A Review on GABA/Glutamate Pathway for Therapeutic Intervention of ASD and ADHD
Purkayastha, Priyanka, Malapati, Aruna, Yogeeswari, Perumal, Sriram, Dharmarajan
Published in Current medicinal chemistry (04.05.2015)
Published in Current medicinal chemistry (04.05.2015)
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Journal Article
Discovery of Antimycobacterial Spiro-piperidin-4-ones: An Atom Economic, Stereoselective Synthesis, and Biological Intervention
Kumar, Raju Ranjith, Perumal, Subbu, Senthilkumar, Palaniappan, Yogeeswari, Perumal, Sriram, Dharmarajan
Published in Journal of medicinal chemistry (25.09.2008)
Published in Journal of medicinal chemistry (25.09.2008)
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Journal Article
Design, synthesis and biological evaluation of imidazo[2,1-b]thiazole and benzo[d]imidazo[2,1-b]thiazole derivatives as Mycobacterium tuberculosis pantothenate synthetase inhibitors
Samala, Ganesh, Devi, Parthiban Brindha, Saxena, Shalini, Meda, Nikhila, Yogeeswari, Perumal, Sriram, Dharmarajan
Published in Bioorganic & medicinal chemistry (15.03.2016)
Published in Bioorganic & medicinal chemistry (15.03.2016)
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Journal Article
Design, Synthesis, and Structure–Activity Correlations of Novel Dibenzo[b,d]furan, Dibenzo[b,d]thiophene, and N-Methylcarbazole Clubbed 1,2,3-Triazoles as Potent Inhibitors of Mycobacterium tuberculosis
Patpi, Santhosh Reddy, Pulipati, Lokesh, Yogeeswari, Perumal, Sriram, Dharmarajan, Jain, Nishant, Sridhar, Balasubramanian, Murthy, Ramalinga, T, Anjana Devi, Kalivendi, Shasi Vardhan, Kantevari, Srinivas
Published in Journal of medicinal chemistry (26.04.2012)
Published in Journal of medicinal chemistry (26.04.2012)
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Journal Article
Design, Synthesis, and Evaluation of Thiol-Activated Sources of Sulfur Dioxide (SO2) as Antimycobacterial Agents
Malwal, Satish R, Sriram, Dharmarajan, Yogeeswari, Perumal, Konkimalla, V. Badireenath, Chakrapani, Harinath
Published in Journal of medicinal chemistry (12.01.2012)
Published in Journal of medicinal chemistry (12.01.2012)
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Journal Article
Design, development of new synthetic methodology, and biological evaluation of substituted quinolines as new anti-tubercular leads
Tanwar, Babita, Kumar, Asim, Yogeeswari, Perumal, Sriram, Dharmarajan, Chakraborti, Asit K.
Published in Bioorganic & medicinal chemistry letters (15.12.2016)
Published in Bioorganic & medicinal chemistry letters (15.12.2016)
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Journal Article
A facile synthesis and antimycobacterial evaluation of novel spiro-pyrido-pyrrolizines and pyrrolidines
Ranjith Kumar, Raju, Perumal, Subbu, Senthilkumar, Palaniappan, Yogeeswari, Perumal, Sriram, Dharmarajan
Published in European journal of medicinal chemistry (01.09.2009)
Published in European journal of medicinal chemistry (01.09.2009)
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Journal Article
Synthesis of novel cytotoxic tetracyclic acridone derivatives and study of their molecular docking, ADMET, QSAR, bioactivity and protein binding properties
Veligeti, Rajkumar, Madhu, Rajesh Bagepalli, Anireddy, Jayashree, Pasupuleti, Visweswara Rao, Avula, Vijaya Kumar Reddy, Ethiraj, Krishna S, Uppalanchi, Srinivas, Kasturi, Sivaprasad, Perumal, Yogeeswari, Anantaraju, Hasitha Shilpa, Polkam, Naveen, Guda, Mallilkarjuna Reddy, Vallela, Swetha, Zyryanov, Grigory Vasilievich
Published in Scientific reports (26.11.2020)
Published in Scientific reports (26.11.2020)
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Journal Article
Targeting hexokinase 2 for oral cancer therapy: structure-based design and validation of lead compounds
Chakraborty, Purbali, Lubna, Syeda, Bhuin, Shouvik, K, Deepika, Chakravarty, Manab, Jamma, Trinath, Yogeeswari, Perumal
Published in Frontiers in pharmacology (11.03.2024)
Published in Frontiers in pharmacology (11.03.2024)
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Journal Article
Design and synthesis of oxaprozin‐1,3,4‐oxadiazole hybrids as potential anticancer and antibacterial agents
Rayam, Parsharamulu, Polkam, Naveen, Kuntala, Naveen, Banothu, Venkanna, Anantaraju, Hasitha Shilpa, Perumal, Yogeeswari, Balasubramanian, Sridhar, Anireddy, Jaya Shree
Published in Journal of heterocyclic chemistry (01.03.2020)
Published in Journal of heterocyclic chemistry (01.03.2020)
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Journal Article
An atom efficient, solvent-free, green synthesis and antimycobacterial evaluation of 2-amino-6-methyl-4-aryl-8-[(E)-arylmethylidene]-5,6,7,8 -tetrahydro -4H -pyrano [3,2 -c ]pyridine -3 -carbonitriles
RAJU RANJITH KUMAR, PERUMAL, Subbu, SENTHILKUMAR, Palaniappan, YOGEESWARI, Perumal, SRIRAM, Dharmarajan
Published in Bioorganic & medicinal chemistry (01.12.2007)
Published in Bioorganic & medicinal chemistry (01.12.2007)
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Journal Article
Antimycobacterial activity of spirooxindolo-pyrrolidine, pyrrolizine and pyrrolothiazole hybrids obtained by a three-component regio- and stereoselective 1,3-dipolar cycloaddition
Rajesh, Stephen Michael, Perumal, Subbu, Menéndez, J. Carlos, Yogeeswari, Perumal, Sriram, Dharmarajan
Published in MedChemComm (01.07.2011)
Published in MedChemComm (01.07.2011)
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Journal Article
Depletion of M. tuberculosis GlmU from Infected Murine Lungs Effects the Clearance of the Pathogen
Soni, Vijay, Upadhayay, Sandeep, Suryadevara, Priyanka, Samla, Ganesh, Singh, Archana, Yogeeswari, Perumal, Sriram, Dharmarajan, Nandicoori, Vinay Kumar
Published in PLoS pathogens (01.10.2015)
Published in PLoS pathogens (01.10.2015)
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Journal Article
Design and synthesis of anticonvulsants from a combined phthalimide–GABA–anilide and hydrazone pharmacophore
Ragavendran, Jegadeesan Vaigunda, Sriram, Dharmarajan, Patel, Sravan Kumar, Reddy, Ingala Vikram, Bharathwajan, Narayanan, Stables, James, Yogeeswari, Perumal
Published in European journal of medicinal chemistry (01.02.2007)
Published in European journal of medicinal chemistry (01.02.2007)
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Journal Article
A highly atom economic, chemo-, regio- and stereoselective synthesis and evaluation of spiro-pyrrolothiazoles as antitubercular agents
Karthikeyan, Subramanian Vedhanarayanan, Bala, Balasubramanian Devi, Raja, Velanganni Paul Alex, Perumal, Subbu, Yogeeswari, Perumal, Sriram, Dharmarajan
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Journal Article
Synthesis and antitubercular evaluation of novel dibenzo[b,d]thiophene tethered imidazo[1,2-a]pyridine-3-carboxamides
Pulipati, Lokesh, Sridevi, Jonnalagadda Padma, Yogeeswari, Perumal, Sriram, Dharmarajan, Kantevari, Srinivas
Published in Bioorganic & medicinal chemistry letters (01.07.2016)
Published in Bioorganic & medicinal chemistry letters (01.07.2016)
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Journal Article
Isonicotinic acid hydrazide derivatives: synthesis, antimicrobial activity, and QSAR studies
Judge, Vikramjeet, Narasimhan, Balasubramanian, Ahuja, Munish, Sriram, Dharmarajan, Yogeeswari, Perumal, De Clercq, Erik, Pannecouque, Christophe, Balzarini, Jan
Published in Medicinal chemistry research (01.07.2012)
Published in Medicinal chemistry research (01.07.2012)
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Journal Article
Rational design, synthesis and evaluation of novel-substituted 1,2,3-triazolylmethyl carbazoles as potent inhibitors of Mycobacterium tuberculosis
Surineni, Goverdhan, Yogeeswari, Perumal, Sriram, Dharmarajan, Kantevari, Srinivas
Published in Medicinal chemistry research (01.03.2015)
Published in Medicinal chemistry research (01.03.2015)
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Journal Article