Enhanced oral bioavailability of koumine by complexation with hydroxypropyl-β-cyclodextrin: preparation, optimization, ex vivo and in vivo characterization
Hu, Qing, Fu, Xiaoling, Su, Yanping, Wang, Yanfang, Gao, Sihuan, Wang, Xiaoqin, Xu, Ying, Yu, Changxi
Published in Drug delivery (01.01.2021)
Published in Drug delivery (01.01.2021)
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Sempervirine Inhibits Proliferation and Promotes Apoptosis by Regulating Wnt/β-Catenin Pathway in Human Hepatocellular Carcinoma
Yue, Rongcai, Liu, Haiping, Huang, Yaxin, Wang, Jing, Shi, Dongmei, Su, Yanping, Luo, Yufei, Cai, Ping, Jin, Guilin, Yu, Changxi
Published in Frontiers in pharmacology (07.12.2021)
Published in Frontiers in pharmacology (07.12.2021)
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Investigation of the Possible Allostery of Koumine Extracted From Gelsemium elegans Benth. And Analgesic Mechanism Associated With Neurosteroids
Xiong, Bojun, You, Wenbing, Luo, Yufei, Jin, Guilin, Wu, Minxia, Xu, Ying, Yang, Jian, Huang, Huihui, Yu, Changxi
Published in Frontiers in pharmacology (04.10.2021)
Published in Frontiers in pharmacology (04.10.2021)
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Puerarin Alleviates Neuropathic Pain by Inhibiting Neuroinflammation in Spinal Cord
Liu, Suhuan, Li, Xuejun, Yu, Changxi, Liao, Kaijun, Liu, Ming, Yang, Shuyu
Published in Mediators of Inflammation (01.01.2014)
Published in Mediators of Inflammation (01.01.2014)
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Identification of Koumine as a Translocator Protein 18 kDa Positive Allosteric Modulator for the Treatment of Inflammatory and Neuropathic Pain
Xiong, Bojun, Jin, Guilin, Xu, Ying, You, Wenbing, Luo, Yufei, Fang, Menghan, Chen, Bing, Huang, Huihui, Yang, Jian, Lin, Xu, Yu, Changxi
Published in Frontiers in pharmacology (24.06.2021)
Published in Frontiers in pharmacology (24.06.2021)
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Immunoregulatory Effect of Koumine on Nonalcoholic Fatty Liver Disease Rats
Chu, Zhiyong, Yu, Changxi, Liu, Ming, Xu, Ying, Zhang, Chenxi, Su, Li, Huang, Huihui, Wei, Shanshan, Jin, Guilin, Yue, Rongcai, Yang, Jian
Published in Journal of Immunology Research (01.01.2019)
Published in Journal of Immunology Research (01.01.2019)
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Ventrolateral Periaqueductal Gray Astrocytes Regulate Nociceptive Sensation and Emotional Motivation in Diabetic Neuropathic Pain
Yang, Lan, Lu, Jingshan, Guo, Jianpeng, Chen, Jian, Xiong, Fangfang, Wang, Xinyao, Chen, Li, Yu, Changxi
Published in The Journal of neuroscience (26.10.2022)
Published in The Journal of neuroscience (26.10.2022)
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The anxiolytic effect of koumine on a predatory sound stress-induced anxiety model and its associated molecular mechanisms
Xiong, Bojun, Zhong, Zhifeng, Chen, Chaojie, Huang, Huihui, Lin, Jinxiang, Xu, Ying, Yang, Jian, Yu, Changxi
Published in Phytomedicine (Stuttgart) (01.08.2022)
Published in Phytomedicine (Stuttgart) (01.08.2022)
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The Modulatory Effect of Motor Cortex Astrocytes on Diabetic Neuropathic Pain
Lu, Jingshan, Yang, Lan, Xu, Ying, Ai, Lijing, Chen, Jian, Xiong, Fangfang, Hu, Lihuan, Chen, Huoshu, Liu, Jiyuan, Yan, Xiongbin, Huang, Huihui, Chen, Li, Yu, Changxi
Published in The Journal of neuroscience (16.06.2021)
Published in The Journal of neuroscience (16.06.2021)
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Novel neuroprotective pyromeconic acid derivatives with concurrent anti-Aβ deposition, anti-inflammatory, and anti-oxidation properties for treatment of Alzheimer's disease
Liu, Xueyan, Yu, Chuanyu, Yao, Yuxing, Lai, Huifang, Ye, Xiaoxia, Xu, Jiexin, Guo, Jianpeng, Xiao, Xian, Lin, Chen, Huang, Zhihong, Lin, Jin, Yu, Changxi, Zha, Daijun
Published in European journal of medicinal chemistry (15.02.2023)
Published in European journal of medicinal chemistry (15.02.2023)
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Formulation and Pharmacokinetic Evaluation of a Drug-in-Adhesive Patch for Transdermal Delivery of Koumine
Su, Yanping, Lu, Wenxiang, Fu, Xiaoling, Xu, Ying, Ye, Lixiang, Yang, Jian, Huang, Huihui, Yu, Changxi
Published in AAPS PharmSciTech (25.10.2020)
Published in AAPS PharmSciTech (25.10.2020)
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Facilitation of Behavioral and Cortical Emergence from Isoflurane Anesthesia by GABAergic Neurons in Basal Forebrain
Cai, Ping, Su, Wei-Kun, Zhang, Jin-Sheng, Liu, Pei-Chang, Liu, Feng, Liu, Ren-Fu, Li, Zhang-Shu, Zhu, Zhong-Hua, Xiao, Wen-Hao, Hu, Yong-Huai, Cai, Hong-Da, Wu, Xiao-Dan, Zhang, Liang-Cheng, Yu, Changxi, Chen, Li
Published in The Journal of neuroscience (19.04.2023)
Published in The Journal of neuroscience (19.04.2023)
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Regulation of wakefulness by astrocytes in the lateral hypothalamus
Cai, Ping, Huang, Sheng-Nan, Lin, Zhi-Hui, Wang, Zewu, Liu, Ren-Fu, Xiao, Wen-Hao, Li, Zhang-Shu, Zhu, Zhong-Hua, Yao, Jing, Yan, Xiong-Bin, Wang, Fu-Dan, Zeng, Shun-Xing, Chen, Guo-Qiang, Yang, Liu-Yun, Sun, Yu-Kun, Yu, Changxi, Chen, Li, Wang, Wen-Xiang
Published in Neuropharmacology (15.12.2022)
Published in Neuropharmacology (15.12.2022)
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Solid-State Forms of Koumine Hydrochloride: Phase Transformations and the Crystal Structure and Properties of the Stable Form
Su, Yanping, Shi, Dongmei, Xiong, Bojun, Xu, Ying, Hu, Qing, Huang, Huihui, Yang, Jian, Yu, Changxi
Published in ACS omega (30.08.2022)
Published in ACS omega (30.08.2022)
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A glutamatergic basal forebrain to midbrain circuit mediates wakefulness and defensive behavior
Cai, Ping, Chen, Hui-Yun, Tang, Wei-Tao, Hu, Yu-Duan, Chen, Shang-Yi, Lu, Jing-Shan, Lin, Zhi-Hui, Huang, Sheng-Nan, Hu, Li-Huan, Su, Wei-Kun, Li, Qi-Xuan, Lin, Zhi-Jie, Kang, Tian-Rui, Yan, Xiong-Bin, Liu, Pei-Chang, Chen, Li, Yin, Dou, Wu, Si-Ying, Li, Huang-Yuan, Yu, Changxi
Published in Neuropharmacology (01.05.2022)
Published in Neuropharmacology (01.05.2022)
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Journal Article
Koumine Attenuates Neuroglia Activation and Inflammatory Response to Neuropathic Pain
Yu, Changxi, Li, Su-Ping, Xu, Ying, Chen, Wan-Qing, Hong, Li-Mian, Lin, Shao-Mei, He, Sai-Di, Jin, Guilin, Yang, Jian
Published in Journal of neural transplantation & plasticity (01.01.2018)
Published in Journal of neural transplantation & plasticity (01.01.2018)
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Puerarin alleviates neuropathic pain by inhibiting neuroinfiammation in spinal cord
Liu, Ming, Liao, Kaijun, Yu, Changxi, Li, Xuejun, Liu, Suhuan, Yang, Shuyu
Published in Mediators of inflammation (01.01.2014)
Published in Mediators of inflammation (01.01.2014)
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