Discovery of (1R,2S)‑2-{[(2,4-Dimethylpyrimidin-5-yl)oxy]methyl}-2-(3-fluorophenyl)‑N‑(5-fluoropyridin-2-yl)cyclopropanecarboxamide (E2006): A Potent and Efficacious Oral Orexin Receptor Antagonist
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Published in Journal of medicinal chemistry (11.06.2015)
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Isolation of a Diterpenoid Substance with Potent Neuroprotective Activity from Fetal Calf Serum
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Published in Proceedings of the National Academy of Sciences - PNAS (05.03.2002)
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Practical Synthesis of Chiral Emopamil Left Hand as a Bioactive Motif
Kimura, Teiji, Yamamoto, Noboru, Suzuki, Yuichi, Kawano, Koki, Norimine, Yoshihiko, Ito, Koichi, Nagato, Satoshi, Iimura, Yoichi, Yonaga, Masahiro
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Published in Journal of organic chemistry (23.08.2002)
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Synthesis and absolute configuration of serofendic acids
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Published in Tetrahedron letters (13.05.2002)
Published in Tetrahedron letters (13.05.2002)
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Discovery of 2‑(2-Oxo-1-phenyl-5-pyridin-2-yl-1,2-dihydropyridin-3-yl)benzonitrile (Perampanel): A Novel, Noncompetitive α‑Amino-3-hydroxy-5-methyl-4-isoxazolepropanoic Acid (AMPA) Receptor Antagonist
Hibi, Shigeki, Ueno, Koshi, Nagato, Satoshi, Kawano, Koki, Ito, Koichi, Norimine, Yoshihiko, Takenaka, Osamu, Hanada, Takahisa, Yonaga, Masahiro
Published in Journal of medicinal chemistry (13.12.2012)
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Synthesis of Optically Active Methyl 7.BETA.-Hydroxykaurenoate with Potent Neuroprotective Activity
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Published in Chemical & pharmaceutical bulletin (2004)
Published in Chemical & pharmaceutical bulletin (2004)
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One-Pot Primary Aminomethylation of Aryl and Heteroaryl Halides with Sodium Phthalimidomethyltrifluoroborate
Murai, Norio, Miyano, Masayuki, Yonaga, Masahiro, Tanaka, Keigo
Published in Organic letters (01.06.2012)
Published in Organic letters (01.06.2012)
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Synthesis and Structure–Activity Relationships of Pyrazolo[1,5-a]pyridine Derivatives: Potent and Orally Active Antagonists of Corticotropin-Releasing Factor 1 Receptor
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Published in Journal of medicinal chemistry (14.06.2012)
Published in Journal of medicinal chemistry (14.06.2012)
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Design, synthesis, and structure–activity relationships of a series of novel N-aryl-2-phenylcyclopropanecarboxamide that are potent and orally active orexin receptor antagonists
Yoshida, Yu, Terauchi, Taro, Naoe, Yoshimitsu, Kazuta, Yuji, Ozaki, Fumihiro, Beuckmann, Carsten T., Nakagawa, Makoto, Suzuki, Michiyuki, Kushida, Ikuo, Takenaka, Osamu, Ueno, Takashi, Yonaga, Masahiro
Published in Bioorganic & medicinal chemistry (01.11.2014)
Published in Bioorganic & medicinal chemistry (01.11.2014)
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Dopamine D3 agonists disrupt social behavior in rats
KAGAYA, T.K, YONAGA, M, FURUYA, Y, HASHIMOTO, T, KUROKI, J, NISHIZAWA, Y
Published in Brain research (20.05.1996)
Published in Brain research (20.05.1996)
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Design, synthesis and structure–activity relationships of 5-alkylaminolquinolines as a novel series of CRF1 receptor antagonists
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Published in Bioorganic & medicinal chemistry letters (15.07.2012)
Published in Bioorganic & medicinal chemistry letters (15.07.2012)
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Design, synthesis, and structure–activity relationships of a series of 2-Ar-8-methyl-5-alkylaminoquinolines as novel CRF1 receptor antagonists
Takeda, Kunitoshi, Terauchi, Taro, Hashizume, Minako, Shin, Kogyoku, Ino, Mitsuhiro, Shibata, Hisashi, Yonaga, Masahiro
Published in Bioorganic & medicinal chemistry letters (01.09.2012)
Published in Bioorganic & medicinal chemistry letters (01.09.2012)
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Corrigendum to “Design, synthesis, and structure–activity relationships of a series of novel N-aryl-2-phenylcyclopropanecarboxamide that are potent and orally active orexin receptor antagonists” [Bioorg. Med. Chem. 22 (2014) 6071–6088]
Yoshida, Yu, Terauchi, Taro, Naoe, Yoshimitsu, Kazuta, Yuji, Ozaki, Fumihiro, Beuckmann, Carsten T., Nakagawa, Makoto, Suzuki, Michiyuki, Kushida, Ikuo, Takenaka, Osamu, Ueno, Takashi, Yonaga, Masahiro
Published in Bioorganic & medicinal chemistry (01.07.2015)
Published in Bioorganic & medicinal chemistry (01.07.2015)
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