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Published in Journal of the American Chemical Society (08.05.1996)
Published in Journal of the American Chemical Society (08.05.1996)
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Published in Bioorganic & medicinal chemistry letters (15.07.2023)
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Published in Bioorganic & medicinal chemistry letters (01.12.2020)
Published in Bioorganic & medicinal chemistry letters (01.12.2020)
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Identification and Preclinical Pharmacology of ((1R,3S)‑1-Amino-3-((S)‑6-(2-methoxyphenethyl)-5,6,7,8-tetrahydronaphthalen-2-yl)cyclopentyl)methanol (BMS-986166): A Differentiated Sphingosine-1-phosphate Receptor 1 (S1P1) Modulator Advanced into Clinical Trials
Gilmore, John L, Xiao, Hai-Yun, Dhar, T. G. Murali, Yang, Michael G, Xiao, Zili, Xie, Jenny, Lehman-McKeeman, Lois D, Gong, Lei, Sun, Huadong, Lecureux, Lloyd, Chen, Cliff, Wu, Dauh-Rurng, Dabros, Marta, Yang, Xiaoxia, Taylor, Tracy L, Zhou, Xia D, Heimrich, Elizabeth M, Thomas, Rochelle, McIntyre, Kim W, Borowski, Virna, Warrack, Bethanne M, Li, Yuwen, Shi, Hong, Levesque, Paul C, Yang, Zheng, Marino, Anthony M, Cornelius, Georgia, D’Arienzo, Celia J, Mathur, Arvind, Rampulla, Richard, Gupta, Anuradha, Pragalathan, Bala, Shen, Ding Ren, Cvijic, Mary Ellen, Salter-Cid, Luisa M, Carter, Percy H, Dyckman, Alaric J
Published in Journal of medicinal chemistry (14.03.2019)
Published in Journal of medicinal chemistry (14.03.2019)
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Xiao, Zili, Yang, Michael G, Dhar, T. G. Murali, Xiao, Hai-Yun, Gilmore, John L, Marcoux, David, McIntyre, Kim W, Taylor, Tracy L, Shi, Hong, Levesque, Paul C, Marino, Anthony M, Cornelius, Georgia, Mathur, Arvind, Shen, Ding Ren, Cvijic, Mary Ellen, Lehman-McKeeman, Lois D, Sun, Huadong, Xie, Jenny H, Carter, Percy H, Dyckman, Alaric J
Published in ACS medicinal chemistry letters (10.09.2020)
Published in ACS medicinal chemistry letters (10.09.2020)
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Azatricyclic Inverse Agonists of RORγt That Demonstrate Efficacy in Models of Rheumatoid Arthritis and Psoriasis
Liu, Qingjie, Xiao, Hai-Yun, Batt, Douglas G, Xiao, Zili, Zhu, Yeheng, Yang, Michael G, Li, Ning, Yip, Shiuhang, Li, Peng, Sun, Dawn, Wu, Dauh-Rurng, Ruzanov, Max, Sack, John S, Weigelt, Carolyn A, Wang, Jinhong, Li, Sha, Shuster, David J, Xie, Jenny H, Song, Yunling, Sherry, Tara, Obermeier, Mary T, Fura, Aberra, Stefanski, Kevin, Cornelius, Georgia, Chacko, Silvi, Khandelwal, Purnima, Dudhgaonkar, Shailesh, Rudra, Anjuman, Nagar, Jignesh, Murali, Venkata, Govindarajan, Arun, Denton, Rex, Zhao, Qihong, Meanwell, Nicholas A, Borzilleri, Robert, Dhar, T. G. Murali
Published in ACS medicinal chemistry letters (13.05.2021)
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Use of a Conformational-Switching Mechanism to Modulate Exposed Polarity: Discovery of CCR2 Antagonist BMS-741672
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Yang, Michael G, Dhar, T. G. Murali, Xiao, Zili, Xiao, Hai-Yun, Duan, James J.-W, Jiang, Bin, Galella, Michael A, Cunningham, Mark, Wang, Jinhong, Habte, Sium, Shuster, David, McIntyre, Kim W, Carman, Julie, Holloway, Deborah A, Somerville, John E, Nadler, Steven G, Salter-Cid, Luisa, Barrish, Joel C, Weinstein, David S
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Published in Journal of medicinal chemistry (28.05.2015)
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Asymmetric Hydroboration Approach to the Scalable Synthesis of ((1R,3S)‑1-Amino-3-((R)‑6-hexyl-5,6,7,8-tetrahydronaphthalen-2-yl)cyclopentyl)methanol (BMS-986104) as a Potent S1P1 Receptor Modulator
Yang, Michael G, Xiao, Zili, Dhar, T. G. Murali, Xiao, Hai-Yun, Gilmore, John L, Marcoux, David, Xie, Jenny H, McIntyre, Kim W, Taylor, Tracy L, Borowski, Virna, Heimrich, Elizabeth, Li, Yu-Wen, Feng, Jianlin, Fernandes, Alda, Yang, Zheng, Balimane, Praveen, Marino, Anthony M, Cornelius, Georgia, Warrack, Bethanne M, Mathur, Arvind, Wu, Dauh-Rurng, Li, Peng, Gupta, Anuradha, Pragalathan, Bala, Shen, Ding Ren, Cvijic, Mary Ellen, Lehman-McKeeman, Lois D, Salter-Cid, Luisa, Barrish, Joel C, Carter, Percy H, Dyckman, Alaric J
Published in Journal of medicinal chemistry (22.12.2016)
Published in Journal of medicinal chemistry (22.12.2016)
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Xiao, Zili, Yang, Michael G., Tebben, Andrew J., Galella, Michael A., Weinstein, David S.
Published in Tetrahedron letters (03.11.2010)
Published in Tetrahedron letters (03.11.2010)
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Asymmetric Hydroboration Approach to the Scalable Synthesis of ((1R,3S)-1-Amino-3-((R)-6-hexyl-5,6,7,8-tetrahydronaphthalen-2-yl)cyclopentyl)methanol (BMS-986104) as a Potent S1P 1 Receptor Modulator
Yang, Michael G, Xiao, Zili, Dhar, T G Murali, Xiao, Hai-Yun, Gilmore, John L, Marcoux, David, Xie, Jenny H, McIntyre, Kim W, Taylor, Tracy L, Borowski, Virna, Heimrich, Elizabeth, Li, Yu-Wen, Feng, Jianlin, Fernandes, Alda, Yang, Zheng, Balimane, Praveen, Marino, Anthony M, Cornelius, Georgia, Warrack, Bethanne M, Mathur, Arvind, Wu, Dauh-Rurng, Li, Peng, Gupta, Anuradha, Pragalathan, Bala, Shen, Ding Ren, Cvijic, Mary Ellen, Lehman-McKeeman, Lois D, Salter-Cid, Luisa, Barrish, Joel C, Carter, Percy H, Dyckman, Alaric J
Published in Journal of medicinal chemistry (22.12.2016)
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The Amyloid-β Rise and γ-Secretase Inhibitor Potency Depend on the Level of Substrate Expression
Burton, Catherine R., Meredith, Jere E., Barten, Donna M., Goldstein, Margi E., Krause, Carol M., Kieras, Cathy J., Sisk, Lisa, Iben, Lawrence G., Polson, Craig, Thompson, Mark W., Lin, Xu-Alan, Corsa, Jason, Fiedler, Tracey, Pierdomenico, Maria, Cao, Yang, Roach, Arthur H., Cantone, Joseph L., Ford, Michael J., Drexler, Dieter M., Olson, Richard E., Yang, Michael G., Bergstrom, Carl P., McElhone, Kate E., Bronson, Joanne J., Macor, John E., Blat, Yuval, Grafstrom, Robert H., Stern, Andrew M., Seiffert, Dietmar A., Zaczek, Robert, Albright, Charles F., Toyn, Jeremy H.
Published in The Journal of biological chemistry (22.08.2008)
Published in The Journal of biological chemistry (22.08.2008)
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Published in Bioorganic & medicinal chemistry letters (01.04.2014)
Published in Bioorganic & medicinal chemistry letters (01.04.2014)
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Diastereoselective Aldol and Allylstannane Addition Reactions. The Merged Stereochemical Impact of .alpha. and .beta. Aldehyde Substituents
Evans, David A, Dart, Michael J, Duffy, Joseph L, Yang, Michael G, Livingston, Alex B
Published in Journal of the American Chemical Society (01.06.1995)
Published in Journal of the American Chemical Society (01.06.1995)
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Published in Bioorganic & medicinal chemistry letters (15.04.2010)
Published in Bioorganic & medicinal chemistry letters (15.04.2010)
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Year of Publication 01.07.2022
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Year of Publication 01.07.2022
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