A Study into the ADP-Ribosylome of IFN-γ-Stimulated THP‑1 Human Macrophage-like Cells Identifies ARTD8/PARP14 and ARTD9/PARP9 ADP-Ribosylation
Higashi, Hideyuki, Maejima, Takashi, Lee, Lang Ho, Yamazaki, Yukiyoshi, Hottiger, Michael O, Singh, Sasha A, Aikawa, Masanori
Published in Journal of proteome research (05.04.2019)
Published in Journal of proteome research (05.04.2019)
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A practical synthesis for (S)-5-(4-(1-methylethoxy)phenyl)-5-methylimidazolidine-2,4-dione and its application in the synthesis of a novel liver X receptor β-selective agonist
Koura, Minoru, Sumida, Hisashi, Yamazaki, Yukiyoshi, Shibuya, Kimiyuki
Published in Tetrahedron: asymmetry (15.01.2016)
Published in Tetrahedron: asymmetry (15.01.2016)
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Multiorgan Systems Study Reveals Igfbp7 as a Suppressor of Gluconeogenesis after Gastric Bypass Surgery
Arima, Naoaki, Sasaki, Yusuke, Lee, Lang Ho, Zhang, Hengmin, Figueiredo, Jose-Luiz, Mlynarchik, Andrew K, Qiao, Jiao, Yamada, Iwao, Higashi, Hideyuki, Ha, Anna H, Halu, Arda, Mizuno, Ken, Singh, Sasha A, Yamazaki, Yukiyoshi, Aikawa, Masanori
Published in Journal of proteome research (03.01.2020)
Published in Journal of proteome research (03.01.2020)
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Novel Synthesis of Butyl (S)-2-Hydroxybutanoate, the Key Intermediate of PPAR alpha Agonist (R)-K-13675 from Butyl (2S,3R)-Epoxybutanoate and Butyl (S)-2,3-Epoxypropanoate
Araki, Takaaki, Koura, Minoru, Yamazaki, Yukiyoshi, Shibuya, Kimiyuki
Published in Synthesis (Stuttgart) (17.05.2013)
Published in Synthesis (Stuttgart) (17.05.2013)
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Abstract 175: Dynamin-Related Protein 1 Regulates Proteostasis and Proprotein Convertase Subtilisin/Kexin Type 9 Secretion
Rogers, Maximillian A, Hutcheson, Joshua D, Goettsch, Claudia, Halu, Arda, Singh, Sasha, Higashi, Hideyuki, Lee, Lang H, Wang, Lixiang, Schlotter, Florian, Morgan, Stephanie, Okui, Takehito, Yamazaki, Yukiyoshi, Daugherty, Alan, Nomura, Masatoshi, Aikawa, Masanori, Aikawa, Elena
Published in Arteriosclerosis, thrombosis, and vascular biology (01.05.2018)
Published in Arteriosclerosis, thrombosis, and vascular biology (01.05.2018)
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Lipase-Catalyzed Enantioselective Hydrolysis of Bis(acyloxymethyl) 1, 4-Dihydro-3, 5-pyridinedicarboxylates Leading to Optically Active Medicines
EBIIKE, Hirosato, MARUYAMA, Kaori, YAMAZAKI, Yukiyoshi, HIROSE, Yoshihiko, KARIYA, Kinya, SASAKI, Ikuharu, KURONO, Yoshiaki, TERAO, Yoshiyasu, ACHIWA, Kazuo
Published in Chemical & pharmaceutical bulletin (1997)
Published in Chemical & pharmaceutical bulletin (1997)
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A practical synthesis of the PPARα agonist, ( R)-K-13675, starting from ( S)-2-hydroxybutyrolactone
Yamazaki, Yukiyoshi, Araki, Takaaki, Koura, Minoru, Shibuya, Kimiyuki
Published in Tetrahedron (25.08.2008)
Published in Tetrahedron (25.08.2008)
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Design and synthesis of highly potent and selective human peroxisome proliferator-activated receptor α agonists
Yamazaki, Yukiyoshi, Abe, Kazutoyo, Toma, Tsutomu, Nishikawa, Masahiro, Ozawa, Hidefumi, Okuda, Ayumu, Araki, Takaaki, Oda, Soichi, Inoue, Keisuke, Shibuya, Kimiyuki, Staels, Bart, Fruchart, Jean-Charles
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
Published in Bioorganic & medicinal chemistry letters (15.08.2007)
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Enantioselective synthesis of the PPAR alpha agonist (R)-K-13675 via (S)-2-hydroxybutyrolactone
Yamazaki, Yukiyoshi, Araki, Takaaki, Koura, Minoru, Shibuya, Kimiyuki
Published in Synthesis (Stuttgart) (01.04.2008)
Published in Synthesis (Stuttgart) (01.04.2008)
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Abstract 19434: The Novel PPARalpha-Selective Agonist K-877 Improves Dyslipidemia, Enhances Reverse Cholesterol Transport and Decreases Inflammation and Atherosclerosis
Hennuyer, Nathalie, Duplan, Isabelle, Paquet, Charlotte, Vanhoutte, Jonathan, Touche, Véronique, Chinetti, Giulia, Lestavel, Sophie, Takizawa, Toshiaki, Yamazaki, Yukiyoshi, Tanabe, Sohei, Staels, Bart
Published in Circulation (New York, N.Y.) (26.11.2013)
Published in Circulation (New York, N.Y.) (26.11.2013)
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Asymmetric Synthesis of (R)-Nilvadipine and (S)-NB 818 via Regioselective Bromination of Chiral 1, 4-Dihydropyridines as a Key Step and Enzymatic Resolution of Racemic 2-Hydroxymethyl-1, 4-dihydropyridine Derivatives
EBIIKE, Hirosato, MARUYAMA, Kaori, OZAWA, Yumi, YAMAZAKI, Yukiyoshi, ACHIWA, Kazuo
Published in Chemical & pharmaceutical bulletin (1997)
Published in Chemical & pharmaceutical bulletin (1997)
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Lipase-catalyzed enantiosynthesis of (R)- and (S)-2-(Benzyl(phenyl)amino)ethyl 5-(5,5-Dimethyl-2-oxo-1,3,2-dioxaphosphorinan-2-yl)-1,4-dihydro-2,6-dimethyl-4-(3-nitrophenyl)-3-pyridinecarboxylate (NZ 105)
EBIIKE, Hirosato, YAMAZAKI, Yukiyoshi, ACHIWA, Kazuo
Published in Chemical & pharmaceutical bulletin (1995)
Published in Chemical & pharmaceutical bulletin (1995)
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