Design and Identification of a GPR40 Full Agonist (SCO-267) Possessing a 2‑Carbamoylphenyl Piperidine Moiety
Furukawa, Hideki, Miyamoto, Yasufumi, Hirata, Yasuhiro, Watanabe, Koji, Hitomi, Yuko, Yoshitomi, Yayoi, Aida, Jumpei, Noguchi, Naoyoshi, Takakura, Nobuyuki, Takami, Kazuaki, Miwatashi, Seiji, Hirozane, Yoshihiko, Hamada, Teruki, Ito, Ryo, Ookawara, Mitsugi, Moritoh, Yusuke, Watanabe, Masanori, Maekawa, Tsuyoshi
Published in Journal of medicinal chemistry (24.09.2020)
Published in Journal of medicinal chemistry (24.09.2020)
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Practical application of 3-substituted-2,6-difluoropyridines in drug discovery: Facile synthesis of novel protein kinase C theta inhibitors
Katoh, Taisuke, Tomata, Yoshihide, Setoh, Masaki, Sasaki, Satoshi, Takai, Takafumi, Yoshitomi, Yayoi, Yukawa, Tomoya, Nakagawa, Hideyuki, Fukumoto, Shoji, Tsukamoto, Tetsuya, Nakada, Yoshihisa
Published in Bioorganic & medicinal chemistry letters (01.06.2017)
Published in Bioorganic & medicinal chemistry letters (01.06.2017)
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Discovery of a novel B-cell lymphoma 6 (BCL6)–corepressor interaction inhibitor by utilizing structure-based drug design
Yasui, Takeshi, Yamamoto, Takeshi, Sakai, Nozomu, Asano, Kouhei, Takai, Takafumi, Yoshitomi, Yayoi, Davis, Melinda, Takagi, Terufumi, Sakamoto, Kotaro, Sogabe, Satoshi, Kamada, Yusuke, Lane, Weston, Snell, Gyorgy, Iwata, Masashi, Goto, Masayuki, Inooka, Hiroshi, Sakamoto, Jun-ichi, Nakada, Yoshihisa, Imaeda, Yasuhiro
Published in Bioorganic & medicinal chemistry (01.09.2017)
Published in Bioorganic & medicinal chemistry (01.09.2017)
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CYCLIC DINUCLEOTIDE AS STING (STIMULATOR OF INTERFERON GENES) AGONIST
SAITO MORIHISA, SHIOKAWA ZENYU, MURATA SHUMPEI, SEDO MASAKI, YOSHIKAWA MASATO, PAUL D GREENSPAN, YOSHITOMI YAYOI, TAWARAISHI TAISUKE, ODA TSUNEO, NAKADA YOSHIHISA, OKANIWA MASANORI, OKABE ATSUTOSHI, WADA YASUFUMI, MOCHIZUKI MICHIYO, KATO TAISUKE, SASAKI YUSUKE, HIDAKA KOSUKE, TOMINARI YUSUKE, SHIBUYA AKITO, SEKI MICHIHIRO, NAKAGAWA YASUO, BRIAN SCOTT FREEZE
Year of Publication 09.04.2020
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Year of Publication 09.04.2020
Patent
STING 작용제로서의 환식 다이뉴클레오타이드
GREENSPAN PAUL D, SHIOKAWA ZENYU, MURATA SHUMPEI, SEKI TOMOHIRO, YOSHIKAWA MASATO, YOSHITOMI YAYOI, TAWARAISHI TAISUKE, ODA TSUNEO, NAKADA YOSHIHISA, OKANIWA MASANORI, OKABE ATSUTOSHI, WADA YASUFUMI, MOCHIZUKI MICHIYO, KATO TAISUKE, SASAKI YUSUKE, HIDAKA KOSUKE, SAITOH MORIHISA, TOMINARI YUSUKE, SHIBUYA AKITO, FREEZE BRIAN SCOTT, SETO MASAKI, NAKAGAWA YASUO
Year of Publication 08.10.2019
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Year of Publication 08.10.2019
Patent
AROMATIC COMPOUND
TOKUNAGA, Norihito, FURUKAWA, Hideki, TAKAKURA, Nobuyuki, TAKAMI, Kazuaki, SHIBUYA, Akito, HITOMI, Yuko, MAEKAWA, Tsuyoshi, AIDA, Jumpei, KASAI, Shizuo, MIYAMOTO, Yasufumi, YOSHITOMI, Yayoi, MIWATASHI, Seiji, NOGUCHI, Naoyoshi, OKAWA, Tomohiro, WATANABE, Koji, KOBAYASHI, Toshitake, HIRATA, Yasuhiro
Year of Publication 04.10.2018
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Year of Publication 04.10.2018
Patent
CYCLIC DINUCLEOTIDE
SAITO MORIHISA, SHIOKAWA ZENYU, MURATA SHUMPEI, SEDO MASAKI, YOSHIKAWA MASATO, YOSHITOMI YAYOI, ODA TSUNEO, NAKADA YOSHIHISA, OKANIWA MASANORI, OKABE ATSUTOSHI, MOCHIZUKI MICHIYO, KATO TAISUKE, SASAKI YUSUKE, HIDAKA KOSUKE, TOMINARI YUSUKE, SHIBUYA AKITO, SEKI MICHIHIRO, NAKAGAWA YASUO
Year of Publication 14.06.2018
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Year of Publication 14.06.2018
Patent
HETEROCYCLIC COMPOUND
SASAKI, SATOSHI, TAKAI, TAKAFUMI, SETOH, MASAKI, KATOH, TAISUKE, NAKADA, YOSHIHISA, TOMATA, YOSHIHIDE, YOSHITOMI, YAYOI, YUKAWA, TOMOYA, TSUKAMOTO, TETSUYA, FUKUMOTO, SHOJI
Year of Publication 13.11.2014
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Year of Publication 13.11.2014
Patent
AROMATIC COMPOUND
MIWATASHI, SEIJI, TAKAKURA, NOBUYUKI, SHIBUYA, AKITO, AIDA, JUMPEI, HITOMI, YUKO, FURUKAWA, HIDEKI, WATANABE, KOJI, MIYAMOTO, YASUFUMI, OKAWA, TOMOHIRO, YOSHITOMI, YAYOI, HIRATA, YASUHIRO, NOGUCHI, NAOYOSHI
Year of Publication 12.02.2015
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Year of Publication 12.02.2015
Patent
CYCLIC DINUCLEOTIDE
Seto, Masaki, Shiokawa, Zenyu, Kato, Taisuke, Saitoh, Morihisa, Hidaka, Kosuke, Tominari, Yusuke, Mochizuki, Michiyo, Yoshitomi, Yayoi, Nakagawa, Yasuo, Yoshikawa, Masato, Seki, Tomohiro, Nakada, Yoshihisa, Shibuya, Akito
Year of Publication 13.05.2021
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Year of Publication 13.05.2021
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PYRAZOLOQUINAZOLINONE ANTITUMOR AGENTS
ASANO, Moriteru, FURUKAWA, Hideki, FOLEY, Michael A, YOSHITOMI, Yayoi, KAPOOR, Tarun, M, ASO, Kazuyoshi, OKAWA, Tomohiro, TAKASHIMA, Sachie, FUKASE, Yoshiyuki, HIRATA, Yasuhiro, TANAKA, Yuta
Year of Publication 18.11.2020
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Year of Publication 18.11.2020
Patent
CYCLIC DINUCLEOTIDES AS STING (STIMULATOR OF INTERFERON GENES) AGONISTS
SEKI, TOMOHIRO, SHIOKAWA, ZENYU, TOMINARI, YUSUKE, SHIBUYA, AKITO, MOCHIZUKI, MICHIYO, YOSHITOMI, YAYOI, NAKAGAWA, YASUO, MURATA, SHUMPEI, OKABE, ATSUTOSHI, SASAKI, YUSUKE, FREEZE, BRIAN SCOTT, GREENSPAN, PAUL D, KATO, TAISUKE, HIDAKA, KOSUKE, NAKADA, YOSHIHISA, SAITOH, MORIHISA, OKANIWA, MASANORI, SETO, MASAKI, YOSHIKAWA, MASATO, ODA, TSUNEO, TAWARAISHI, TAISUKE, WADA, YASUFUMI
Year of Publication 21.04.2022
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Year of Publication 21.04.2022
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PYRAZOLOQUINAZOLINONE ANTITUMOR AGENTS
ASANO, Moriteru, FURUKAWA, Hideki, FOLEY, Michael A, YOSHITOMI, Yayoi, ASO, Kazuyoshi, KAPOOR, Tarun M, OKAWA, Tomohiro, TAKASHIMA, Sachie, HIRATA, Yashuhiro, FUKASE, Yoshiyuki, TANAKA, Yuta
Year of Publication 14.05.2020
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Year of Publication 14.05.2020
Patent
Cyclic dinucleotides as STING (stimulator of interferon genes) agonists
Seto, Masaki, Shiokawa, Zenyu, Kato, Taisuke, Saitoh, Morihisa, Hidaka, Kosuke, Freeze, Brian Scott, Tominari, Yusuke, Oda, Tsuneo, Mochizuki, Michiyo, Yoshitomi, Yayoi, Nakagawa, Yasuo, Murata, Shumpei, Okaniwa, Masanori, Yoshikawa, Masato, Tawaraishi, Taisuke, Wada, Yasufumi, Seki, Tomohiro, Nakada, Yoshihisa, Okabe, Atsutoshi, Shibuya, Akito, Sasaki, Yusuke, Greenspan, Paul D
Year of Publication 10.03.2022
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Year of Publication 10.03.2022
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PYRAZOLOQUINAZOLINONE ANTITUMOR AGENTS
ASANO, Moriteru, FURUKAWA, Hideki, FOLEY, Michael A, YOSHITOMI, Yayoi, KAPOOR, Tarun, M, ASO, Kazuyoshi, OKAWA, Tomohiro, TAKASHIMA, Sachie, FUKASE, Yoshiyuki, HIRATA, Yasuhiro, TANAKA, Yuta
Year of Publication 25.03.2020
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Year of Publication 25.03.2020
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CYCLIC DINUCLEOTIDES AS STING (STIMULATOR OF INTEFERON GENES) AGONISTS
Seto, Masaki, Shiokawa, Zenyu, Kato, Taisuke, Saitoh, Morihisa, Hidaka, Kosuke, Freeze, Brian Scott, Tominari, Yusuke, Oda, Tsuneo, Mochizuki, Michiyo, Yoshitomi, Yayoi, Nakagawa, Yasuo, Murata, Shumpei, Okaniwa, Masanori, Yoshikawa, Masato, Tawaraishi, Taisuke, Wada, Yasufumi, Seki, Tomohiro, Nakada, Yoshihisa, Okabe, Atsutoshi, Shibuya, Akito, Sasaki, Yusuke, Greenspan, Paul D
Year of Publication 01.10.2021
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Year of Publication 01.10.2021
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CYCLIC DINUCLEOTIDES AS STING (STIMULATOR OF INTERFERON GENES) AGONISTS
ODA, Tsuneo, FREEZE, Brian Scott, OKABE, Atsutoshi, NAKADA, Yoshihisa, SHIBUYA, Akito, KATO, Taisuke, SAITOH, Morihisa, MOCHIZUKI, Michiyo, MURATA, Shumpei, SETO, Masaki, WADA, Yasufumi, SASAKI, Yusuke, TAWARAISHI, Taisuke, YOSHITOMI, Yayoi, NAKAGAWA, Yasuo, SHIOKAWA, Zenyu, YOSHIKAWA, Masato, GREENSPAN, Paul D, SEKI, Tomohiro, OKANIWA, Masanori, TOMINARI, Yusuke, HIDAKA, Kosuke
Year of Publication 28.09.2021
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Year of Publication 28.09.2021
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