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Published in Journal of medicinal chemistry (29.06.2000)
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Cannabinoid CB1 receptor expression, activation and detection of endogenous ligand in trabecular meshwork and ciliary process tissues
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Published in European journal of pharmacology (23.11.2001)
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Molecular biology and pharmacology of cloned opioid receptors
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Published in The FASEB journal (01.04.1995)
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Antinociceptive profile of biphalin, a dimeric enkephalin analog
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Published in The Journal of pharmacology and experimental therapeutics (01.06.1993)
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Published in The Journal of pharmacology and experimental therapeutics (01.06.1993)
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Glycopeptide Enkephalin Analogues Produce Analgesia in Mice: Evidence for Penetration of the Blood-Brain Barrier
Polt, Robin, Porreca, Frank, Szabo, Lajos Z., Bilsky, Edward J., Davis, Peg, Abbruscato, Thomas J., Davis, Thomas P., Horvath, Robert, Yamamura, Henry I., Hruby, Victor J.
Published in Proceedings of the National Academy of Sciences - PNAS (19.07.1994)
Published in Proceedings of the National Academy of Sciences - PNAS (19.07.1994)
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New endomorphin analogs with mu-agonist and delta-antagonist properties
Tóth, G., Keresztes, A., Tömböly, Cs, Péter, A., Fülöp, F., Tourwé, D., Navratilova, E., Varga, É., Roeske, W. R., Yamamura, H. I., Szucs, M., Borsodi, A.
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Published in Pure and applied chemistry (01.01.2004)
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Whole body and brain distribution of [3H]cyclic [D-Pen2,D-Pen5] enkephalin after intraperitoneal, intravenous, oral and subcutaneous administration
WEBER, S. J, GREENE, D. L, HRUBY, V. J, YAMAMURA, H. I, PORRECA, F, DAVIS, T. P
Published in The Journal of pharmacology and experimental therapeutics (01.12.1992)
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Published in The Journal of pharmacology and experimental therapeutics (01.12.1992)
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Relative efficacies of cannabinoid CB1 receptor agonists in the mouse brain
BURKEY, T. H, QUOCK, R. M, CONSROE, P, EHLERT, F. J, HOSOHATA, Y, ROESKE, W. R, YAMAMURA, H. I
Published in European journal of pharmacology (08.10.1997)
Published in European journal of pharmacology (08.10.1997)
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Characterization of [3H]naltrindole binding to delta opioid receptors in mouse brain and mouse vas deferens: evidence for delta opioid receptor heterogeneity
LEI FANG, KNAPP, R. J, HORVATH, R, MATSUNAGA, T. O, HAASETH, R. C, HRUBY, V. J, PORRECA, F, YAMAMURA, H. I
Published in The Journal of pharmacology and experimental therapeutics (01.02.1994)
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Published in The Journal of pharmacology and experimental therapeutics (01.02.1994)
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De Novo Design, Synthesis, and Biological Activities of High-Affinity and Selective Non-Peptide Agonists of the δ-Opioid Receptor
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Published in Journal of medicinal chemistry (19.11.1998)
Published in Journal of medicinal chemistry (19.11.1998)
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Biological activity of fragments and analogues of the potent dimeric opioid peptide, biphalin
Lipkowski, Andrzej W., Misicka, Aleksandra, Davis, Peg, Stropova, Dagmar, Janders, Jacqueline, Lachwa, Magdalena, Porreca, Frank, Yamamura, Henry I., Hruby, Victor J.
Published in Bioorganic & medicinal chemistry letters (20.09.1999)
Published in Bioorganic & medicinal chemistry letters (20.09.1999)
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Distribution and analgesia of [3H][D-Pen2, D-Pen5]enkephalin and two halogenated analogs after intravenous administration
Weber, S J, Greene, D L, Sharma, S D, Yamamura, H I, Kramer, T H, Burks, T F, Hruby, V J, Hersh, L B, Davis, T P
Published in The Journal of pharmacology and experimental therapeutics (01.12.1991)
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Published in The Journal of pharmacology and experimental therapeutics (01.12.1991)
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AM630 antagonism of cannabinoid-stimulated [ 35S]GTPγS binding in the mouse brain
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Published in European journal of pharmacology (19.02.1997)
Published in European journal of pharmacology (19.02.1997)
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Assessment of Stereoselectivity of Trimethylphenylalanine Analogues of δ‐Opioid [D‐Pen2,D‐Pen5]‐Enkephalin
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Published in Journal of neurochemistry (01.07.2000)
Published in Journal of neurochemistry (01.07.2000)
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Exploring the Structure−Activity Relationships of [1-(4-tert-Butyl-3‘-hydroxy)benzhydryl-4-benzylpiperazine] (SL-3111), A High-Affinity and Selective δ-Opioid Receptor Nonpeptide Agonist Ligand
Alfaro-Lopez, Josue, Okayama, Toru, Hosohata, Keiko, Davis, Peg, Porreca, Frank, Yamamura, Henry I, Hruby, Victor J
Published in Journal of medicinal chemistry (30.12.1999)
Published in Journal of medicinal chemistry (30.12.1999)
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Opiate Aromatic Pharmacophore Structure−Activity Relationships in CTAP Analogues Determined by Topographical Bias, Two-Dimensional NMR, and Biological Activity Assays
Bonner, G. Gregg, Davis, Peg, Stropova, Dagmar, Edsall, Sidney, Yamamura, Henry I, Porreca, Frank, Hruby, Victor J
Published in Journal of medicinal chemistry (24.02.2000)
Published in Journal of medicinal chemistry (24.02.2000)
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