J, Herold, E
Published in Drug metabolism and disposition (01.09.1993)
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Published in Drug metabolism and disposition (01.09.1993)
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Synthesis, characterization, and activity of metabolites derived from the cyclooxygenase-2 inhibitor rofecoxib (MK-0966, Vioxx ™)
Nicoll-Griffith, Deborah A, Yergey, James A, Trimble, Laird A, Silva, José M, Li, Chun, Chauret, Nathalie, Gauthier, Jacques Yves, Grimm, Erich, Léger, Serge, Roy, Patrick, Thérien, Michel, Wang, Zhaoyin, Prasit, Peppi, Zamboni, Robert, Young, Robert N, Brideau, Christine, Chan, Chi-Chung, Mancini, Joseph, Riendeau, Denis
Published in Bioorganic & medicinal chemistry letters (04.12.2000)
Published in Bioorganic & medicinal chemistry letters (04.12.2000)
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Integrated Application of Capillary HPLC/Continuous-Flow Liquid Secondary Ion Mass Spectrometry to Discovery Stage Metabolism Studies
Li, Chun, Chauret, Nathalie, Ducharme, Yves, Trimble, Laird A, Nicoll-Griffith, Deborah A, Yergey, James A
Published in Analytical chemistry (Washington) (01.09.1995)
Published in Analytical chemistry (Washington) (01.09.1995)
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CYP1A1 specificity of Verlukast epoxidation in mice, rats, rhesus monkeys, and humans
Grossman, S J, Herold, E G, Drey, J M, Alberts, D W, Umbenhauer, D R, Patrick, D H, Nicoll-Griffith, D, Chauret, N, Yergey, J A
Published in Drug metabolism and disposition (01.11.1993)
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Published in Drug metabolism and disposition (01.11.1993)
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