Sustained Morphine Treatment Augments Capsaicin-Evoked Calcitonin Gene-Related Peptide Release from Primary Sensory Neurons in a Protein Kinase A- and Raf-1-Dependent Manner
Tumati, Suneeta, Yamamura, Henry I, Vanderah, Todd W, Roeske, William R, Varga, Eva V
Published in The Journal of pharmacology and experimental therapeutics (01.09.2009)
Published in The Journal of pharmacology and experimental therapeutics (01.09.2009)
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Antinociceptive Structure-Activity Studies with Enkephalin-Based Opioid Glycopeptides
Elmagbari, Nura O, Egleton, Richard D, Palian, Michael M, Lowery, John J, Schmid, Wendi R, Davis, Peg, Navratilova, Edita, Dhanasekaran, Muthu, Keyari, Charles M, Yamamura, Henry I, Porreca, Frank, Hruby, Victor J, Polt, Robin, Bilsky, Edward J
Published in The Journal of pharmacology and experimental therapeutics (01.10.2004)
Published in The Journal of pharmacology and experimental therapeutics (01.10.2004)
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Constitutive Activity at the Cannabinoid CB1 Receptor Is Required for Behavioral Response to Noxious Chemical Stimulation of TRPV1: Antinociceptive Actions of CB1 Inverse Agonists
Fioravanti, Beatriz, De Felice, Milena, Stucky, Cheryl L, Medler, Karen A, Luo, Miaw-Chyi, Gardell, Luis R, Ibrahim, Mohab, Malan, T. Phil, Jr, Yamamura, Henry I, Ossipov, Michael H, King, Tamara, Lai, Josephine, Porreca, Frank, Vanderah, Todd W
Published in The Journal of neuroscience (05.11.2008)
Published in The Journal of neuroscience (05.11.2008)
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Unique agonist-bound cannabinoid CB1 receptor conformations indicate agonist specificity in signaling
GEORGIEVA, Teodora, DEVANATHAN, Savitha, STROPOVA, Dagmar, PARK, Chad K, SALAMON, Zdzislaw, TOLLIN, Gordon, HRUBY, Victor J, ROESKE, William R, YAMAMURA, Henry I, VARGA, Eva
Published in European journal of pharmacology (26.02.2008)
Published in European journal of pharmacology (26.02.2008)
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Discovery of a Potent and Efficacious Peptide Derivative for δ/μ Opioid Agonist/Neurokinin 1 Antagonist Activity with a 2′,6′-Dimethyl-l-Tyrosine: In vitro, In vivo, and NMR-Based Structural Studies
Yamamoto, Takashi, Nair, Padma, Largent-Milnes, Tally M, Jacobsen, Neil E, Davis, Peg, Ma, Shou-Wu, Yamamura, Henry I, Vanderah, Todd W, Porreca, Frank, Lai, Josephine, Hruby, Victor J
Published in Journal of medicinal chemistry (14.04.2011)
Published in Journal of medicinal chemistry (14.04.2011)
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Improving Metabolic Stability by Glycosylation: Bifunctional Peptide Derivatives That Are Opioid Receptor Agonists and Neurokinin 1 Receptor Antagonists
Yamamoto, Takashi, Nair, Padma, Jacobsen, Neil E, Vagner, Josef, Kulkarni, Vinod, Davis, Peg, Ma, Shou-wu, Navratilova, Edita, Yamamura, Henry I, Vanderah, Todd W, Porreca, Frank, Lai, Josephine, Hruby, Victor J
Published in Journal of medicinal chemistry (27.08.2009)
Published in Journal of medicinal chemistry (27.08.2009)
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Design, Synthesis, and Biological Evaluation of Novel Bifunctional C-Terminal-Modified Peptides for δ/μ Opioid Receptor Agonists and Neurokinin-1 Receptor Antagonists
Yamamoto, Takashi, Nair, Padma, Davis, Peg, Ma, Shou-wu, Navratilova, Edita, Moye, Sharif, Tumati, Suneeta, Lai, Josephine, Vanderah, Todd W, Yamamura, Henry I, Porreca, Frank, Hruby, Victor J
Published in Journal of medicinal chemistry (14.06.2007)
Published in Journal of medicinal chemistry (14.06.2007)
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The biological activity and metabolic stability of peptidic bifunctional compounds that are opioid receptor agonists and neurokinin-1 receptor antagonists with a cystine moiety
Yamamoto, Takashi, Nair, Padma, Ma, Shou-wu, Davis, Peg, Yamamura, Henry I., Vanderah, Todd W., Porreca, Frank, Lai, Josephine, Hruby, Victor J.
Published in Bioorganic & medicinal chemistry (15.10.2009)
Published in Bioorganic & medicinal chemistry (15.10.2009)
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A Structure–Activity Relationship Study and Combinatorial Synthetic Approach of C-Terminal Modified Bifunctional Peptides That Are δ/μ Opioid Receptor Agonists and Neurokinin 1 Receptor Antagonists
Yamamoto, Takashi, Nair, Padma, Vagner, Josef, Largent-Milnes, Tally, Davis, Peg, Ma, Shou-wu, Navratilova, Edita, Moye, Sharif, Tumati, Suneeta, Lai, Josephine, Yamamura, Henry I, Vanderah, Todd W, Porreca, Frank, Hruby, Victor J
Published in Journal of medicinal chemistry (13.03.2008)
Published in Journal of medicinal chemistry (13.03.2008)
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The Importance of Micelle-Bound States for the Bioactivities of Bifunctional Peptide Derivatives for δ/μ Opioid Receptor Agonists and Neurokinin 1 Receptor Antagonists
Yamamoto, Takashi, Nair, Padma, Jacobsen, Neil E, Davis, Peg, Ma, Shou-wu, Navratilova, Edita, Moye, Sharif, Lai, Josephine, Yamamura, Henry I, Vanderah, Todd W, Porreca, Frank, Hruby, Victor J
Published in Journal of medicinal chemistry (23.10.2008)
Published in Journal of medicinal chemistry (23.10.2008)
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Biological and Conformational Evaluation of Bifunctional Compounds for Opioid Receptor Agonists and Neurokinin 1 Receptor Antagonists Possessing Two Penicillamines
Yamamoto, Takashi, Nair, Padma, Jacobsen, Neil E, Kulkarni, Vinod, Davis, Peg, Ma, Shou-wu, Navratilova, Edita, Yamamura, Henry I, Vanderah, Todd W, Porreca, Frank, Lai, Josephine, Hruby, Victor J
Published in Journal of medicinal chemistry (12.08.2010)
Published in Journal of medicinal chemistry (12.08.2010)
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Direct Observation of G-protein Binding to the Human δ-Opioid Receptor Using Plasmon-Waveguide Resonance Spectroscopy
Alves, Isabel D., Salamon, Zdzislaw, Varga, Eva, Yamamura, Henry I., Tollin, Gordon, Hruby, Victor J.
Published in The Journal of biological chemistry (05.12.2003)
Published in The Journal of biological chemistry (05.12.2003)
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Sustained morphine treatment augments basal CGRP release from cultured primary sensory neurons in a Raf-1 dependent manner
Yue, Xu, Tumati, Suneeta, Navratilova, Edita, Strop, Dagmar, St John, Paul A., Vanderah, Todd W., Roeske, William R., Yamamura, Henry I., Varga, Eva V.
Published in European journal of pharmacology (28.04.2008)
Published in European journal of pharmacology (28.04.2008)
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Journal Article
Lipid Bilayers on Polyacrylamide Brushes for Inclusion of Membrane Proteins
Smith, Emily A, Coym, Jason W, Cowell, Scott M, Tokimoto, Takahira, Hruby, Victor J, Yamamura, Henry I, Wirth, Mary J
Published in Langmuir (11.10.2005)
Published in Langmuir (11.10.2005)
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Lanthanide-based time-resolved fluorescence of in cyto ligand–receptor interactions
Handl, Heather L, Vagner, Josef, Yamamura, Henry I, Hruby, Victor J, Gillies, Robert J
Published in Analytical biochemistry (15.07.2004)
Published in Analytical biochemistry (15.07.2004)
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Selectivity, cooperativity, and reciprocity in the interactions between the delta-opioid receptor, its ligands, and G-proteins
Alves, Isabel D, Ciano, Kathy A, Boguslavski, Valentina, Varga, Eva, Salamon, Zdzislaw, Yamamura, Henry I, Hruby, Victor J, Tollin, Gordon
Published in The Journal of biological chemistry (22.10.2004)
Published in The Journal of biological chemistry (22.10.2004)
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