Novel orally bioavailable EZH1/2 dual inhibitors with greater antitumor efficacy than an EZH2 selective inhibitor
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Published in Cancer science (01.10.2017)
Published in Cancer science (01.10.2017)
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Modeling and Reproducibility of Suzaku HXD PIN/GSO Background
Fukazawa, Yasushi, Mizuno, Tsunefumi, Watanabe, Shin, Kokubun, Motohide, Takahashi, Hiromitsu, Kawano, Naomi, Nishino, Sho, Sasada, Mahito, Shirai, Hirohisa, Takahashi, Takuya, Umeki, Yudai, Yamasaki, Tomonori, Yasuda, Tomonori, Bamba, Aya, Ohno, Masanori, Takahashi, Tadayuki, Ushio, Masayoshi, Enoto, Teruaki, Kitaguchi, Takao, Makishima, Kazuhiro, Nakazawa, Kazuo, Uehara, Yuichi, Yamada, Shin’ya, Yuasa, Takayuki, Isobe, Naoki, Kawaharada, Madoka, Tanaka, Takaaki, Tashiro, Makoto S., Terada, Yukikatsu, Yamaoka, Kazutaka
Published in Publications of the Astronomical Society of Japan (30.01.2009)
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A Novel Inhibitor of I-KappaB Kinase Beta Ameliorates Experimental Arthritis through Downregulation of Proinflammatory Cytokines in Arthritic Joints
Tanaka, Shinji, Toki, Tadashi, Yokoyama, Mika, Shimizu, Hiroki, Yamasaki, Tomonori, Yoneda, Yoshiyuki, Muro, Fumihito, Yasukochi, Takanori, Iimura, Shin, Morishita, Kaoru
Published in Biological & pharmaceutical bulletin (01.01.2014)
Published in Biological & pharmaceutical bulletin (01.01.2014)
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Fe-K Line Probing of Material Around the Active Galactic Nucleus Central Engine with Suzaku
Fukazawa, Yasushi, Hiragi, Kazuyoshi, Mizuno, Motohiro, Nishino, Sho, Hayashi, Katsuhiro, Yamasaki, Tomonori, Shirai, Hirohisa, Takahashi, Hiromitsu, Ohno, Masanori
Published in The Astrophysical journal (20.01.2011)
Published in The Astrophysical journal (20.01.2011)
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Development and Characterization of the Novel Orally Bioavailable EZH1/2 Dual Inhibitor DS-3201
Honma, Daisuke, Adachi, Nobuaki, Kanno, Osamu, Watanabe, Jun, Hirasawa, Makoto, Nosaka, Emi, Shiroishi, Machiko, Takizawa, Takeshi, Yasumatsu, Isao, Horiuchi, Takao, Nakao, Akira, Suzuki, Keisuke, Yamasaki, Tomonori, Nakajima, Katsuyoshi, Hayakawa, Miho, Yamazaki, Takanori, Araki, Kazushi, Fujiwara, Kosaku
Published in Blood (08.12.2017)
Published in Blood (08.12.2017)
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Discovery of imidazo[1,2- b]pyridazines as IKKβ inhibitors. Part 3: Exploration of effective compounds in arthritis models
Shimizu, Hiroki, Yamasaki, Tomonori, Yoneda, Yoshiyuki, Muro, Fumihito, Hamada, Tomoaki, Yasukochi, Takanori, Tanaka, Shinji, Toki, Tadashi, Yokoyama, Mika, Morishita, Kaoru, Iimura, Shin
Published in Bioorganic & medicinal chemistry letters (01.08.2011)
Published in Bioorganic & medicinal chemistry letters (01.08.2011)
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Discovery of imidazo[1,2- b]pyridazine derivatives as IKKβ inhibitors. Part 1: Hit-to-lead study and structure–activity relationship
Shimizu, Hiroki, Tanaka, Shinji, Toki, Tadashi, Yasumatsu, Isao, Akimoto, Toshihiko, Morishita, Kaoru, Yamasaki, Tomonori, Yasukochi, Takanori, Iimura, Shin
Published in Bioorganic & medicinal chemistry letters (01.09.2010)
Published in Bioorganic & medicinal chemistry letters (01.09.2010)
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Discovery of imidazo[1,2- b]pyridazines as IKKβ inhibitors. Part 2: Improvement of potency in vitro and in vivo
Shimizu, Hiroki, Yasumatsu, Isao, Hamada, Tomoaki, Yoneda, Yoshiyuki, Yamasaki, Tomonori, Tanaka, Shinji, Toki, Tadashi, Yokoyama, Mika, Morishita, Kaoru, Iimura, Shin
Published in Bioorganic & medicinal chemistry letters (01.02.2011)
Published in Bioorganic & medicinal chemistry letters (01.02.2011)
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Fe-K LINE PROBING OF MATERIAL AROUND THE ACTIVE GALACTIC NUCLEUS CENTRAL ENGINE WITH SUZAKU
FUKAZAWA, Yasushi, HIRAGI, Kazuyoshi, MIZUNO, Motohiro, NISHINO, Sho, HAYASHI, Katsuhiro, YAMASAKI, Tomonori, SHIRAI, Hirohisa, TAKAHASHI, Hiromitsu, OHNO, Masanori
Published in The Astrophysical journal (2011)
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Published in The Astrophysical journal (2011)
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Revealing the High Energy Emission from the Obscured Seyfert Galaxy MCG−5–23–16 with Suzaku
Reeves, James N., Awaki, Hisamitsu, Dewangan, Gulab C., Fabian, Andy C., Fukazawa, Yasushi, Gallo, Luigi, Griffiths, Richard, Inoue, Hajime, Kunieda, Hideyo, Markowitz, Alex, Miniutti, Giovanni, Mizuno, Tsunefumi, Mushotzky, Richard, Okajima, Takashi, Ptak, Andy, Takahashi, Tadayuki, Terashima, Yuichi, Ushio, Masayoshi, Watanabe, Shin, Yamasaki, Tomonori, Yamauchi, Makoto, Yaqoob, Tahir
Published in Publications of the Astronomical Society of Japan (30.01.2007)
Published in Publications of the Astronomical Society of Japan (30.01.2007)
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WATANABE JUN, HORIUCHI TAKAO, KANNO OSAMU, ADACHI NOBUAKI, HONMA DAISUKE, HAMADA YOSHITO, YAMASAKI TOMONORI, NAKAO AKIRA, SUZUKI KEISUKE
Year of Publication 18.11.2016
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Year of Publication 18.11.2016
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Year of Publication 24.09.2015
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Year of Publication 24.09.2015
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Reduction of Peptide Character of HIV Protease Inhibitors That Exhibit Nanomolar Potency against Multidrug Resistant HIV-1 Strains
Tamamura, Hirokazu, Koh, Yasuhiro, Ueda, Satoshi, Sasaki, Yoshikazu, Yamasaki, Tomonori, Aoki, Manabu, Maeda, Kenji, Watai, Yoriko, Arikuni, Hisashi, Otaka, Akira, Mitsuya, Hiroaki, Fujii, Nobutaka
Published in Journal of medicinal chemistry (24.04.2003)
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IMIDAZO[1,2-B]PYRIDAZINE DERIVATIVE
YONEDA, YOSHIYUKI, YAMASAKI, TOMONORI, YASUKOCHI, TAKANORI, IIMURA, SHIN, SHIMIZU, HIROKI
Year of Publication 19.06.2008
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Year of Publication 19.06.2008
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Discovery of imidazo[1,2-b]pyridazine derivatives as IKKbeta inhibitors. Part 1: Hit-to-lead study and structure-activity relationship
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Published in Bioorganic & medicinal chemistry letters (01.09.2010)
Published in Bioorganic & medicinal chemistry letters (01.09.2010)
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YAMASAKI, TOMONORI, NAKAO, AKIRA, HAMADA, YOSHITO, SUZUKI, KEISUKE, KANNO, OSAMU, HONMA, DAISUKE, ADACHI, NOBUAKI, WATANABE, JUN, HORIUCHI, TAKAO
Year of Publication 29.08.2022
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Year of Publication 29.08.2022
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1,3-benzodioxole derivative
Horiuchi, Takao, Hamada, Yoshito, Kanno, Osamu, Suzuki, Keisuke, Adachi, Nobuaki, Yamasaki, Tomonori, Honma, Daisuke, Nakao, Akira, Watanabe, Jun
Year of Publication 23.03.2021
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Year of Publication 23.03.2021
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