Histone deacetylase inhibitor KBH-A42 inhibits cytokine production in RAW 264.7 macrophage cells and in vivo endotoxemia model
Choi, Yongseok, Park, Song-Kyu, Kim, Hwan Mook, Kang, Jong Soon, Yoon, Yeo Dae, Han, Sang Bae, Han, Jeung Whan, Yang, Jee Sun, Han, Gyoonhee
Published in Experimental & molecular medicine (31.10.2008)
Published in Experimental & molecular medicine (31.10.2008)
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Control of leucine-dependent mTORC1 pathway through chemical intervention of leucyl-tRNA synthetase and RagD interaction
Kim, Jong Hyun, Lee, Chulho, Lee, Minji, Wang, Haipeng, Kim, Kibum, Park, Seung Joon, Yoon, Ina, Jang, Jayun, Zhao, Hanchao, Kim, Hoi Kyoung, Kwon, Nam Hoon, Jeong, Seung Jae, Yoo, Hee Chan, Kim, Jae Hyun, Yang, Jee Sun, Lee, Myeong Youl, Lee, Chang Woo, Yun, Jieun, Oh, Soo Jin, Kang, Jong Soon, Martinis, Susan A, Hwang, Kwang Yeon, Guo, Min, Han, Gyoonhee, Han, Jung Min, Kim, Sunghoon
Published in Nature communications (29.09.2017)
Published in Nature communications (29.09.2017)
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A Ras destabilizer KYA1797K overcomes the resistance of EGFR tyrosine kinase inhibitor in KRAS-mutated non-small cell lung cancer
Park, Jieun, Cho, Yong-Hee, Shin, Wook-Jin, Lee, Sang-Kyu, Lee, JaeHeon, Kim, Taehyung, Cha, Pu-Hyeon, Yang, Jee Sun, Cho, Jaebeom, Min, Do Sik, Han, Gyoonhee, Lee, Ho-Young, Choi, Kang-Yell
Published in Scientific reports (24.01.2019)
Published in Scientific reports (24.01.2019)
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A novel antitumor piperazine alkyl compound causes apoptosis by inducing RhoB expression via ROS-mediated c-Abl/p38 MAPK signaling
Chung, Kyung-Sook, Han, Gyoonhee, Kim, Bo-Kyung, Kim, Hwan-Mook, Yang, Jee Sun, Ahn, Jiwon, Lee, Kyeong, Song, Kyung-Bin, Won, Misun
Published in Cancer chemotherapy and pharmacology (01.12.2013)
Published in Cancer chemotherapy and pharmacology (01.12.2013)
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Journal Article
Synthesis of amide and urea derivatives of benzothiazole as Raf-1 inhibitor
Song, Eun Young, Kaur, Navneet, Park, Mi-Young, Jin, Yinglan, Lee, Kyeong, Kim, Guncheol, Lee, Ki Youn, Yang, Jee Sun, Shin, Jae Hong, Nam, Ky-Youb, No, Kyoung Tai, Han, Gyoonhee
Published in European journal of medicinal chemistry (01.07.2008)
Published in European journal of medicinal chemistry (01.07.2008)
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Synthesis and biological evaluation of novel aliphatic amido-quaternary ammonium salts for anticancer chemotherapy: Part I
Yang, Jee Sun, Song, Doona, Lee, Boah, Ko, Won Jin, Park, Song-Kyu, Won, Misun, Lee, Kiho, Kim, Hwan Mook, Han, Gyoonhee
Published in European journal of medicinal chemistry (01.07.2011)
Published in European journal of medicinal chemistry (01.07.2011)
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Structure based optimization of chromen-based TNF-α converting enzyme (TACE) inhibitors on S1′ pocket and their quantitative structure–activity relationship (QSAR) study
Yang, Jee Sun, Chun, Kwangwoo, Park, Jung Eun, Cho, Misun, Seo, Jeongjea, Song, Doona, Yoon, Hongchul, Park, Chun-Ho, Joe, Bo-Young, Choi, Jong-Hee, Kim, Myung-Hwa, Han, Gyoonhee
Published in Bioorganic & medicinal chemistry (15.12.2010)
Published in Bioorganic & medicinal chemistry (15.12.2010)
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Journal Article
NOVEL BENZENESULFONAMIDE DERIVATIVE AND USE THEREOF
KIM, Jae Hyun, KIM, Sunghoon, HAN, Jung Min, YANG, Jee Sun, HAN, Gyoonhee, LEE, Chulho, JUNG, Kilsoo, KIM, Jong Hyun
Year of Publication 21.09.2017
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Year of Publication 21.09.2017
Patent
Novel benzenesulfonamide derivatives and uses thereof
HAN, JUNG MIN, KIM, SUNG HOON, HAN, GYOON HEE, YANG, JEE SUN, LEE, CHUL HO, KIM, JAE HYUN, JASON ANTHONY WITEK, KIM, JONG HYUN
Year of Publication 25.09.2017
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Year of Publication 25.09.2017
Patent
Small-molecule binding of the axin RGS domain promotes β-catenin and Ras degradation
Cha, Pu-Hyeon, Cho, Yong-Hee, Lee, Sang-Kyu, Lee, JaeHeon, Jeong, Woo-Jeong, Moon, Byoung-San, Yun, Ji-Hye, Yang, Jee Sun, Choi, Sooho, Yoon, Juyong, Kim, Hyun-Yi, Kim, Mi-Yeon, Kaduwal, Saluja, Lee, Weontae, Min, Do Sik, Kim, Hoguen, Han, Gyoonhee, Choi, Kang-Yell
Published in Nature chemical biology (01.08.2016)
Published in Nature chemical biology (01.08.2016)
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Structural modifications at the 6-position of thieno[2,3-d]pyrimidines and their effects on potency at FLT3 for treatment of acute myeloid leukemia
Kim, Hyuntae, Lee, Chulho, Yang, Jee Sun, Choi, Seonghwi, Park, Chun-Ho, Kang, Jong Soon, Oh, Soo Jin, Yun, Jieun, Kim, Myung-Hwa, Han, Gyoonhee
Published in European journal of medicinal chemistry (14.09.2016)
Published in European journal of medicinal chemistry (14.09.2016)
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Journal Article
Chemical inhibition of prometastatic lysyl-tRNA synthetase-laminin receptor interaction
Kim, Dae Gyu, Lee, Jin Young, Kwon, Nam Hoon, Fang, Pengfei, Zhang, Qian, Wang, Jing, Young, Nicolas L, Guo, Min, Cho, Hye Young, Mushtaq, Ameeq Ul, Jeon, Young Ho, Choi, Jin Woo, Han, Jung Min, Kang, Ho Woong, Joo, Jae Eun, Hur, Youn, Kang, Wonyoung, Yang, Heekyoung, Nam, Do-Hyun, Lee, Mi-Sook, Lee, Jung Weon, Kim, Eun-Sook, Moon, Aree, Kim, Kibom, Kim, Doyeun, Kang, Eun Joo, Moon, Youngji, Rhee, Kyung Hee, Han, Byung Woo, Yang, Jee Sun, Han, Gyoonhee, Yang, Won Suk, Lee, Cheolju, Wang, Ming-Wei, Kim, Sunghoon
Published in Nature chemical biology (01.01.2014)
Published in Nature chemical biology (01.01.2014)
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Journal Article
Synthesis and biological evaluation of novel thieno[2,3-d]pyrimidine-based FLT3 inhibitors as anti-leukemic agents
Yang, Jee Sun, Park, Chun-Ho, Lee, Chulho, Kim, Hwan, Oh, Changmok, Choi, Yejoo, Kang, Jong Soon, Yun, Jieun, Jeong, Jin-Hyun, Kim, Myung-Hwa, Han, Gyoonhee
Published in European journal of medicinal chemistry (06.10.2014)
Published in European journal of medicinal chemistry (06.10.2014)
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Journal Article
Discovery of thienopyrimidine-based FLT3 inhibitors from the structural modification of known IKKβ inhibitors
Park, Chun-Ho, Lee, Chulho, Yang, Jee Sun, Joe, Bo-Young, Chun, Kwangwoo, Kim, Hyuntae, Kim, Hye Yun, Kang, Jong Soon, Lee, Jangik I., Kim, Myung-Hwa, Han, Gyoonhee
Published in Bioorganic & medicinal chemistry letters (15.06.2014)
Published in Bioorganic & medicinal chemistry letters (15.06.2014)
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