Selective Class I Phosphoinositide 3‑Kinase Inhibitors: Optimization of a Series of Pyridyltriazines Leading to the Identification of a Clinical Candidate, AMG 511
Norman, Mark H, Andrews, Kristin L, Bo, Yunxin Y, Booker, Shon K, Caenepeel, Sean, Cee, Victor J, D’Angelo, Noel D, Freeman, Daniel J, Herberich, Bradley J, Hong, Fang-Tsao, Jackson, Claire L. M, Jiang, Jian, Lanman, Brian A, Liu, Longbin, McCarter, John D, Mullady, Erin L, Nishimura, Nobuko, Pettus, Liping H, Reed, Anthony B, Miguel, Tisha San, Smith, Adrian L, Stec, Markian M, Tadesse, Seifu, Tasker, Andrew, Aidasani, Divesh, Zhu, Xiaochun, Subramanian, Raju, Tamayo, Nuria A, Wang, Ling, Whittington, Douglas A, Wu, Bin, Wu, Tian, Wurz, Ryan P, Yang, Kevin, Zalameda, Leeanne, Zhang, Nancy, Hughes, Paul E
Published in Journal of medicinal chemistry (13.09.2012)
Published in Journal of medicinal chemistry (13.09.2012)
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Journal Article
Structure-Based Design of a Novel Series of Potent, Selective Inhibitors of the Class I Phosphatidylinositol 3-Kinases
Smith, Adrian L, D’Angelo, Noel D, Bo, Yunxin Y, Booker, Shon K, Cee, Victor J, Herberich, Brad, Hong, Fang-Tsao, Jackson, Claire L. M, Lanman, Brian A, Liu, Longbin, Nishimura, Nobuko, Pettus, Liping H, Reed, Anthony B, Tadesse, Seifu, Tamayo, Nuria A, Wurz, Ryan P, Yang, Kevin, Andrews, Kristin L, Whittington, Douglas A, McCarter, John D, Miguel, Tisha San, Zalameda, Leeanne, Jiang, Jian, Subramanian, Raju, Mullady, Erin L, Caenepeel, Sean, Freeman, Daniel J, Wang, Ling, Zhang, Nancy, Wu, Tian, Hughes, Paul E, Norman, Mark H
Published in Journal of medicinal chemistry (14.06.2012)
Published in Journal of medicinal chemistry (14.06.2012)
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Journal Article
Correction to Selective Class I Phosphoinositide 3‑Kinase Inhibitors: Optimization of a Series of Pyridyltriazines Leading to the Identification of a Clinical Candidate, AMG 511
Norman, Mark H, Andrews, Kristin L, Bo, Yunxin Y, Booker, Shon K, Caenepeel, Sean, Cee, Victor J, D’Angelo, Noel D, Freeman, Daniel J, Herberich, Bradley J, Hong, Fang-Tsao, Jackson, Claire L. M, Jiang, Jian, Lanman, Brian A, Liu, Longbin, McCarter, John D, Mullady, Erin L, Nishimura, Nobuko, Pettus, Liping H, Reed, Anthony B, Miguel, Tisha San, Smith, Adrian L, Stec, Markian M, Tadesse, Seifu, Tasker, Andrew, Aidasani, Divesh, Zhu, Xiaochun, Subramanian, Raju, Tamayo, Nuria A, Wang, Ling, Whittington, Douglas A, Wu, Bin, Wu, Tian, Wurz, Ryan P, Yang, Kevin, Zalameda, Leeanne, Zhang, Nancy, Hughes, Paul E
Published in Journal of medicinal chemistry (25.10.2012)
Published in Journal of medicinal chemistry (25.10.2012)
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Journal Article
inibidores de pl3 quinase e/ou motor
KEVIN YANG, MARK H. NORMAN, NOEL D' ANGELO, BIN WU, BRIAN A. LANMAN, BRADLEY J. HERBERICH, RYAN WURZ, LIPING H. PETTUS, NOBUKO NISHIMURA, FANG- TSAO HONG, HONGYU LIAO, SEIFU TADESSE, CLAIRE L.M. JACKSON, ADRIAN L. SMITH, ANTHONY B. REED, NURIA A. TAMAYO, SHON BOOKER, VICTOR J. CEE, KRISTIN ANDREWS, YUNXIN Y. BO, LONGBIN LIU
Year of Publication 03.05.2016
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Year of Publication 03.05.2016
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Vanilloid receptor ligands and their use in treatments
Bo, Yunxin Y, Chakrabarti, Partha P, Chen, Ning, Liao, Hongyu, Norman, Mark H, Stec, Markian, Tamayo, Nuria, Wang, Xianghong
Year of Publication 27.11.2007
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Year of Publication 27.11.2007
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Inhibitors of PI3 kinase
KEVIN YANG, MARK H. NORMAN, HOLLY L. DEAK, KATHLEEN PANTER, MARIAN BRYAN, NOBUKO NISHIMURA, NURIA A. TAMAYO, SHON BOOKER, AARON C. SIEGMUND, YUNXIN Y. BO, KRISTIN ANDREWS, LONGBIN LIU, LAURIE SCHENKEL
Year of Publication 23.12.2009
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Year of Publication 23.12.2009
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Vanilloid receptor ligands and their use in treatments
Bo, Yunxin Y, Chakrabarti, Partha P, Chen, Ning, Doherty, Elizabeth M, Fotsch, Christopher H, Han, Nianhe, Kelly, Michael G, Liu, Qingyian, Norman, Mark Henry, Ognyanov, Vassil I, Wang, Xianghong, Zhu, Jiawang
Year of Publication 25.08.2009
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Year of Publication 25.08.2009
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Vanilloid receptor ligands and their use in treatments
QINGYIAN LIU, CHRISTOPHER H FOTSCH, MARK HENRY NORMAN, JIAWANG ZHU, YUNXIN Y BO, ELIZABETH M DOHERTY, XIANGHONG WANG, NIANHE HAN, MICHAEL G KELLY, NING CHEN, PARTHA P CHAKRABARTI
Year of Publication 22.11.2007
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Year of Publication 22.11.2007
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INHIBITORS OF PI3 KINASE
MARK H. NORMAN, KEVIN YANG, NURIA A. TAMAYO, YUNXIN Y. BO, AARON C. SIEGMUND, NOBUKO NISHIMURA, LONGBIN LIU
Year of Publication 14.12.2011
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Year of Publication 14.12.2011
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Vanilloid receptor ligands and their use in treatments
MICHAEL G. KELLY, QINGYIAN LIU, MARK HENRY NORMAN, JIAWANG ZHU, ELIZABETH M. DOHERTY, PARTHA P. CHAKRABARTI, YUNXIN Y. BO, CHRISTOPHER H. FOTSCH, XIANGHONG WANG, NIANHE HAN, NING CHEN
Year of Publication 01.02.2007
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Year of Publication 01.02.2007
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VANILLOID RECEPTOR LIGANDS AND THEIR USE IN TREATMENTS
MARK, HENRY NORMAN, QINGYIAN LIU, CHRISTOPHER, H. FOTSCH, ELIZABETH, M. DOHERTY, JIAWANG ZHU, YUNXIN, Y. BO, PARTHA, P. CHAKRABARTI, XIANGHONG WANG, NIANHE HAN, MICHAEL, G. KELLY, NING CHEN
Year of Publication 23.06.2003
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Year of Publication 23.06.2003
Patent
INHIBITORS OF PI3 KINASE
MARK H. NORMAN, KEVIN YANG, HOLLY L. DEAK, KATHLEEN PANTER, MARIAN BRYAN, NOBUKO NISHIMURA, NURIA A. TAMAYO, SHON BOOKER, YUNXIN Y. BO, AARON C. SIEGMUND, KRISTIN ANDREWS, LONGBIN LIU, LAURIE SCHENKEL
Year of Publication 20.12.2010
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Year of Publication 20.12.2010
Patent
INHIBITORS OF PI3 KINASE AND / OR MTOR
MARK H. NORMAN, KEVIN YANG, NOEL D´ANGELO, BIN WU, BRIAN A. LANMAN, BRADLEY J. HERBERICH, RYAN WURZ, LIPING H. PETTUS, NOBUKO NISHIMURA, SEIFU TADESSE, HONGYU LIAO, CLAIRE L.M. JACKSON, FANG-TSAO HONG, ADRIAN L. SMITH, NURIA A. TAMAYO, ANTHONY B. REED, SHON BOOKER, VICTOR J. CEE, YUNXIN Y. BO, KRISTIN ANDREWS, LONGBIN LIU
Year of Publication 18.11.2011
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Year of Publication 18.11.2011
Patent
INHIBITORS OF PI3 KINASE
YANG, KEVIN, NISHIMURA, NOBUKO, BO, YUNXIN Y, SIEGMUND, AARON C, TAMAYO, NURIA A, LIU, LONGBIN, NORMAN, MARK H
Year of Publication 11.02.2014
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Year of Publication 11.02.2014
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Inhibitors of PI3 kinase
NISHIMURA NOBUKO, TAMAYO NURIA A, BO YUNXIN Y, SIEGMUND AARON C, LIU LONGBIN, YANG KEVIN C, NORMAN MARK H
Year of Publication 20.05.2014
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Year of Publication 20.05.2014
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INHIBITORS OF PI3 KINASE
YANG, KEVIN, TAMAYO, NURIA, A, BO, YUNXIN, Y, NISHIMURA, NOBUKO, LIU, LONGBIN, NORMAN, MARK, H, SIEGMUND, AARON, C
Year of Publication 25.01.2012
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Year of Publication 25.01.2012
Patent
INHIBITORS OF PI3 KINASE
SCHENKEL, LAURIE, NISHIMURA, NOBUKO, BO, YUNXIN Y, TAMAYO, NURIA A, DEAK, HOLLY L, NORMAN, MARK H, PANTER, KATHLEEN, YANG, KEVIN, ANDREWS, KRISTIN, SIEGMUND, AARON C, BOOKER, SHON, LIU, LONGBIN, BRYAN, MARIAN
Year of Publication 17.06.2014
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Year of Publication 17.06.2014
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INHIBITORS OF PI3 KINASE
SCHENKEL, LAURIE, NISHIMURA, NOBUKO, BO, YUNXIN Y, TAMAYO, NURIA A, DEAK, HOLLY L, NORMAN, MARK H, PANTER, KATHLEEN, YANG, KEVIN, ANDREWS, KRISTIN, SIEGMUND, AARON C, BOOKER, SHON, LIU, LONGBIN, BRYAN, MARIAN
Year of Publication 23.04.2014
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Year of Publication 23.04.2014
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Inhibitors of PI3 kinase
YANG, KEVIN, NISHIMURA, NOBUKO, BO, YUNXIN Y, SIEGMUND, AARON C, TAMAYO, NURIA A, LIU, LONGBIN, NORMAN, MARK H
Year of Publication 06.10.2011
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Year of Publication 06.10.2011
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