Practical Synthetic Method for the Preparation of Pyrone Diesters: An Efficient Synthetic Route for the Synthesis of Dolutegravir Sodium
Yasukata, Tatsuro, Masui, Moriyasu, Ikarashi, Fumiya, Okamoto, Kazuya, Kurita, Takanori, Nagai, Masahiko, Sugata, Yoshihide, Miyake, Naoki, Hara, Shinichiro, Adachi, You, Sumino, Yukihito
Published in Organic process research & development (19.04.2019)
Published in Organic process research & development (19.04.2019)
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Practical and Scalable Synthetic Method for Preparation of Dolutegravir Sodium: Improvement of a Synthetic Route for Large-Scale Synthesis
Aoyama, Yasunori, Hakogi, Toshikazu, Fukui, Yuki, Yamada, Daisuke, Ooyama, Takao, Nishino, Yutaka, Shinomoto, Shoji, Nagai, Masahiko, Miyake, Naoki, Taoda, Yoshiyuki, Yoshida, Hiroshi, Yasukata, Tatsuro
Published in Organic process research & development (19.04.2019)
Published in Organic process research & development (19.04.2019)
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Novel semi-synthetic glycopeptide antibiotics active against methicillin-resistant staphylococcus aureus (MRSA) and vancomycin-resistant Enterococci (VRE): doubly-modified water-soluble derivatives of chloroorienticin B
Yoshida, Osamu, Yasukata, Tatsuro, Sumino, Yukihito, Munekage, Tadashi, Narukawa, Yukitoshi, Nishitani, Yasuhiro
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
Published in Bioorganic & medicinal chemistry letters (04.11.2002)
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Practical Manufacturing Process for Baloxavir Marboxil: Efficient Route to a Tricyclic Triazinanone Scaffold
Fukui, Nobuaki, Maki, Toshikatsu, Ban, Kazunori, Kijima, Akihito, Shibahara, Setsuya, Okamoto, Kazuya, Kamiya, Sho, Yasukata, Tatsuro, Tsuritani, Takayuki
Published in Organic process research & development (21.06.2024)
Published in Organic process research & development (21.06.2024)
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Practical Manufacturing Process for Baloxavir Marboxil: Effective Selection and Replacement of Protective Group toward Enhancement of Crystallization-Induced Diastereomer Transformation
Fukui, Nobuaki, Shibahara, Setsuya, Maki, Toshikatsu, Ueno, Tatsuhiko, Yanagisawa, Shuichi, Okamoto, Kazuya, Tanimoto, Emi, Ohara, Takafumi, Yasukata, Tatsuro, Tsuritani, Takayuki
Published in Organic process research & development (21.06.2024)
Published in Organic process research & development (21.06.2024)
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Stereoselective reactions. 30. Enantioselective alkylation of the lithium enolates of six-membered cyclic ketones using tetradentate chiral amines in the presence of lithium bromide
Murakata, Masatoshi, Yasukata, Tatsuro, Aoki, Takumi, Nakajima, Makoto, Koga, Kenji
Published in Tetrahedron (12.03.1998)
Published in Tetrahedron (12.03.1998)
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Synthesis and in vitro/in vivo antibacterial activity of oxazolidinones having thiocarbamate at C-5 on the A-ring and an amide- or ureasubstituted [1,2,5]triazepane or [1,2,5]oxadiazepane as the C-ring
Suzuki, Hideyuki, Utsunomiya, Iwao, Shudo, Koichi, Fukuhara, Norio, Iwaki, Tsutomu, Yasukata, Tatsuro
Published in European journal of medicinal chemistry (01.11.2013)
Published in European journal of medicinal chemistry (01.11.2013)
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Journal Article
Synthesis and in vitro/in vivo antibacterial activity of oxazolidinones having thiocarbamate at C-5 on the A-ring and an amide- or urea-substituted [1,2,5]triazepane or [1,2,5]oxadiazepane as the C-ring
Suzuki, Hideyuki, Utsunomiya, Iwao, Shudo, Koichi, Fukuhara, Norio, Iwaki, Tsutomu, Yasukata, Tatsuro
Published in European journal of medicinal chemistry (01.11.2013)
Published in European journal of medicinal chemistry (01.11.2013)
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Journal Article
Antibacterial oxazolidinone analogues having a N-hydroxyacetyl-substituted seven-membered [1,2,5]triazepane or [1,2,5]oxadiazepane C-ring unit
Suzuki, Hideyuki, Utsunomiya, Iwao, Shudo, Koichi, Fukuhara, Norio, Iwaki, Tsutomu, Yasukata, Tatsuro
Published in European journal of medicinal chemistry (01.05.2013)
Published in European journal of medicinal chemistry (01.05.2013)
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Journal Article
Stereoselective Reactions. XXII. Design and Synthesis of Chiral Chelated Lithium Amides for Enantioselective Reactions
SHIRAI, Ryuichi, AOKI, Kazumasa, SATO, Daisaku, KIM, Hee-Doo, MURAKATA, Masatoshi, YASUKATA, Tatsuro, KOGA, Kenji
Published in Chemical & pharmaceutical bulletin (1994)
Published in Chemical & pharmaceutical bulletin (1994)
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A novel series of parenteral cephalosporins exhibiting potent activities against Pseudomonas aeruginosa and other Gram-negative pathogens: Synthesis and structure–activity relationships
Yamawaki, Kenji, Nomura, Takashi, Yasukata, Tatsuro, Uotani, Koichi, Miwa, Hideaki, Takeda, Kei, Nishitani, Yasuhiro
Published in Bioorganic & medicinal chemistry (01.11.2007)
Published in Bioorganic & medicinal chemistry (01.11.2007)
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Journal Article
A Catalytic Asymmetric Wagner−Meerwein Shift
Trost, Barry M, Yasukata, Tatsuro
Published in Journal of the American Chemical Society (25.07.2001)
Published in Journal of the American Chemical Society (25.07.2001)
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Journal Article
A novel series of parenteral cephalosporins exhibiting potent activities against both Pseudomonas aeruginosa and other Gram-negative pathogens. Part 2: Synthesis and structure–activity relationships
Yamawaki, Kenji, Nomura, Takashi, Yasukata, Tatsuro, Tanimoto, Norihiko, Uotani, Koichi, Miwa, Hideaki, Yamano, Yoshinori, Takeda, Kei, Nishitani, Yasuhiro
Published in Bioorganic & medicinal chemistry (15.02.2008)
Published in Bioorganic & medicinal chemistry (15.02.2008)
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Journal Article
CARNOSADINE LACTAM DERIVATIVE HAVING ANTIBACTERIAL ACTIVITY
UEDA, TAICHI, OHWADA, TOMOHIKO, SUZUKI, NAOYUKI, FUMOTO, MASATAKA, YASUKATA, TATSURO, MINAGAWA, KAZUYUKI
Year of Publication 08.05.2014
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Year of Publication 08.05.2014
Patent
OXAZOLIDINONE DERIVATIVE HAVING 7-MEMBERED HETERO RING
UTSUNOMIYA, IWAO, SHUDO, KOICHI, YASUKATA, TATSURO, IWAKI, TSUTOMU, SUZUKI, HIDEYUKI
Year of Publication 09.04.2009
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Year of Publication 09.04.2009
Patent