Stereoselective Construction of Cisoidal Bisspiroacetal Frameworks through Magnesium Coordination of the Bilateral Acetal Oxygen Atoms
Yasukawa, Yoshifumi, Tsuchikawa, Hiroshi, Todokoro, Yasuto, Murata, Michio
Published in Asian journal of organic chemistry (01.06.2018)
Published in Asian journal of organic chemistry (01.06.2018)
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Highly Efficient Syntheses of C-N Axially Chiral 1-(ortho-hydroxyaryl)uracil using a Chiral Auxiliary and a Chiral Base
Hasegawa, Futoshi, Yasukawa, Yoshifumi, Kawamura, Kazushi, Tsuchikawa, Hiroshi, Murata, Michio
Published in Asian journal of organic chemistry (01.08.2018)
Published in Asian journal of organic chemistry (01.08.2018)
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Remote C−H alkylation and C−C bond cleavage enabled by an in situ generated palladacycle
Ye, Juntao, Shi, Zhihao, Sperger, Theresa, Yasukawa, Yoshifumi, Kingston, Cian, Schoenebeck, Franziska, Lautens, Mark
Published in Nature chemistry (01.04.2017)
Published in Nature chemistry (01.04.2017)
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Discovery of TP0628103: A Highly Potent and Selective MMP‑7 Inhibitor with Reduced OATP-Mediated Clearance Designed by Shifting Isoelectric Points
Oka, Yusuke, Abe-Sato, Kumi, Tabuse, Hideaki, Yasukawa, Yoshifumi, Yahara, Tohru, Nishimoto, Tomohiro, Kamitani, Masafumi, Fukunaga, Takuya, Ochiai, Nagahiro, Kumasaka-Abe, Tomoko, Hitaka, Kosuke, Gunji, Emi, Ohara, Hiroki, Takeda, Takuya, Kojima, Naoki, Asami, Taiji
Published in Journal of medicinal chemistry (25.01.2024)
Published in Journal of medicinal chemistry (25.01.2024)
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The stereoselective construction of E- and Z-Delta-Ile from E-dehydroamino acid ester: the synthesis of the phomopsin A tripeptide side chain
Yasuno, Yoko, Nishimura, Akito, Yasukawa, Yoshifumi, Karita, Yuma, Ohfune, Yasufumi, Shinada, Tetsuro
Published in Chemical communications (Cambridge, England) (25.01.2016)
Published in Chemical communications (Cambridge, England) (25.01.2016)
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SULFONAMIDE HAVING MMP 7-INHIBITING ACTION
OKA, Yusuke, ABE, Kumi, KIM, Chunhae, TABUSE, Hideaki, YASUKAWA, Yoshifumi
Year of Publication 10.11.2022
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Year of Publication 10.11.2022
Patent
The stereoselective construction of E- and Z-Δ-Ile from E-dehydroamino acid ester: the synthesis of the phomopsin A tripeptide side chainElectronic supplementary information (ESI) available. See DOI: 10.1039/c5cc08458j
Yasuno, Yoko, Nishimura, Akito, Yasukawa, Yoshifumi, Karita, Yuma, Ohfune, Yasufumi, Shinada, Tetsuro
Year of Publication 14.01.2016
Year of Publication 14.01.2016
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