Improvement of the Oral Drug Absorption of Topotecan through the Inhibition of Intestinal Xenobiotic Efflux Transporter, Breast Cancer Resistance Protein, by Excipients
YAMAGATA, Tetsuo, KUSUHARA, Hiroyuki, MORISHITA, Mariko, TAKAYAMA, Kozo, BENAMEUR, Hassan, SUGIYAMA, Yuichi
Published in Drug metabolism and disposition (01.07.2007)
Published in Drug metabolism and disposition (01.07.2007)
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Journal Article
Characterization of insulin protection properties of complexation hydrogels in gastric and intestinal enzyme fluids
Yamagata, Tetsuo, Morishita, Mariko, Kavimandan, Nikhil J., Nakamura, Koji, Fukuoka, Yu, Takayama, Kozo, Peppas, Nicholas A.
Published in Journal of controlled release (30.05.2006)
Published in Journal of controlled release (30.05.2006)
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Journal Article
Key functions in polymer carriers for intestinal absorption of insulin
Nakamura, Koji, Morishita, Mariko, Ehara, Junpei, Onuki, Yoshinori, Yamagata, Tetsuo, Kamei, Noriyasu, Lowman, Anthony M., Peppas, Nicholaos A., Takayma, Kozo
Published in International journal of pharmaceutics (16.04.2008)
Published in International journal of pharmaceutics (16.04.2008)
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Journal Article
Variability in P-glycoprotein inhibitory potency (IC₅₀) using various in vitro experimental systems: implications for universal digoxin drug-drug interaction risk assessment decision criteria
Bentz, Joe, O'Connor, Michael P, Bednarczyk, Dallas, Coleman, Joann, Lee, Caroline, Palm, Johan, Pak, Y Anne, Perloff, Elke S, Reyner, Eric, Balimane, Praveen, Brännström, Marie, Chu, Xiaoyan, Funk, Christoph, Guo, Ailan, Hanna, Imad, Herédi-Szabó, Krisztina, Hillgren, Kate, Li, Libin, Hollnack-Pusch, Evelyn, Jamei, Masoud, Lin, Xuena, Mason, Andrew K, Neuhoff, Sibylle, Patel, Aarti, Podila, Lalitha, Plise, Emile, Rajaraman, Ganesh, Salphati, Laurent, Sands, Eric, Taub, Mitchell E, Taur, Jan-Shiang, Weitz, Dietmar, Wortelboer, Heleen M, Xia, Cindy Q, Xiao, Guangqing, Yabut, Jocelyn, Yamagata, Tetsuo, Zhang, Lei, Ellens, Harma
Published in Drug metabolism and disposition (01.07.2013)
Published in Drug metabolism and disposition (01.07.2013)
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Journal Article
Comparison of methods for the prediction of human clearance from hepatocyte intrinsic clearance for a set of reference compounds and an external evaluation set
Yamagata, Tetsuo, Zanelli, Ugo, Gallemann, Dieter, Perrin, Dominique, Dolgos, Hugues, Petersson, Carl
Published in Xenobiotica (02.09.2017)
Published in Xenobiotica (02.09.2017)
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Journal Article
Application of receiver operating characteristic analysis to refine the prediction of potential digoxin drug interactions
Ellens, Harma, Deng, Shibing, Coleman, Joann, Bentz, Joe, Taub, Mitchell E, Ragueneau-Majlessi, Isabelle, Chung, Sophie P, Herédi-Szabó, Krisztina, Neuhoff, Sibylle, Palm, Johan, Balimane, Praveen, Zhang, Lei, Jamei, Masoud, Hanna, Imad, O'Connor, Michael, Bednarczyk, Dallas, Forsgard, Malin, Chu, Xiaoyan, Funk, Christoph, Guo, Ailan, Hillgren, Kathleen M, Li, Libin, Pak, Anne Y, Perloff, Elke S, Rajaraman, Ganesh, Salphati, Laurent, Taur, Jan-Shiang, Weitz, Dietmar, Wortelboer, Heleen M, Xia, Cindy Q, Xiao, Guangqing, Yamagata, Tetsuo, Lee, Caroline A
Published in Drug metabolism and disposition (01.07.2013)
Published in Drug metabolism and disposition (01.07.2013)
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Journal Article
Characterization of the inhibition of breast cancer resistance protein-mediated efflux of mitoxantrone by pharmaceutical excipients
Yamagata, Tetsuo, Morishita, Mariko, Kusuhara, Hiroyuki, Takayama, Kozo, Benameur, Hassan, Sugiyama, Yuichi
Published in International journal of pharmaceutics (31.03.2009)
Published in International journal of pharmaceutics (31.03.2009)
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Journal Article
Mucosal insulin delivery systems based on complexation polymer hydrogels: effect of particle size on insulin enteral absorption
Morishita, Mariko, Goto, Takahiro, Peppas, Nicholas A, Joseph, Jeffery I, Torjman, Marc C, Munsick, Carey, Nakamura, Koji, Yamagata, Tetsuo, Takayama, Kozo, Lowman, Anthony M
Published in Journal of controlled release (31.05.2004)
Published in Journal of controlled release (31.05.2004)
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Journal Article
In vitro and in vivo drug disposition of cilengitide in animals and human
Dolgos, Hugues, Freisleben, Achim, Wimmer, Elmar, Scheible, Holger, Krätzer, Friedrich, Yamagata, Tetsuo, Gallemann, Dieter, Fluck, Markus
Published in Pharmacology research & perspectives (01.04.2016)
Published in Pharmacology research & perspectives (01.04.2016)
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