Chelation-Mediated Palladium(II)-Catalyzed Domino Heck−Mizoroki/Suzuki−Miyaura Reactions Using Arylboronic Acids: Increasing Scope and Mechanistic Understanding
Yahiaoui, Samir, Fardost, Ashkan, Trejos, Alejandro, Larhed, Mats
Published in Journal of organic chemistry (15.04.2011)
Published in Journal of organic chemistry (15.04.2011)
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A Novel in vivo Anti-amnesic Agent, Specially Designed to Express Both Acetylcholinesterase (AChE) Inhibitory, Serotonergic Subtype 4 Receptor (5-HT 4 R) Agonist and Serotonergic Subtype 6 Receptor (5-HT 6 R) Inverse Agonist Activities, With a Potential Interest Against Alzheimer's Disease
Hatat, Bérénice, Yahiaoui, Samir, Lecoutey, Cédric, Davis, Audrey, Freret, Thomas, Boulouard, Michel, Claeysen, Sylvie, Rochais, Christophe, Dallemagne, Patrick
Published in Frontiers in aging neuroscience (19.06.2019)
Published in Frontiers in aging neuroscience (19.06.2019)
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A New PqsR Inverse Agonist Potentiates Tobramycin Efficacy to Eradicate Pseudomonas aeruginosa Biofilms
Schütz, Christian, Ho, Duy‐Khiet, Hamed, Mostafa Mohamed, Abdelsamie, Ahmed Saad, Röhrig, Teresa, Herr, Christian, Kany, Andreas Martin, Rox, Katharina, Schmelz, Stefan, Siebenbürger, Lorenz, Wirth, Marius, Börger, Carsten, Yahiaoui, Samir, Bals, Robert, Scrima, Andrea, Blankenfeldt, Wulf, Horstmann, Justus Constantin, Christmann, Rebekka, Murgia, Xabier, Koch, Marcus, Berwanger, Aylin, Loretz, Brigitta, Hirsch, Anna Katharina Herta, Hartmann, Rolf Wolfgang, Lehr, Claus‐Michael, Empting, Martin
Published in Advanced science (01.06.2021)
Published in Advanced science (01.06.2021)
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Journal Article
Refinement of arylthiosemicarbazone pharmacophore in inhibition of mushroom tyrosinase
Yi, Wei, Dubois, Carole, Yahiaoui, Samir, Haudecoeur, Romain, Belle, Catherine, Song, Huacan, Hardré, Renaud, Réglier, Marius, Boumendjel, Ahcène
Published in European journal of medicinal chemistry (01.09.2011)
Published in European journal of medicinal chemistry (01.09.2011)
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Journal Article
Identification of Xanthones as Selective Killers of Cancer Cells Overexpressing the ABC Transporter MRP1
Genoux-Bastide, Estelle, Lorendeau, Doriane, Nicolle, Edwige, Yahiaoui, Samir, Magnard, Sandrine, Di Pietro, Attilio, Baubichon-Cortay, Hélène, Boumendjel, Ahcène
Published in ChemMedChem (01.08.2011)
Published in ChemMedChem (01.08.2011)
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Data in support of substrate flexibility of a mutated acyltransferase domain and implications for polyketide biosynthesis
Klopries, Stephan, Bravo-Rodriguez, Kenny, Koopmans, Kyra R.M., Sundermann, Uschi, Yahiaoui, Samir, Arens, Julia, Kushnir, Susanna, Sanchez-Garcia, Elsa, Schulz, Frank
Published in Data in brief (01.12.2015)
Published in Data in brief (01.12.2015)
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Journal Article
Modified DRASTIC index model for groundwater vulnerability mapping using geostatistic methods and GIS in the Mitidja plain area (Algeria)
Boufekane, Abdelmadjid, Yahiaoui, Samir, Meddi, Hind, Meddi, Mohamed, Busico, Gianluigi
Published in Environmental forensics (01.11.2022)
Published in Environmental forensics (01.11.2022)
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Journal Article
Hydrogeochemical and isotopic assessment for characterizing groundwater quality in the Mitidja plain (northern Algeria)
Yahiaoui, Samir, Meddi, Mohamed, Razack, Moumtaz, Boufekane, Abdelmadjid, Bekkoussa, Belkacem Samir
Published in Environmental science and pollution research international (01.07.2023)
Published in Environmental science and pollution research international (01.07.2023)
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Journal Article
Substrate Flexibility of a Mutated Acyltransferase Domain and Implications for Polyketide Biosynthesis
Bravo-Rodriguez, Kenny, Klopries, Stephan, Koopmans, Kyra R.M., Sundermann, Uschi, Yahiaoui, Samir, Arens, Julia, Kushnir, Susanna, Schulz, Frank, Sanchez-Garcia, Elsa
Published in Chemistry & biology (19.11.2015)
Published in Chemistry & biology (19.11.2015)
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Journal Article
Dual inhibitors of Pseudomonas aeruginosa virulence factors LecA and LasB
Metelkina, Olga, Konstantinović, Jelena, Klein, Andreas, Shafiei, Roya, Fares, Mario, Alhayek, Alaa, Yahiaoui, Samir, Elgaher, Walid A M, Haupenthal, Jörg, Titz, Alexander, Hirsch, Anna K H
Published in Chemical science (Cambridge) (22.08.2024)
Published in Chemical science (Cambridge) (22.08.2024)
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Novel Multitarget-Directed Ligands (MTDLs) with Acetylcholinesterase (AChE) Inhibitory and Serotonergic Subtype 4 Receptor (5-HT4R) Agonist Activities As Potential Agents against Alzheimer’s Disease: The Design of Donecopride
Rochais, Christophe, Lecoutey, Cédric, Gaven, Florence, Giannoni, Patrizia, Hamidouche, Katia, Hedou, Damien, Dubost, Emmanuelle, Genest, David, Yahiaoui, Samir, Freret, Thomas, Bouet, Valentine, Dauphin, François, Sopkova de Oliveira Santos, Jana, Ballandonne, Céline, Corvaisier, Sophie, Malzert-Fréon, Aurélie, Legay, Remi, Boulouard, Michel, Claeysen, Sylvie, Dallemagne, Patrick
Published in Journal of medicinal chemistry (09.04.2015)
Published in Journal of medicinal chemistry (09.04.2015)
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Substrate‐Inspired Fragment Merging and Growing Affords Efficacious LasB Inhibitors
Kaya, Cansu, Walter, Isabell, Yahiaoui, Samir, Sikandar, Asfandyar, Alhayek, Alaa, Konstantinović, Jelena, Kany, Andreas M., Haupenthal, Jörg, Köhnke, Jesko, Hartmann, Rolf W., Hirsch, Anna K. H.
Published in Angewandte Chemie International Edition (26.01.2022)
Published in Angewandte Chemie International Edition (26.01.2022)
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Journal Article
Palladium(II)-catalyzed coupling reactions with a chelating vinyl ether and arylboronic acids: a new Heck/Suzuki domino diarylation reaction
Trejos, Alejandro, Fardost, Ashkan, Yahiaoui, Samir, Larhed, Mats
Published in Chemical communications (Cambridge, England) (01.01.2009)
Published in Chemical communications (Cambridge, England) (01.01.2009)
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N‑Aryl-3-mercaptosuccinimides as Antivirulence Agents Targeting Pseudomonas aeruginosa Elastase and Clostridium Collagenases
Konstantinović, Jelena, Yahiaoui, Samir, Alhayek, Alaa, Haupenthal, Jörg, Schönauer, Esther, Andreas, Anastasia, Kany, Andreas M, Müller, Rolf, Koehnke, Jesko, Berger, Fabian K, Bischoff, Markus, Hartmann, Rolf W, Brandstetter, Hans, Hirsch, Anna K. H
Published in Journal of medicinal chemistry (13.08.2020)
Published in Journal of medicinal chemistry (13.08.2020)
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Design, synthesis, and pharmacological evaluation of multitarget-directed ligands with both serotonergic subtype 4 receptor (5-HT4R) partial agonist and 5-HT6R antagonist activities, as potential treatment of Alzheimer’s disease
Yahiaoui, Samir, Hamidouche, Katia, Ballandonne, Céline, Davis, Audrey, de Oliveira Santos, Jana Sopkova, Freret, Thomas, Boulouard, Michel, Rochais, Christophe, Dallemagne, Patrick
Published in European journal of medicinal chemistry (04.10.2016)
Published in European journal of medicinal chemistry (04.10.2016)
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N -Aryl Mercaptopropionamides as Broad-Spectrum Inhibitors of Metallo-β-Lactamases
Kaya, Cansu, Konstantinović, Jelena, Kany, Andreas M, Andreas, Anastasia, Kramer, Jan S, Brunst, Steffen, Weizel, Lilia, Rotter, Marco J, Frank, Denia, Yahiaoui, Samir, Müller, Rolf, Hartmann, Rolf W, Haupenthal, Jörg, Proschak, Ewgenij, Wichelhaus, Thomas A, Hirsch, Anna K H
Published in Journal of medicinal chemistry (10.03.2022)
Published in Journal of medicinal chemistry (10.03.2022)
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