High-resolution structure of the human GPR40 receptor bound to allosteric agonist TAK-875
Srivastava, Ankita, Yano, Jason, Hirozane, Yoshihiko, Kefala, Georgia, Gruswitz, Franz, Snell, Gyorgy, Lane, Weston, Ivetac, Anthony, Aertgeerts, Kathleen, Nguyen, Jasmine, Jennings, Andy, Okada, Kengo
Published in Nature (London) (04.09.2014)
Published in Nature (London) (04.09.2014)
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"What Keeps Me Awake at Night": Assisted Living Administrator Responses to COVID-19
Kyler-Yano, Jason Z, Tunalilar, Ozcan, Hasworth, Serena, Kohon, Jacklyn, Winfree, Jaclyn, Wilton, Riley, Tuttle, Aliza, Carder, Paula
Published in The Gerontologist (09.02.2022)
Published in The Gerontologist (09.02.2022)
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Adaptations for the Oxidation of Polycyclic Aromatic Hydrocarbons Exhibited by the Structure of Human P450 1A2
Sansen, Stefaan, Yano, Jason K., Reynald, Rosamund L., Schoch, Guillaume A., Griffin, Keith J., Stout, C. David, Johnson, Eric F.
Published in The Journal of biological chemistry (11.05.2007)
Published in The Journal of biological chemistry (11.05.2007)
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Structural Analysis of the Mechanism of Inhibition and Allosteric Activation of the Kinase Domain of HER2 Protein
Aertgeerts, Kathleen, Skene, Robert, Yano, Jason, Sang, Bi-Ching, Zou, Hua, Snell, Gyorgy, Jennings, Andy, Iwamoto, Keiji, Habuka, Noriyuki, Hirokawa, Aki, Ishikawa, Tomoyasu, Tanaka, Toshimasa, Miki, Hiroshi, Ohta, Yoshikazu, Sogabe, Satoshi
Published in The Journal of biological chemistry (27.05.2011)
Published in The Journal of biological chemistry (27.05.2011)
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The Structure of Human Microsomal Cytochrome P450 3A4 Determined by X-ray Crystallography to 2.05-Å Resolution
Yano, Jason K., Wester, Michael R., Schoch, Guillaume A., Griffin, Keith J., Stout, C. David, Johnson, Eric F.
Published in The Journal of biological chemistry (10.09.2004)
Published in The Journal of biological chemistry (10.09.2004)
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Soticlestat, a novel cholesterol 24-hydroxylase inhibitor shows a therapeutic potential for neural hyperexcitation in mice
Nishi, Toshiya, Kondo, Shinichi, Miyamoto, Maki, Watanabe, Sayuri, Hasegawa, Shigeo, Kondo, Shigeru, Yano, Jason, Watanabe, Etsurou, Ishi, Tsuyoshi, Yoshikawa, Masato, Ando, Haruhi Kamisaki, Farnaby, William, Fujimoto, Shinji, Sunahara, Eiji, Ohori, Momoko, During, Matthew J, Kuroita, Takanobu, Koike, Tatsuki
Published in Scientific reports (13.10.2020)
Published in Scientific reports (13.10.2020)
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Design and Synthesis of Novel Human Epidermal Growth Factor Receptor 2 (HER2)/Epidermal Growth Factor Receptor (EGFR) Dual Inhibitors Bearing a Pyrrolo[3,2-d]pyrimidine Scaffold
Ishikawa, Tomoyasu, Seto, Masaki, Banno, Hiroshi, Kawakita, Youichi, Oorui, Mami, Taniguchi, Takahiko, Ohta, Yoshikazu, Tamura, Toshiya, Nakayama, Akiko, Miki, Hiroshi, Kamiguchi, Hidenori, Tanaka, Toshimasa, Habuka, Noriyuki, Sogabe, Satoshi, Yano, Jason, Aertgeerts, Kathleen, Kamiyama, Keiji
Published in Journal of medicinal chemistry (08.12.2011)
Published in Journal of medicinal chemistry (08.12.2011)
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Discovery of Novel 3-Piperidinyl Pyridine Derivatives as Highly Potent and Selective Cholesterol 24-Hydroxylase (CH24H) Inhibitors
Kajita, Yuichi, Ikeda, Shuhei, Yoshikawa, Masato, Fukuda, Hiromi, Watanabe, Etsurou, Yano, Jason, Lane, Weston, Miyamoto, Maki, Ishii, Tsuyoshi, Nishi, Toshiya, Koike, Tatsuki
Published in Journal of medicinal chemistry (24.02.2022)
Published in Journal of medicinal chemistry (24.02.2022)
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Determinants of Cytochrome P450 2C8 Substrate Binding: STRUCTURES OF COMPLEXES WITH MONTELUKAST, TROGLITAZONE, FELODIPINE, AND 9-CIS-RETINOIC ACID
Schoch, Guillaume A, Yano, Jason K, Sansen, Stefaan, Dansette, Patrick M, Stout, C. David, Johnson, Eric F
Published in The Journal of biological chemistry (20.06.2008)
Published in The Journal of biological chemistry (20.06.2008)
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The Structure of Human Cytochrome P450 2C9 Complexed with Flurbiprofen at 2.0-Ã Resolution
Wester, Michael R, Yano, Jason K, Schoch, Guillaume A, Yang, Christine, Griffin, Keith J, Stout, C David, Johnson, Eric F
Published in The Journal of biological chemistry (20.08.2004)
Published in The Journal of biological chemistry (20.08.2004)
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Translational and Therapeutic Evaluation of RAS-GTP Inhibition by RMC-6236 in RAS-Driven Cancers
Jiang, Jingjing, Jiang, Lingyan, Maldonato, Benjamin J, Wang, Yingyun, Holderfield, Matthew, Aronchik, Ida, Winters, Ian P, Salman, Zeena, Blaj, Cristina, Menard, Marie, Brodbeck, Jens, Chen, Zhe, Wei, Xing, Rosen, Michael J, Gindin, Yevgeniy, Lee, Bianca J, Evans, James W, Chang, Stephanie, Wang, Zhican, Seamon, Kyle J, Parsons, Dylan, Cregg, James, Marquez, Abby, Tomlinson, Aidan C A, Yano, Jason K, Knox, John E, Quintana, Elsa, Aguirre, Andrew J, Arbour, Kathryn C, Reed, Abby, Gustafson, W Clay, Gill, Adrian L, Koltun, Elena S, Wildes, David, Smith, Jacqueline A M, Wang, Zhengping, Singh, Mallika
Published in Cancer discovery (03.06.2024)
Published in Cancer discovery (03.06.2024)
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Synthetic Inhibitors of Cytochrome P-450 2A6: Inhibitory Activity, Difference Spectra, Mechanism of Inhibition, and Protein Cocrystallization
Yano, Jason K, Denton, Travis T, Cerny, Matthew A, Zhang, Xiaodong, Johnson, Eric F, Cashman, John R
Published in Journal of medicinal chemistry (30.11.2006)
Published in Journal of medicinal chemistry (30.11.2006)
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Synthesis and biological evaluation of novel selective androgen receptor modulators (SARMs) Part III: Discovery of 4-(5-oxopyrrolidine-1-yl)benzonitrile derivative 2f as a clinical candidate
Aikawa, Katsuji, Asano, Moriteru, Ono, Koji, Habuka, Noriyuki, Yano, Jason, Wilson, Keith, Fujita, Hisashi, Kandori, Hitoshi, Hara, Takahito, Morimoto, Megumi, Santou, Takashi, Yamaoka, Masuo, Nakayama, Masaharu, Hasuoka, Atsushi
Published in Bioorganic & medicinal chemistry (01.07.2017)
Published in Bioorganic & medicinal chemistry (01.07.2017)
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Discovery of potent, selective, and orally bioavailable quinoline-based dipeptidyl peptidase IV inhibitors targeting Lys554
Maezaki, Hironobu, Banno, Yoshihiro, Miyamoto, Yasufumi, Moritou, Yuusuke, Asakawa, Tomoko, Kataoka, Osamu, Takeuchi, Koji, Suzuki, Nobuhiro, Ikedo, Koji, Kosaka, Takuo, Sasaki, Masako, Tsubotani, Shigetoshi, Tani, Akiyoshi, Funami, Miyuki, Yamamoto, Yoshio, Tawada, Michiko, Aertgeerts, Kathleen, Yano, Jason, Oi, Satoru
Published in Bioorganic & medicinal chemistry (01.08.2011)
Published in Bioorganic & medicinal chemistry (01.08.2011)
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