Pharmacological evaluation of novel (6-aminopyridin-3-yl)(4-(pyridin-2-yl)piperazin-1-yl) methanone derivatives as TRPV4 antagonists for the treatment of pain
Tsuno, Naoki, Yukimasa, Akira, Yoshida, Osamu, Suzuki, Shinji, Nakai, Hiromi, Ogawa, Tomoyuki, Fujiu, Motohiro, Takaya, Kenji, Nozu, Azusa, Yamaguchi, Hiroki, Matsuda, Hidetoshi, Funaki, Satoko, Yamanada, Natsue, Tanimura, Miki, Nagamatsu, Daiki, Asaki, Toshiyuki, Horita, Narumi, Yamamoto, Miyuki, Hinata, Mikie, Soga, Masahiko, Imai, Masayuki, Morioka, Yasuhide, Kanemasa, Toshiyuki, Sakaguchi, Gaku, Iso, Yasuyoshi
Published in Bioorganic & medicinal chemistry (01.04.2017)
Published in Bioorganic & medicinal chemistry (01.04.2017)
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Creation of Novel Protein Transduction Domain (PTD) Mutants by a Phage Display-Based High-Throughput Screening System
Mukai, Yohei, Sugita, Toshiki, Yamato, Tomoko, Yamanada, Natsue, Shibata, Hiroko, Imai, Sunao, Abe, Yasuhiro, Nagano, Kazuya, Nomura, Tetsuya, Tsutsumi, Yasuo, Kamada, Haruhiko, Nakagawa, Shinsaku, Tsunoda, Shin-ichi
Published in Biological & Pharmaceutical Bulletin (2006)
Published in Biological & Pharmaceutical Bulletin (2006)
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Discovery of novel 2′,4′-dimethyl-[4,5′-bithiazol]-2-yl amino derivatives as orally bioavailable TRPV4 antagonists for the treatment of pain: Part 1
Tsuno, Naoki, Yukimasa, Akira, Yoshida, Osamu, Ichihashi, Yusuke, Inoue, Takatsugu, Ueno, Tatsuhiko, Yamaguchi, Hiroki, Matsuda, Hidetoshi, Funaki, Satoko, Yamanada, Natsue, Tanimura, Miki, Nagamatsu, Daiki, Nishimura, Yoko, Ito, Tetsuji, Soga, Masahiko, Horita, Narumi, Yamamoto, Miyuki, Hinata, Mikie, Imai, Masayuki, Morioka, Yasuhide, Kanemasa, Toshiyuki, Sakaguchi, Gaku, Iso, Yasuyoshi
Published in Bioorganic & medicinal chemistry letters (15.10.2016)
Published in Bioorganic & medicinal chemistry letters (15.10.2016)
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Improved cytosolic translocation and tumor-killing activity of Tat-shepherdin conjugates mediated by co-treatment with Tat-fused endosome-disruptive HA2 peptide
Sugita, Toshiki, Yoshikawa, Tomoaki, Mukai, Yohei, Yamanada, Natsue, Imai, Sunao, Nagano, Kazuya, Yoshida, Yasunobu, Shibata, Hiroko, Yoshioka, Yasuo, Nakagawa, Shinsaku, Kamada, Haruhiko, Tsunoda, Shin-ichi, Tsutsumi, Yasuo
Published in Biochemical and biophysical research communications (30.11.2007)
Published in Biochemical and biophysical research communications (30.11.2007)
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Organelle-Targeted Delivery of Biological Macromolecules Using the Protein Transduction Domain: Potential Applications for Peptide Aptamer Delivery into the Nucleus
Yoshikawa, Tomoaki, Sugita, Toshiki, Mukai, Yohei, Yamanada, Natsue, Nagano, Kazuya, Nabeshi, Hiromi, Yoshioka, Yasuo, Nakagawa, Shinsaku, Abe, Yasuhiro, Kamada, Haruhiko, Tsunoda, Shin-ichi, Tsutsumi, Yasuo
Published in Journal of molecular biology (25.07.2008)
Published in Journal of molecular biology (25.07.2008)
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