Design and Synthesis of 2-(1-Alkylaminoalkyl)pyrazolo[1,5-a]pyrimidines as New Respiratory Syncytial Virus Fusion Protein Inhibitors
Yamaguchi-Sasaki, Toru, Tamura, Yunoshin, Ogata, Yuya, Kawaguchi, Takanori, Kurosaka, Jun, Sugaya, Yutaka, Iwakiri, Kanako, Busujima, Tsuyoshi, Takahashi, Ryo, Ueda-Yonemoto, Naoko, Tanigawa, Eiji, Abe-Kumasaka, Tomoko, Sugiyama, Hiroyuki, Kanuma, Kosuke
Published in Chemical & pharmaceutical bulletin (01.04.2020)
Published in Chemical & pharmaceutical bulletin (01.04.2020)
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Fragment-Based Discovery of Novel Non-Hydroxamate LpxC Inhibitors with Antibacterial Activity
Yamada, Yousuke, Takashima, Hajime, Walmsley, David Lee, Ushiyama, Fumihito, Matsuda, Yohei, Kanazawa, Harumi, Yamaguchi-Sasaki, Toru, Tanaka-Yamamoto, Nozomi, Yamagishi, Junya, Kurimoto-Tsuruta, Risa, Ogata, Yuya, Ohtake, Norikazu, Angove, Hayley, Baker, Lisa, Harris, Richard, Macias, Alba, Robertson, Alan, Surgenor, Allan, Watanabe, Hayato, Nakano, Koichiro, Mima, Masashi, Iwamoto, Kunihiko, Okada, Atsushi, Takata, Iichiro, Hitaka, Kosuke, Tanaka, Akihiro, Fujita, Kiyoko, Sugiyama, Hiroyuki, Hubbard, Roderick E
Published in Journal of medicinal chemistry (10.12.2020)
Published in Journal of medicinal chemistry (10.12.2020)
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Discovery of novel indole derivatives as potent and selective inhibitors of proMMP-9 activation
Nishikawa-Shimono, Rie, Kuwabara, Motoi, Fujisaki, Sho, Matsuda, Daisuke, Endo, Mayumi, Kamitani, Masafumi, Futamura, Aya, Nomura, Yusaku, Yamaguchi-Sasaki, Toru, Yabuuchi, Tetsuya, Yamaguchi, Chitose, Tanaka-Yamamoto, Nozomi, Satake, Shunya, Abe-Sato, Kumi, Funayama, Kosuke, Sakata, Mayumi, Takahashi, Shinji, Hirano, Koga, Fukunaga, Takuya, Uozumi, Yoriko, Kato, Sayaka, Tamura, Yunoshin, Nakamori, Tomoaki, Mima, Masashi, Mishima-Tsumagari, Chiemi, Nozawa, Dai, Imai, Yudai, Asami, Taiji
Published in Bioorganic & medicinal chemistry letters (01.01.2024)
Published in Bioorganic & medicinal chemistry letters (01.01.2024)
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Discovery of a potent dual inhibitor of wild-type and mutant respiratory syncytial virus fusion proteins through the modulation of atropisomer interconversion properties
Yamaguchi-Sasaki, Toru, Kawaguchi, Takanori, Okada, Atsushi, Tokura, Seiken, Tanaka-Yamamoto, Nozomi, Takeuchi, Tomoki, Ogata, Yuya, Takahashi, Ryo, Kurimoto-Tsuruta, Risa, Tamaoki, Tomokazu, Sugaya, Yutaka, Abe-Kumasaka, Tomoko, Arikawa, Kaho, Yoshida, Ippei, Sugiyama, Hiroyuki, Kanuma, Kosuke, Yoshinaga, Mitsukane
Published in Bioorganic & medicinal chemistry (15.12.2020)
Published in Bioorganic & medicinal chemistry (15.12.2020)
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Journal Article
Discovery of a Potent Dual Inhibitor of Wild-Type and Mutant Respiratory Syncytial Virus Fusion Proteins
Yamaguchi-Sasaki, Toru, Tokura, Seiken, Ogata, Yuya, Kawaguchi, Takanori, Sugaya, Yutaka, Takahashi, Ryo, Iwakiri, Kanako, Abe-Kumasaka, Tomoko, Yoshida, Ippei, Arikawa, Kaho, Sugiyama, Hiroyuki, Kanuma, Kosuke
Published in ACS medicinal chemistry letters (11.06.2020)
Published in ACS medicinal chemistry letters (11.06.2020)
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