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Published in Cancer research (Chicago, Ill.) (15.10.2009)
Published in Cancer research (Chicago, Ill.) (15.10.2009)
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Cabozantinib (XL184), a novel MET and VEGFR2 inhibitor, simultaneously suppresses metastasis, angiogenesis, and tumor growth
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Published in Molecular cancer therapeutics (01.12.2011)
Published in Molecular cancer therapeutics (01.12.2011)
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In vitro and in vivo activity of cabozantinib (XL184), an inhibitor of RET, MET, and VEGFR2, in a model of medullary thyroid cancer
Bentzien, Frauke, Zuzow, Marcus, Heald, Nathan, Gibson, Anna, Shi, Yongchang, Goon, Leanne, Yu, Peiwen, Engst, Stefan, Zhang, Wentao, Huang, Donghui, Zhao, Lora, Vysotskaia, Valentina, Chu, Felix, Bautista, Rajana, Cancilla, Belinda, Lamb, Peter, Joly, Alison H, Yakes, F Michael
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Published in Thyroid (New York, N.Y.) (01.12.2013)
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The Novel Bacterial N-Demethylase PdmAB Is Responsible for the Initial Step of N,N-Dimethyl-Substituted Phenylurea Herbicide Degradation
Gu, Tao, Zhou, Chaoyang, Sørensen, Sebastian R, Zhang, Ji, He, Jian, Yu, Peiwen, Yan, Xin, Li, Shunpeng
Published in Applied and Environmental Microbiology (01.12.2013)
Published in Applied and Environmental Microbiology (01.12.2013)
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Converting Immune Cold into Hot by Biosynthetic Functional Vesicles to Boost Systematic Antitumor Immunity
Wu, Ming, Zheng, Dongye, Zhang, Da, Yu, Peiwen, Peng, Lianli, Chen, Feng, Lin, Ziguo, Cai, Zhixiong, Li, Jiong, Wei, Zuwu, Lin, Xinyi, Liu, Jingfeng, Liu, Xiaolong
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Published in iScience (24.07.2020)
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Serum N-glycome characterization and anti-carbohydrate antibody profiling in oral squamous cell carcinoma patients
Guu, Shih-Yun, Lin, Tsung-Hsien, Chang, Su-Chieh, Wang, Rei-Jing, Hung, Ling-Yi, Fang, Po-Jan, Tang, Wei-Chien, Yu, Peiwen, Chang, Chuan-Fa
Published in PloS one (08.06.2017)
Published in PloS one (08.06.2017)
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Protocol to prepare functional cellular nanovesicles with PD1 and TRAIL to boost antitumor response
Yu, Peiwen, Zheng, Dongye, Zhang, Cuilin, Wu, Ming, Liu, Xiaolong
Published in STAR protocols (19.03.2021)
Published in STAR protocols (19.03.2021)
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Oral azacitidine preserves favorable level of fatigue and health-related quality of life for patients with acute myeloid leukemia in remission: results from the phase 3, placebo-controlled QUAZAR AML-001 trial
Roboz, Gail J, Döhner, Hartmut, Pocock, Christopher, Dombret, Herve, Ravandi, Farhad, Jang, Jun Ho, Selleslag, Dominik, Mayer, Jiři, Martens, Uwe M, Liesveld, Jane, Bernal, Teresa, Wang, Ming Chung, Yu, Peiwen, Shi, Ling, Guo, Shien, La Torre, Ignazia, Skikne, Barry, Dong, Qian, Braverman, Julia, Nehme, Salem Abi, Beach, C L, Wei, Andrew H
Published in Haematologica (Roma) (01.12.2021)
Published in Haematologica (Roma) (01.12.2021)
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Bridging the Gap between Preclinical and Clinical Studies Using Pharmacokinetic-Pharmacodynamic Modeling: An Analysis of GDC-0973, a MEK Inhibitor
WONG, Harvey, VERNILLET, Laurent, HOEFLICH, Klaus P, YONGCHANG SHI, AFTAB, Blake T, AOYAMA, Ron, TAN LAM, Sanh, BELVIN, Marcia, PRESCOTT, John, PETERSON, Amy, WARE, Joseph A, LEE, Lillian, MARTINI, Jean-Francois, PEIWEN YU, CONGFEN LI, DEL ROSARIO, Geoffrey, CHOO, Edna F
Published in Clinical cancer research (01.06.2012)
Published in Clinical cancer research (01.06.2012)
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The Selective PI3K Inhibitor XL147 (SAR245408) Inhibits Tumor Growth and Survival and Potentiates the Activity of Chemotherapeutic Agents in Preclinical Tumor Models
Foster, Paul, Yamaguchi, Kyoko, Hsu, Pin P, Qian, Fawn, Du, Xiangnan, Wu, Jianming, Won, Kwang-Ai, Yu, Peiwen, Jaeger, Christopher T, Zhang, Wentao, Marlowe, Charles K, Keast, Paul, Abulafia, Wendy, Chen, Jason, Young, Jenny, Plonowski, Artur, Yakes, F Michael, Chu, Felix, Engell, Kelly, Bentzien, Frauke, Lam, Sanh T, Dale, Stephanie, Yturralde, Olivia, Matthews, David J, Lamb, Peter, Laird, A Douglas
Published in Molecular cancer therapeutics (01.04.2015)
Published in Molecular cancer therapeutics (01.04.2015)
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Effect of Ionic Liquids on the Fibril-Formation and Gel Properties of Grass Carp (Ctenopharyngodon idellus) Skin Collagen
Zhai, Zhongwei, Wang, Haibo, Wei, Benmei, Yu, Peiwen, Xu, Chengzhi, He, Lang, Zhang, Juntao, Xu, Yuling
Published in Macromolecular research (01.07.2018)
Published in Macromolecular research (01.07.2018)
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Clinical observation of Yiqi Qingdu prescription on the treatment of intermediate-stage and advanced non-small-cell lung cancer
Liang, Qijun, Tang, Xiaoling, Yu, Jiong, Xiong, Monian, Zhu, Huifang, Xiong, Linkai, Zeng, Ru, Yu, Peiwen
Published in Journal of traditional Chinese medicine = Chung i tsa chih ying wen pan (01.04.2021)
Published in Journal of traditional Chinese medicine = Chung i tsa chih ying wen pan (01.04.2021)
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Novel Carboxamide-Based Allosteric MEK Inhibitors: Discovery and Optimization Efforts toward XL518 (GDC-0973)
Rice, Kenneth D, Aay, Naing, Anand, Neel K, Blazey, Charles M, Bowles, Owen J, Bussenius, Joerg, Costanzo, Simona, Curtis, Jeffry K, Defina, Steven C, Dubenko, Larisa, Engst, Stefan, Joshi, Anagha A, Kennedy, Abigail R, Kim, Angie I, Koltun, Elena S, Lougheed, Julie C, Manalo, Jean-Claire L, Martini, Jean-Francois, Nuss, John M, Peto, Csaba J, Tsang, Tsze H, Yu, Peiwen, Johnston, Stuart
Published in ACS medicinal chemistry letters (10.05.2012)
Published in ACS medicinal chemistry letters (10.05.2012)
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Discovery of XL413, a potent and selective CDC7 inhibitor
Koltun, Elena S., Tsuhako, Amy Lew, Brown, David S., Aay, Naing, Arcalas, Arlyn, Chan, Vicky, Du, Hongwang, Engst, Stefan, Ferguson, Kim, Franzini, Maurizio, Galan, Adam, Holst, Charles R., Huang, Ping, Kane, Brian, Kim, Moon H., Li, Jia, Markby, David, Mohan, Manisha, Noson, Kevin, Plonowski, Arthur, Richards, Steven J., Robertson, Scott, Shaw, Kenneth, Stott, Gordon, Stout, Thomas J., Young, Jenny, Yu, Peiwen, Zaharia, Cristiana A., Zhang, Wentao, Zhou, Peiwen, Nuss, John M., Xu, Wei, Kearney, Patrick C.
Published in Bioorganic & medicinal chemistry letters (01.06.2012)
Published in Bioorganic & medicinal chemistry letters (01.06.2012)
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The design, synthesis, and biological evaluation of PIM kinase inhibitors
Tsuhako, Amy Lew, Brown, David S., Koltun, Elena S., Aay, Naing, Arcalas, Arlyn, Chan, Vicky, Du, Hongwang, Engst, Stefan, Franzini, Maurizio, Galan, Adam, Huang, Ping, Johnston, Stuart, Kane, Brian, Kim, Moon H., Douglas Laird, A., Lin, Rui, Mock, Lillian, Ngan, Iris, Pack, Michael, Stott, Gordon, Stout, Thomas J., Yu, Peiwen, Zaharia, Cristiana, Zhang, Wentao, Zhou, Peiwen, Nuss, John M., Kearney, Patrick C., Xu, Wei
Published in Bioorganic & medicinal chemistry letters (01.06.2012)
Published in Bioorganic & medicinal chemistry letters (01.06.2012)
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Inhibition of the T790M Gatekeeper Mutant of the Epidermal Growth Factor Receptor by EXEL-7647
GENDREAU, Steven B, VENTURA, Richard, JACKMAN, Lisa, YONGCHANG SHI, PEIWEN YU, JING WANG, AFTAB, Dana T, JAEGER, Christopher T, MEYER, Stephanie M, DE COSTA, Anushka, ENGELL, Kelly, CHEN, Jason, KEAST, Paul, MARTINI, Jean-Francois, JOLY, Alison H, LAIRD, A. Douglas, YAKES, F. Michael, WENTAO ZHANG, BENTZIEN, Frauke, CANCILLA, Belinda, LUTMAN, Jeffery, CHU, Felix
Published in Clinical cancer research (15.06.2007)
Published in Clinical cancer research (15.06.2007)
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SAR and in vivo evaluation of 4-aryl-2-aminoalkylpyrimidines as potent and selective Janus kinase 2 (JAK2) inhibitors
Forsyth, Timothy, Kearney, Patrick C., Kim, Byung Gyu, Johnson, Henry W.B., Aay, Naing, Arcalas, Arlyn, Brown, David S., Chan, Vicky, Chen, Jeff, Du, Hongwang, Epshteyn, Sergey, Galan, Adam A., Huynh, Tai P., Ibrahim, Mohamed A., Kane, Brian, Koltun, Elena S., Mann, Grace, Meyr, Lisa E., Lee, Matthew S., Lewis, Gary L., Noguchi, Robin T., Pack, Michael, Ridgway, Brian H., Shi, Xian, Takeuchi, Craig S., Zu, Peiwen, Leahy, James W., Nuss, John M., Aoyama, Ron, Engst, Stefan, Gendreau, Steven B., Kassees, Robert, Li, Jia, Lin, Shwu-Hwa, Martini, Jean-Francois, Stout, Thomas, Tong, Philip, Woolfrey, John, Zhang, Wentao, Yu, Peiwen
Published in Bioorganic & medicinal chemistry letters (15.12.2012)
Published in Bioorganic & medicinal chemistry letters (15.12.2012)
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The design, synthesis, and biological evaluation of potent receptor tyrosine kinase inhibitors
Kim, Moon H., Tsuhako, Amy Lew, Co, Erick W., Aftab, Dana T., Bentzien, Frauke, Chen, Jason, Cheng, Wei, Engst, Stefan, Goon, Levina, Klein, Rhett R., Le, Donna T., Mac, Morrison, Parks, Jason J., Qian, Fawn, Rodriquez, Monica, Stout, Thomas J., Till, Jeffrey H., Won, Kwang-Ai, Wu, Xiang, Michael Yakes, F., Yu, Peiwen, Zhang, Wentao, Zhao, Yeping, Lamb, Peter, Nuss, John M., Xu, Wei
Published in Bioorganic & medicinal chemistry letters (01.08.2012)
Published in Bioorganic & medicinal chemistry letters (01.08.2012)
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