Search Results - "YOSHIAKI WASHIO" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

DNA-Encoded Library Technology-Based Discovery, Lead Optimization, and Prodrug Strategy toward Structurally Unique Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors

DNA-Encoded Library Technology-Based Discovery, Lead Optimization, and Prodrug Strategy toward Structurally Unique Indoleamine 2,3-Dioxygenase-1 (IDO1) Inhibitors

by Kazmierski, Wieslaw M, Xia, Bing, Miller, John, De la Rosa, Martha, Favre, David, Dunham, Richard M, Washio, Yoshiaki, Zhu, Zhengrong, Wang, Feng, Mebrahtu, Makda, Deng, Hongfeng, Basilla, Jonathan, Wang, Liping, Evindar, Ghotas, Fan, Lijun, Olszewski, Alison, Prabhu, Ninad, Davie, Christopher, Messer, Jeffrey A, Samano, Vicente
Published in Journal of medicinal chemistry (09.04.2020)

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Journal Article

Optimization of Novel Indazoles as Highly Potent and Selective Inhibitors of Phosphoinositide 3‑Kinase δ for the Treatment of Respiratory Disease

Optimization of Novel Indazoles as Highly Potent and Selective Inhibitors of Phosphoinositide 3‑Kinase δ for the Treatment of Respiratory Disease

by Down, Kenneth, Amour, Augustin, Baldwin, Ian R, Cooper, Anthony W. J, Deakin, Angela M, Felton, Leigh M, Guntrip, Stephen B, Hardy, Charlotte, Harrison, Zoë A, Jones, Katherine L, Jones, Paul, Keeling, Suzanne E, Le, Joelle, Livia, Stefano, Lucas, Fiona, Lunniss, Christopher J, Parr, Nigel J, Robinson, Ed, Rowland, Paul, Smith, Sarah, Thomas, Daniel A, Vitulli, Giovanni, Washio, Yoshiaki, Hamblin, J. Nicole
Published in Journal of medicinal chemistry (24.09.2015)

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A Turing Test for Molecular Generators

A Turing Test for Molecular Generators

by Bush, Jacob T, Pogany, Peter, Pickett, Stephen D, Barker, Mike, Baxter, Andrew, Campos, Sebastien, Cooper, Anthony W. J, Hirst, David, Inglis, Graham, Nadin, Alan, Patel, Vipulkumar K, Poole, Darren, Pritchard, John, Washio, Yoshiaki, White, Gemma, Green, Darren V. S
Published in Journal of medicinal chemistry (22.10.2020)

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Identification and Optimization of Novel Small c‑Abl Kinase Activators Using Fragment and HTS Methodologies

Identification and Optimization of Novel Small c‑Abl Kinase Activators Using Fragment and HTS Methodologies

by Simpson, Graham L, Bertrand, Sophie M, Borthwick, Jennifer A, Campobasso, Nino, Chabanet, Julien, Chen, Susan, Coggins, Julia, Cottom, Josh, Christensen, Siegfried B, Dawson, Helen C, Evans, Helen L, Hobbs, Andrew N, Hong, Xuan, Mangatt, Biju, Munoz-Muriedas, Jordi, Oliff, Allen, Qin, Donghui, Scott-Stevens, Paul, Ward, Paris, Washio, Yoshiaki, Yang, Jingsong, Young, Robert J
Published in Journal of medicinal chemistry (28.02.2019)

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Discovery of Novel Benzimidazoles as Potent Inhibitors of TIE-2 and VEGFR-2 Tyrosine Kinase Receptors

Discovery of Novel Benzimidazoles as Potent Inhibitors of TIE-2 and VEGFR-2 Tyrosine Kinase Receptors

by Hasegawa, Masaichi, Nishigaki, Naohiko, Washio, Yoshiaki, Kano, Kazuya, Harris, Philip A, Sato, Hideyuki, Mori, Ichiro, West, Rob I, Shibahara, Megumi, Toyoda, Hiroko, Wang, Liping, Nolte, Robert T, Veal, James M, Cheung, Mui
Published in Journal of medicinal chemistry (06.09.2007)

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The Design of Potent, Selective and Drug-Like RGD alpha v beta 1 Small-Molecule Inhibitors Derived from non-RGD alpha 4 beta 1 Antagonists

The Design of Potent, Selective and Drug-Like RGD alpha v beta 1 Small-Molecule Inhibitors Derived from non-RGD alpha 4 beta 1 Antagonists

by Hatley, Richard J. D., Barrett, Tim N., Slack, Robert J., Watson, Morag E., Baillache, Daniel J., Gruszka, Anna, Washio, Yoshiaki, Rowedder, James E., Pogany, Peter, Pal, Sandeep, Macdonald, Simon J. F.
Published in ChemMedChem (17.07.2019)

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Journal Article

The Design of Potent, Selective and Drug‐Like RGD αvβ1 Small‐Molecule Inhibitors Derived from non‐RGD α4β1 Antagonists

The Design of Potent, Selective and Drug‐Like RGD αvβ1 Small‐Molecule Inhibitors Derived from non‐RGD α4β1 Antagonists

by Hatley, Richard J. D., Barrett, Tim N., Slack, Robert J., Watson, Morag E., Baillache, Daniel J., Gruszka, Anna, Washio, Yoshiaki, Rowedder, James E., Pogány, Peter, Pal, Sandeep, Macdonald, Simon J. F.
Published in ChemMedChem (17.07.2019)

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Journal Article

The Discovery of in Vivo Active Mitochondrial Branched-Chain Aminotransferase (BCATm) Inhibitors by Hybridizing Fragment and HTS Hits

The Discovery of in Vivo Active Mitochondrial Branched-Chain Aminotransferase (BCATm) Inhibitors by Hybridizing Fragment and HTS Hits

by Bertrand, Sophie M, Ancellin, Nicolas, Beaufils, Benjamin, Bingham, Ryan P, Borthwick, Jennifer A, Boullay, Anne-Bénédicte, Boursier, Eric, Carter, Paul S, Chung, Chun-wa, Churcher, Ian, Dodic, Nerina, Fouchet, Marie-Hélène, Fournier, Charlène, Francis, Peter L, Gummer, Laura A, Herry, Kenny, Hobbs, Andrew, Hobbs, Clare I, Homes, Paul, Jamieson, Craig, Nicodeme, Edwige, Pickett, Stephen D, Reid, Iain H, Simpson, Graham L, Sloan, Lisa A, Smith, Sarah E, Somers, Donald O’N, Spitzfaden, Claus, Suckling, Colin J, Valko, Klara, Washio, Yoshiaki, Young, Robert J
Published in Journal of medicinal chemistry (24.09.2015)

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Journal Article

From PIM1 to PI3Kδ via GSK3β: Target Hopping through the Kinome

From PIM1 to PI3Kδ via GSK3β: Target Hopping through the Kinome

by Henley, Zoë A, Bax, Benjamin D, Inglesby, Laura M, Champigny, Aurélie, Gaines, Simon, Faulder, Paul, Le, Joelle, Thomas, Daniel A, Washio, Yoshiaki, Baldwin, Ian R
Published in ACS medicinal chemistry letters (12.10.2017)

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Journal Article

ACYCLIC 1,2-ASYMMETRIC INDUCTION IN ADDITION-REACTIONS OF ALKYL RADICALS TO CHIRAL OLEFINS

ACYCLIC 1,2-ASYMMETRIC INDUCTION IN ADDITION-REACTIONS OF ALKYL RADICALS TO CHIRAL OLEFINS

by MORIKAWA, T, WASHIO, Y, SHIRO, M, TAGUCHI, T
Published in Chemistry letters (01.02.1993)

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Journal Article

Structure-guided optimization of small molecule c-Abl activators

Structure-guided optimization of small molecule c-Abl activators

by Hong, Xuan, Cao, Ping, Washio, Yoshiaki, Simpson, Graham, Campobasso, Nino, Yang, Jingsong, Borthwick, Jennifer, Burton, George, Chabanet, Julien, Bertrand, Sophie, Evans, Helen, Young, Robert J., Qu, Junya, Li, Hu, Cottom, Josh, Ward, Paris, Zhang, Hong, Ho, Thau, Qin, Donghui, Christensen, Siegfried, Head, Martha S.
Published in Journal of computer-aided molecular design (01.02.2014)

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Anilinopyrazole as selective CDK2 inhibitors: design, synthesis, biological evaluation, and x-ray crystallographic analysis

Anilinopyrazole as selective CDK2 inhibitors: design, synthesis, biological evaluation, and x-ray crystallographic analysis

by Tang, Jun, Shewchuk, Lisa M., Sato, Hideyuki, Hasegawa, Masaichi, Washio, Yoshiaki, Nishigaki, Naohiko
Published in Bioorganic & medicinal chemistry letters (15.09.2003)

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Journal Article

FLUORESCENT DISPLAY DEVICE

FLUORESCENT DISPLAY DEVICE

by HIROSHI, YAMAGUCHI, YOSHIAKI, WASHIO
Year of Publication 16.04.1998

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Patent

Anilinopyrazole as selective CDK2 inhibitors

Anilinopyrazole as selective CDK2 inhibitors

by Tang, Jun, Shewchuk, Lisa M., Sato, Hideyuki, Hasegawa, Masaichi, Washio, Yoshiaki, Nishigaki, Naohiko
Published in Bioorganic & medicinal chemistry letters (01.09.2003)

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Journal Article

ATOMIC-LAYER DEPOSITION APPARATUS AND ATOMIC-LAYER DEPOSITION METHOD

ATOMIC-LAYER DEPOSITION APPARATUS AND ATOMIC-LAYER DEPOSITION METHOD

by WASHIO YOSHIAKI
Year of Publication 06.10.2011

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Patent

ATOMIC LAYER DEPOSITION DEVICE AND ATOMIC LAYER DEPOSITION METHOD

ATOMIC LAYER DEPOSITION DEVICE AND ATOMIC LAYER DEPOSITION METHOD

by WASHIO YOSHIAKI
Year of Publication 29.09.2011

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Patent

ATOMIC LAYER DEPOSITION METHOD AND ATOMIC LAYER DEPOSITION DEVICE

ATOMIC LAYER DEPOSITION METHOD AND ATOMIC LAYER DEPOSITION DEVICE

by WASHIO YOSHIAKI
Year of Publication 15.09.2011

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Patent

Anilinopyrazole as selective CDK2 inhibitors: Design, synthesis, biological evaluation, and X-ray crystallographic analysis: Recent advances in the design of kinase inhibitors as novel therapeutic agents

Anilinopyrazole as selective CDK2 inhibitors: Design, synthesis, biological evaluation, and X-ray crystallographic analysis: Recent advances in the design of kinase inhibitors as novel therapeutic agents

by JUN TANG, SHEWCHUK, Lisa M, SATO, Hideyuki, HASEGAWA, Masaichi, WASHIO, Yoshiaki, NISHIGAKI, Naohiko
Published in Bioorganic & medicinal chemistry letters (2003)

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Journal Article

ATOMIC LAYER DEPOSITION DEVICE AND METHOD THEREFOR

ATOMIC LAYER DEPOSITION DEVICE AND METHOD THEREFOR

by WASHIO YOSHIAKI
Year of Publication 16.09.2010

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Patent

SUBSTITUTE ISOQUINOLINES USEFUL IN THE TREATMENT OF DISEASES SUCH AS CANCER AND ATHEROSCLEROSIS

SUBSTITUTE ISOQUINOLINES USEFUL IN THE TREATMENT OF DISEASES SUCH AS CANCER AND ATHEROSCLEROSIS

by WASHIO YOSHIAKI
Year of Publication 26.11.2009

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Patent

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