Transporters in Drug Development: 2018 ITC Recommendations for Transporters of Emerging Clinical Importance
Zamek-Gliszczynski, Maciej J, Taub, Mitchell E, Chothe, Paresh P, Chu, Xiaoyan, Giacomini, Kathleen M, Kim, Richard B, Ray, Adrian S, Stocker, Sophie L, Unadkat, Jashvant D, Wittwer, Matthias B, Xia, Cindy, Yee, Sook-Wah, Zhang, Lei, Zhang, Yan
Published in Clinical pharmacology and therapeutics (01.11.2018)
Published in Clinical pharmacology and therapeutics (01.11.2018)
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Journal Article
Organic Anion Transporter 2 (SLC22A7) Is a Facilitative Transporter of cGMP
Cropp, Cheryl D, Komori, Takafumi, Shima, James E, Urban, Thomas J, Yee, Sook Wah, More, Swati S, Giacomini, Kathleen M
Published in Molecular pharmacology (01.04.2008)
Published in Molecular pharmacology (01.04.2008)
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Journal Article
SLC transporters as therapeutic targets: emerging opportunities
Lin, Lawrence, Yee, Sook Wah, Kim, Richard B, Giacomini, Kathleen M
Published in Nature reviews. Drug discovery (01.08.2015)
Published in Nature reviews. Drug discovery (01.08.2015)
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Journal Article
Identification and characterization of novel polymorphisms in the basal promoter of the human transporter, MATE1
Ha Choi, Ji, Wah Yee, Sook, Kim, Mee J, Nguyen, Loan, Ho Lee, Jeong, Kang, Ji-One, Hesselson, Stephanie, Castro, Richard A, Stryke, Doug, Johns, Susan J, Kwok, Pui-Yan, Ferrin, Thomas E, Goo Lee, Min, Black, Brain L, Ahituv, Nadav, Giacomini, Kathleen M
Published in Pharmacogenetics and genomics (01.10.2009)
Published in Pharmacogenetics and genomics (01.10.2009)
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Journal Article
Influence of Transporter Polymorphisms on Drug Disposition and Response: A Perspective From the International Transporter Consortium
Yee, Sook Wah, Brackman, Deanna J, Ennis, Elizabeth A, Sugiyama, Yuichi, Kamdem, Landry K, Blanchard, Rebecca, Galetin, Aleksandra, Zhang, Lei, Giacomini, Kathleen M
Published in Clinical pharmacology and therapeutics (01.11.2018)
Published in Clinical pharmacology and therapeutics (01.11.2018)
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Journal Article
Membrane transporters in drug development
Giacomini, Kathleen M, Huang, Shiew-Mei, Tweedie, Donald J, Benet, Leslie Z, Brouwer, Kim L R, Chu, Xiaoyan, Dahlin, Amber, Evers, Raymond, Fischer, Volker, Hillgren, Kathleen M, Hoffmaster, Keith A, Ishikawa, Toshihisa, Keppler, Dietrich, Kim, Richard B, Lee, Caroline A, Niemi, Mikko, Polli, Joseph W, Sugiyama, Yuichi, Swaan, Peter W, Ware, Joseph A, Wright, Stephen H, Yee, Sook Wah, Zamek-Gliszczynski, Maciej J, Zhang, Lei
Published in Nature reviews. Drug discovery (01.03.2010)
Published in Nature reviews. Drug discovery (01.03.2010)
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Journal Article
OCT1 is a high-capacity thiamine transporter that regulates hepatic steatosis and is a target of metformin
Chen, Ligong, Shu, Yan, Liang, Xiaomin, Chen, Eugene C., Yee, Sook Wah, Zur, Arik A., Li, Shuanglian, Xu, Lu, Keshari, Kayvan R., Lin, Michael J., Chien, Huan-Chieh, Zhang, Youcai, Morrissey, Kari M., Liu, Jason, Ostrem, Jonathan, Younger, Noah S., Kurhanewicz, John, Shokat, Keven M., Ashrafi, Kaveh, Giacomini, Kathleen M.
Published in Proceedings of the National Academy of Sciences - PNAS (08.07.2014)
Published in Proceedings of the National Academy of Sciences - PNAS (08.07.2014)
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Journal Article
SLC13A3 is a major effector downstream of activated β-catenin in liver cancer pathogenesis
Zhao, Wennan, Wang, Xue, Han, Lifeng, Zhang, Chunze, Wang, Chenxi, Kong, Dexin, Zhang, Mingzhe, Xu, Tong, Li, Gen, Hu, Ge, Luo, Jiahua, Yee, Sook Wah, Yang, Jia, Stahl, Andreas, Chen, Xin, Zhang, Youcai
Published in Nature communications (30.08.2024)
Published in Nature communications (30.08.2024)
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Journal Article
Drugs in COVID-19 Clinical Trials: Predicting Transporter-Mediated Drug-Drug Interactions Using In Vitro Assays and Real-World Data
Yee, Sook Wah, Vora, Bianca, Oskotsky, Tomiko, Zou, Ling, Jakobsen, Sebastian, Enogieru, Osatohanmwen J, Koleske, Megan L, Kosti, Idit, Rödin, Mattias, Sirota, Marina, Giacomini, Kathleen M
Published in Clinical pharmacology and therapeutics (01.07.2021)
Published in Clinical pharmacology and therapeutics (01.07.2021)
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Journal Article
Rosace: a robust deep mutational scanning analysis framework employing position and mean-variance shrinkage
Rao, Jingyou, Xin, Ruiqi, Macdonald, Christian, Howard, Matthew K, Estevam, Gabriella O, Yee, Sook Wah, Wang, Mingsen, Fraser, James S, Coyote-Maestas, Willow, Pimentel, Harold
Published in Genome Biology (24.05.2024)
Published in Genome Biology (24.05.2024)
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Journal Article
Deorphaning a solute carrier 22 family member, SLC22A15, through functional genomic studies
Yee, Sook Wah, Buitrago, Dina, Stecula, Adrian, Ngo, Huy X, Chien, Huan-Chieh, Zou, Ling, Koleske, Megan L, Giacomini, Kathleen M
Published in The FASEB journal (01.12.2020)
Published in The FASEB journal (01.12.2020)
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Journal Article
Organic cation transporter 3 (Oct3) is a distinct catecholamines clearance route in adipocytes mediating the beiging of white adipose tissue
Song, Wenxin, Luo, Qi, Zhang, Yuping, Zhou, Linkang, Liu, Ye, Ma, Zhilong, Guo, Jianan, Huang, Yuedong, Cheng, Lili, Meng, Ziyi, Li, Zicheng, Zhang, Bin, Li, Siqi, Yee, Sook Wah, Fan, Hao, Li, Peng, Giacomini, Kathleen M, Chen, Ligong
Published in PLoS biology (01.01.2019)
Published in PLoS biology (01.01.2019)
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Journal Article
Organic cation transporter 1 (OCT1) modulates multiple cardiometabolic traits through effects on hepatic thiamine content
Liang, Xiaomin, Yee, Sook Wah, Chien, Huan-Chieh, Chen, Eugene C, Luo, Qi, Zou, Ling, Piao, Meiling, Mifune, Arias, Chen, Ligong, Calvert, Meredith E, King, Sarah, Norheim, Frode, Abad, Janna, Krauss, Ronald M, Giacomini, Kathleen M
Published in PLoS biology (01.04.2018)
Published in PLoS biology (01.04.2018)
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Journal Article
Metformin Is a Substrate and Inhibitor of the Human Thiamine Transporter, THTR‑2 (SLC19A3)
Liang, Xiaomin, Chien, Huan-Chieh, Yee, Sook Wah, Giacomini, Marilyn M, Chen, Eugene C, Piao, Meiling, Hao, Jia, Twelves, Jolyn, Lepist, Eve-Irene, Ray, Adrian S, Giacomini, Kathleen M
Published in Molecular pharmaceutics (07.12.2015)
Published in Molecular pharmaceutics (07.12.2015)
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Journal Article
Genome-Wide Meta-analysis Identifies Genetic Variants Associated With Glycemic Response to Sulfonylureas
Dawed, Adem Y, Yee, Sook Wah, Zhou, Kaixin, van Leeuwen, Nienke, Zhang, Yanfei, Siddiqui, Moneeza K, Etheridge, Amy, Innocenti, Federico, Xu, Fei, Li, Josephine H, Beulens, Joline W, van der Heijden, Amber A, Slieker, Roderick C, Chang, Yu-Chuan, Mercader, Josep M, Kaur, Varinderpal, Witte, John S, Lee, Ming Ta Michael, Kamatani, Yoichiro, Momozawa, Yukihide, Kubo, Michiaki, Palmer, Colin N A, Florez, Jose C, Hedderson, Monique M, 't Hart, Leen M, Giacomini, Kathleen M, Pearson, Ewan R
Published in Diabetes care (01.12.2021)
Published in Diabetes care (01.12.2021)
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Journal Article
Organic Anion Transporter Polypeptide 1B1 Polymorphism Modulates the Extent of Drug–Drug Interaction and Associated Biomarker Levels in Healthy Volunteers
Yee, Sook Wah, Giacomini, Marilyn M., Shen, Hong, Humphreys, W. Griffith, Horng, Howard, Brian, William, Lai, Yurong, Kroetz, Deanna L., Giacomini, Kathleen M.
Published in Clinical and translational science (01.07.2019)
Published in Clinical and translational science (01.07.2019)
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